IL309708B2 - Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one - Google Patents

Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one

Info

Publication number
IL309708B2
IL309708B2 IL309708A IL30970823A IL309708B2 IL 309708 B2 IL309708 B2 IL 309708B2 IL 309708 A IL309708 A IL 309708A IL 30970823 A IL30970823 A IL 30970823A IL 309708 B2 IL309708 B2 IL 309708B2
Authority
IL
Israel
Prior art keywords
composition
mixture
solution
plant
crystalline
Prior art date
Application number
IL309708A
Other languages
English (en)
Hebrew (he)
Other versions
IL309708A (en
IL309708B1 (en
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of IL309708A publication Critical patent/IL309708A/en
Publication of IL309708B1 publication Critical patent/IL309708B1/en
Publication of IL309708B2 publication Critical patent/IL309708B2/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL309708A 2017-07-17 2018-07-16 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one IL309708B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201762533509P 2017-07-17 2017-07-17
PCT/IB2018/000875 WO2019038583A1 (en) 2017-07-17 2018-07-16 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2-ONE POLYMORPHS

Publications (3)

Publication Number Publication Date
IL309708A IL309708A (en) 2024-02-01
IL309708B1 IL309708B1 (en) 2025-10-01
IL309708B2 true IL309708B2 (en) 2026-02-01

Family

ID=63517924

Family Applications (5)

Application Number Title Priority Date Filing Date
IL309708A IL309708B2 (en) 2017-07-17 2018-07-16 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
IL271950A IL271950B2 (en) 2017-07-17 2018-07-16 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
IL323268A IL323268A (en) 2017-07-17 2025-09-10 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
IL323266A IL323266A (en) 2017-07-17 2025-09-10 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
IL323267A IL323267A (en) 2017-07-17 2025-09-10 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one

Family Applications After (4)

Application Number Title Priority Date Filing Date
IL271950A IL271950B2 (en) 2017-07-17 2018-07-16 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
IL323268A IL323268A (en) 2017-07-17 2025-09-10 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
IL323266A IL323266A (en) 2017-07-17 2025-09-10 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
IL323267A IL323267A (en) 2017-07-17 2025-09-10 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one

Country Status (11)

Country Link
US (1) US11632954B2 (https=)
EP (1) EP3655396A1 (https=)
JP (3) JP2020527563A (https=)
CN (2) CN118515619A (https=)
AR (1) AR112276A1 (https=)
AU (1) AU2018320492C1 (https=)
CA (1) CA3069619A1 (https=)
IL (5) IL309708B2 (https=)
MA (1) MA49639A (https=)
WO (1) WO2019038583A1 (https=)
ZA (1) ZA202000411B (https=)

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EP3876717A1 (en) 2018-11-05 2021-09-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
IL321760A (en) * 2019-07-22 2025-08-01 Adama Makhteshim Ltd Fungicidal combinations, mixtures and compositions and uses thereof
PY2057637A (es) * 2019-09-23 2021-10-05 Adama Makhteshim Ltd Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto
EP4146632A1 (en) * 2020-05-04 2023-03-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
BR112023014997A2 (pt) 2021-01-27 2023-10-03 Adama Makhteshim Ltd 5-fluoro-4-imino-3-metil-1-tosil-3,4-di-hidropirimidin-2(1h)-ona para controle de doenças de plantas
US20240237649A1 (en) 2021-05-04 2024-07-18 Adama Makhteshim Ltd. Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
UY40172A (es) 2022-03-03 2023-10-13 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
EP4609713A3 (en) 2022-05-26 2025-10-29 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AU2023318916A1 (en) 2022-08-03 2025-02-20 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1h)-one for fungicide-resistant fungus
AU2024233301A1 (en) 2023-03-09 2025-09-18 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AU2024236967A1 (en) 2023-03-14 2025-09-25 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
AR132381A1 (es) 2023-04-11 2025-06-18 Adama Makhteshim Ltd Compuestos y procesos relativos a flumetilsulforim
WO2025046581A1 (en) 2023-08-31 2025-03-06 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereo
PY24105707A (es) 2023-11-28 2025-06-25 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
WO2026038217A1 (en) 2024-08-15 2026-02-19 Adama Makhteshim Ltd. Mixtures and compositions comprising flumetylsulforim and methods of use thereof

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Also Published As

Publication number Publication date
IL271950B1 (en) 2024-02-01
ZA202000411B (en) 2023-10-25
US11632954B2 (en) 2023-04-25
BR112020000953A2 (pt) 2020-07-14
JP2020527563A (ja) 2020-09-10
IL309708A (en) 2024-02-01
WO2019038583A1 (en) 2019-02-28
AR112276A1 (es) 2019-10-09
IL323268A (en) 2025-11-01
EP3655396A1 (en) 2020-05-27
IL323266A (en) 2025-11-01
CN111094252A (zh) 2020-05-01
IL309708B1 (en) 2025-10-01
AU2018320492B2 (en) 2022-12-01
JP2023145572A (ja) 2023-10-11
CN118515619A (zh) 2024-08-20
IL271950A (en) 2020-02-27
AU2018320492A1 (en) 2020-02-13
CA3069619A1 (en) 2019-02-28
NZ761039A (en) 2023-09-29
US20200229437A1 (en) 2020-07-23
MA49639A (fr) 2020-05-27
AU2018320492C1 (en) 2023-07-13
CN111094252B (zh) 2024-05-24
JP2025163080A (ja) 2025-10-28
IL271950B2 (en) 2024-06-01
IL323267A (en) 2025-11-01

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