IL107289A - METHYL a(o-SUBSTITUTED PHENYL)-b-METHOXY- ACRYLATE DERIVATIVES, THEIR PREPARATION AND FUNGICIDAL COMPOSITIONS CONTAINING THEM - Google Patents

METHYL a(o-SUBSTITUTED PHENYL)-b-METHOXY- ACRYLATE DERIVATIVES, THEIR PREPARATION AND FUNGICIDAL COMPOSITIONS CONTAINING THEM

Info

Publication number
IL107289A
IL107289A IL107289A IL10728988A IL107289A IL 107289 A IL107289 A IL 107289A IL 107289 A IL107289 A IL 107289A IL 10728988 A IL10728988 A IL 10728988A IL 107289 A IL107289 A IL 107289A
Authority
IL
Israel
Prior art keywords
alkyl
phenyl
alkoxy
alkenyl
hydroxy
Prior art date
Application number
IL107289A
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to GB878702845A priority Critical patent/GB8702845D0/en
Priority to GB878710594A priority patent/GB8710594D0/en
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Priority to IL8512288A priority patent/IL85122A/en
Publication of IL107289A publication Critical patent/IL107289A/en

Links

Abstract

Compounds of the formula R1YR2C R3X11 CCH302c CH.OR6 and stereoisomers thereof, wherein R1 is an aryl moiety which is optionally substituted by one or more of: halogen, hydroxy, C1-4 alkyl, C2-4 alkenyl, C2-4 alkynyl, C1-4 alkoxy, C2-4 alkenyloxy, C2-4 alkynyloxy, halo (C1-4) alkyl, halo (C1-4) alkoxy, C1-4 alkylthio, hydroxy (C1-4) alkyl, (C1-4) alkoxy (C1-4) alkyl, C3-6 cycloalkyl, C3-6 cycloalkyl (C1-4) alkyl, phenyl, heteroaryl, phenoxy, heteroaryloxy, phenyl (C1-4) alkyl in which the alkyl moiety is optionally substituted with hydroxy, heteroaryl (C1-4) alkyl, phenyl (C2-4) alkenyl, heteroraryl (C2-4) alkenyl, phenyl (C1-4) alkoxy, heteroaryl (C1-4) alkoxy, phenoxy (C1-4) alkyl, heteroaryloxy (C1-4) alkyl, (C1-4) alkylcarbonyloxy, benzoyloxy, cyano, thiocyanato, nitro, -NR:R", -NHCOR:, -NHCONR:R", -CONR:R", -COOR:, -OSO2R:, -SO2R:, -COR:, -CR: =NR" or -N=CR:R"; or substituents on the aryl moiety of R1, when they are in adjacent positions, may join to form a methylenedioxy group or may join together with R1 to form a dibenzo-p-dioxinyl, dibenzofuranyl or dibenzothienyl fused ring system; phenyl or heteroaryl moieties comprised in any of the foregoing substituents are optionally substituted by one or more of: halogen, hydroxy, C1-4 alkyl, C2-4 alkenyl, C2-4 alkynyl, C1-4 alkoxy, C2-4 alkenyloxy, C2-4 alkynyloxy, halo (C1-4) alkyl, halo (C1-4) alkoxy, C1-4 alkylthio, hydroxy (C1-4) alkyl, (C1-4) alkoxy (C1-4) alkyl, C3-6 cycloalkyl, C3-6 cycloalkyl (C1-4) alkyl, phenyl, heteroaryl, phenoxy, heteroaryloxy, phenyl (C1-4) alkyl in which the alkyl moiety is optionally substituted with hydroxy, heteroaryl (C1-4) alkyl, phenyl (C2-4) alkenyl, heteroaryl (C2-4) alkenyl, phenyl (C1-4) alkoxy, heteroaryl (C1-4) alkoxy, phenoxy (C1-4) alkyl, heteroaryloxy (C1-4) alkyl, C1-4 alkylcarbonyloxy, benzoyloxy, cyano, thiocyanato, nitro, -NR:R", -NHCOR:, -NHCONR:R", -CONR:R", -COOR:, -OSO2R:, -SO2R:, -COR:, -CR:=NR" or -N=CR:R", wherein phenyl or heteroaryl moieties comprised in any of these substituents are optionally substituted by one or more of: halogen, hydroxy, C1-4 alkyl, C2-4 alkenyl, C2-4 alkynyl, C1-4 alkoxy, C2-4 alkenyloxy, C2-4 alkynyloxy, halo (C1-4) alkyl, halo (C1-4) alkoxy, C1-4 alkylthio, hydroxy (C1-4) alkyl, (C1-4) alkoxy (C1-4) alkyl, C3-6 cycloalkyl, C3-6 cycloalkyl (C1-4) alkyl, C1-4 alkylcarbonyloxy, cyano, thiocyanato, nitro, -NR:R", -NHCOR:, -NHCONR:R", -CONR:R", -COOR:, -OSO2R:, -SO2R:, -COR:, -CR:=NR" or -N=CR:R"; R: and R" are independently hydrogen, C1-4 alkyl, C1-4 alkoxy (other than R: in -COR:), C1-4 alkylthio, C3-6 cycloalkyl, C3-6 cycloalkyl (C1-4) alkyl, phenyl or phenyl (C1-4) alkyl, the phenyl or phenyl (C1-4) alkyl groups being optionally substituted with halogen, C1-4 alkyl or C1-4 alkoxy; aryl is phenyl or naphthyl; the heteroaryl moieties are, independently, pyridinyl, pyrimidinyl, pyrazinyl, pyridazinyl, 1, 2, 3-, 1, 2, 4- or 1, 3, 5-triazinyl, 1, 2, 4, 5-tetrazinyl, thienyl, quinolinyl, isoquinolinyl, quinoxalinyl or benzothienyl; Y is oxygen, sulphur or NR4; R2, R3 and R4, which may be the same or different, are hydrogen, C1-4 alkyl or C2-4 alkenyl; X is halogen, C1-4 alkyl, C2-4 alkenyl, C1-4 alkoxy, nitro or cyano; n is 0 or an integer of 1 to 4; and R6 is methyl, hydrogen, sodium or potassium; provided that when Y is oxygen, R2 and R3 are independently hydrogen or alkyl, n is 0, 1 or 2 and R6 is methyl, the R1 is not phenyl optionally substituted with one or more of halogen, hydroxy, C1-4 alkyl, C1-4 alkoxy (itself substituted with halogen), phenyl, phenoxy, nitro, cyano, amino, mono-or di- (C1-4) alkylamino, C1-4 alkanoylamino, benzoylamino, carboxy or C1-4 alkoxycarbonyl.
IL107289A 1987-02-09 1988-01-19 METHYL a(o-SUBSTITUTED PHENYL)-b-METHOXY- ACRYLATE DERIVATIVES, THEIR PREPARATION AND FUNGICIDAL COMPOSITIONS CONTAINING THEM IL107289A (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
GB878702845A GB8702845D0 (en) 1987-02-09 1987-02-09 Fungicides
GB878710594A GB8710594D0 (en) 1987-05-05 1987-05-05 Fungicides
IL8512288A IL85122A (en) 1987-02-09 1988-01-19 Methyl 2-(2-(1-substituted alk(en)yl) phenyl)-3-methoxypropenoate derivatives, their preparation and fungicidal compositions containing them

Publications (1)

Publication Number Publication Date
IL107289A true IL107289A (en) 1997-06-10

Family

ID=27263311

Family Applications (5)

Application Number Title Priority Date Filing Date
IL9874288A IL98742A (en) 1987-02-09 1988-01-19 Methyl-2-(substituted methyl)-alpha-(dimethoxymethyl)-benzeneacetate
IL98741A IL98741A (en) 1987-02-09 1988-01-19 Methyl 3-methoxy-2- ((2-chloromethyl or formyl) phenyl) acrylates
IL107289A IL107289A (en) 1987-02-09 1988-01-19 METHYL a(o-SUBSTITUTED PHENYL)-b-METHOXY- ACRYLATE DERIVATIVES, THEIR PREPARATION AND FUNGICIDAL COMPOSITIONS CONTAINING THEM
IL9874388A IL98743A (en) 1987-02-09 1988-01-19 Methyl 2-(substituted methyl)-alpha-oxobenzeneacetate intermediates for fungicides
IL107289A IL107289D0 (en) 1987-02-09 1993-10-14 Methyl a-phenylacrylate derivatives, their preparation and fungicidal compositions containing them

Family Applications Before (2)

Application Number Title Priority Date Filing Date
IL9874288A IL98742A (en) 1987-02-09 1988-01-19 Methyl-2-(substituted methyl)-alpha-(dimethoxymethyl)-benzeneacetate
IL98741A IL98741A (en) 1987-02-09 1988-01-19 Methyl 3-methoxy-2- ((2-chloromethyl or formyl) phenyl) acrylates

Family Applications After (2)

Application Number Title Priority Date Filing Date
IL9874388A IL98743A (en) 1987-02-09 1988-01-19 Methyl 2-(substituted methyl)-alpha-oxobenzeneacetate intermediates for fungicides
IL107289A IL107289D0 (en) 1987-02-09 1993-10-14 Methyl a-phenylacrylate derivatives, their preparation and fungicidal compositions containing them

Country Status (1)

Country Link
IL (5) IL98742A (en)

Also Published As

Publication number Publication date
IL98743A (en) 1996-10-16
IL107289D0 (en) 1994-01-25
IL98741A (en) 1993-03-15
IL98742A (en) 1996-06-18

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