IL70075D0 - Improvements in or relating to 3-aryl-5-pyrazole derivatives - Google Patents

Improvements in or relating to 3-aryl-5-pyrazole derivatives

Info

Publication number
IL70075D0
IL70075D0 IL7007583A IL7007583A IL70075D0 IL 70075 D0 IL70075 D0 IL 70075D0 IL 7007583 A IL7007583 A IL 7007583A IL 7007583 A IL7007583 A IL 7007583A IL 70075 D0 IL70075 D0 IL 70075D0
Authority
IL
Israel
Prior art keywords
aryl
relating
improvements
pyrazole derivatives
pyrazole
Prior art date
Application number
IL7007583A
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US06/437,994 priority Critical patent/US4495195A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of IL70075D0 publication Critical patent/IL70075D0/en

Links

IL7007583A 1982-11-01 1983-10-27 Improvements in or relating to 3-aryl-5-pyrazole derivatives IL70075D0 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
US06/437,994 US4495195A (en) 1982-11-01 1982-11-01 Xanthine oxidase inhibiting 3(5)-phenyl-substituted-5(3)-pyrazole-carboxylic acid derivatives, compositions, and methods of use

Publications (1)

Publication Number Publication Date
IL70075D0 true IL70075D0 (en) 1984-01-31

Family

ID=23738785

Family Applications (1)

Application Number Title Priority Date Filing Date
IL7007583A IL70075D0 (en) 1982-11-01 1983-10-27 Improvements in or relating to 3-aryl-5-pyrazole derivatives

Country Status (13)

Country Link
US (1) US4495195A (en)
EP (1) EP0112623A2 (en)
JP (1) JPS5995272A (en)
KR (1) KR840006629A (en)
AU (1) AU2068583A (en)
DD (1) DD210265A5 (en)
DK (1) DK492783D0 (en)
ES (1) ES8601900A1 (en)
FI (1) FI833931A (en)
GB (1) GB2130205A (en)
GR (1) GR79640B (en)
IL (1) IL70075D0 (en)
PT (1) PT77583B (en)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ208555A (en) * 1983-06-23 1987-06-30 American Cyanamid Co (3-amino-1h-pyrazol-4-yl)-arylmethanone derivatives
IE59813B1 (en) * 1986-05-09 1994-04-06 Warner Lambert Co Styryl pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxy-genase inhibitors and pharmaceutical compositions containing them
JPH0551582B2 (en) 1987-04-24 1993-08-03 Mitsubishi Chem Ind
US4861777A (en) * 1987-09-11 1989-08-29 Mitsubishi Kasei Corporation Pyrazole derivative and insecticidal and miticidal composition containing the derivative as active ingredient
JP2751309B2 (en) * 1988-02-16 1998-05-18 三菱化学株式会社 Pyrazoles and insecticides that it as an active ingredient, acaricidal, fungicides
JP2784925B2 (en) * 1988-09-07 1998-08-13 日本農薬株式会社 3 or 5-phenyl-pyrazoles or a salt thereof and the herbicide
CA2036192A1 (en) 1990-02-13 1991-08-14 Nicholas Meanwell Heterocyclic carboxylic acids and esters
US4956379A (en) * 1990-02-13 1990-09-11 Bristol-Myers Squibb Company Pyrazole carboxylic acids and esters and inhibition of blood platelet aggregation therewith
FR2665898B1 (en) * 1990-08-20 1994-03-11 Sanofi Amide derivatives of 3-pyrazole, process for their preparation and pharmaceutical compositions containing them.
US5294630A (en) * 1992-07-07 1994-03-15 Eli Lilly And Company Treatment of inflammatory bowel disease
US5436258A (en) * 1992-09-09 1995-07-25 Eli Lilly And Company Prevention of bone resorption
GB9312853D0 (en) * 1993-06-22 1993-08-04 Euro Celtique Sa Chemical compounds
US5591776A (en) * 1994-06-24 1997-01-07 Euro-Celtique, S.A. Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV
HRP950330A2 (en) * 1994-07-05 1997-10-31 Ciba Geigy Ag New herbicides
US6166041A (en) * 1995-10-11 2000-12-26 Euro-Celtique, S.A. 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
EP0814809B1 (en) * 1994-12-13 2003-08-13 Euroceltique S.A. Aryl thioxanthines
AT247655T (en) * 1994-12-13 2003-09-15 Euro Celtique Sa Triple Substituted thioxanthines
US6025361A (en) * 1994-12-13 2000-02-15 Euro-Celtique, S.A. Trisubstituted thioxanthines
US6075016A (en) * 1996-04-10 2000-06-13 Euro-Celtique S.A. 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
ID21775A (en) * 1996-10-25 1999-07-22 Yoshitomi Pharmaceutical The compounds 1-fenilpirazol and use of its pharmaceutical
US5723608A (en) * 1996-12-31 1998-03-03 Neurogen Corporation 3-aryl substituted pyrazolo 4,3-d!pyrimidine derivatives; corticotropin-releasing factor receptor (CRF1) specific ligands
EP1044002A4 (en) * 1997-11-07 2003-05-02 Univ Johns Hopkins Methods for treatment of disorders of cardiac contractility
US7820700B2 (en) * 2004-08-27 2010-10-26 Astellas Pharma Inc. 2-phenylpyridine derivative
JPWO2006022375A1 (en) * 2004-08-27 2008-05-08 アステラス製薬株式会社 2-phenyl thiophene derivatives
RU2008118156A (en) 2005-10-07 2009-11-20 Астеллас Фарма Инк. (Jp) Acid derivative triarilkarbonovoy
AT555810T (en) 2006-02-24 2012-05-15 Astellas Pharma Inc Means for treatment or prevention of peptic ulcers
KR101639834B1 (en) 2009-02-27 2016-07-14 데이진 화-마 가부시키가이샤 Process for producing phenyl-substituted heterocyclic derivative through coupling using transition metal catalyst
WO2012026565A1 (en) 2010-08-27 2012-03-01 帝人ファーマ株式会社 Method for producing phenyl-substituted heterocyclic derivative by means of coupling method using a palladium compound
EP2980085B1 (en) 2013-03-29 2018-03-14 Teijin Pharma Limited Pyrazole derivative
EP2944635B1 (en) * 2014-05-15 2018-11-28 Council of Scientific & Industrial Research Pyrazole linked benzimidazole conjugates and a process for preparation thereof

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1261124B (en) * 1961-09-22 1968-02-15 Hoechst Ag A process for the preparation of pyrazoles
IT1053661B (en) * 1966-09-27 1981-10-10 Farmacosmici S P A Acid amides of methyl 3 5 5 3 pyrazol carboxylic acid
FR2104931B1 (en) * 1970-09-08 1975-01-10 Ferlux
DE2508934A1 (en) * 1974-03-04 1975-09-11 Byk Gulden Lomberg Chem Fab Xanthinoxidase-inhibiotory 5-amino-4-formylcarbamoyl pyrrazoles - prepd. from N'-(2-cyano-3-formylamino-hydroxy-allylidene)nicotinic hydrazide
DE2410653A1 (en) * 1974-03-06 1975-10-30 Byk Gulden Lomberg Chem Fab 5-Amino-5-(N-formyl-carbamoyl)-pyrazole derivs - prepd. by cyclizing N-formyl-alpha-(acylhydrazinomethylene)-cyanoacetamides
US3895027A (en) * 1974-04-12 1975-07-15 Lilly Co Eli Process for preparing pyrazole-3-carboxylic acids
US3903106A (en) * 1974-04-12 1975-09-02 Lilly Co Eli Pyrazole-3-carboxylic acids
US3899508A (en) * 1974-04-12 1975-08-12 Lilly Co Eli 5-(2-Aminophenyl)pyrazole-3-carboxylic acids and esters thereof
FR2353292B1 (en) * 1975-08-05 1978-12-15 Sogeras
FR2320093B1 (en) * 1975-08-05 1979-09-14 Sogeras
US4134987A (en) * 1976-01-14 1979-01-16 Huppatz John L Compounds and compositions
US4214090A (en) * 1976-01-14 1980-07-22 Commonwealth Scientific And Industrial Research Organization Fungicidal carboxamidopyrazoles
US4245106A (en) * 1979-07-05 1981-01-13 Monsanto Company Process for the preparation of 1-alkyl-3-aryl-4-pyrazolecarboxylates
US4346097A (en) * 1980-09-30 1982-08-24 Warner-Lambert Company Method for treating convulsions with pyrazole-4-carboxamide derivatives

Also Published As

Publication number Publication date
ES8601900A1 (en) 1985-05-01
JPS5995272A (en) 1984-06-01
FI833931D0 (en)
PT77583B (en) 1986-05-27
GB8328755D0 (en) 1983-11-30
DD210265A5 (en) 1984-06-06
DK492783D0 (en) 1983-10-27
PT77583A (en) 1983-11-01
FI833931A0 (en) 1983-10-27
KR840006629A (en) 1984-12-01
EP0112623A2 (en) 1984-07-04
ES526869A0 (en) 1985-05-01
ES526869D0 (en)
US4495195A (en) 1985-01-22
GR79640B (en) 1984-10-31
FI833931A (en) 1984-05-02
GB2130205A (en) 1984-05-31
AU2068583A (en) 1984-05-10

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