HU217346B - Process for producing amlodipin-bezilate - Google Patents

Process for producing amlodipin-bezilate

Info

Publication number
HU217346B
HU217346B HU9402708A HU9402708A HU217346B HU 217346 B HU217346 B HU 217346B HU 9402708 A HU9402708 A HU 9402708A HU 9402708 A HU9402708 A HU 9402708A HU 217346 B HU217346 B HU 217346B
Authority
HU
Hungary
Prior art keywords
bezilate
amlodipin
producing
formula
present
Prior art date
Application number
HU9402708A
Other languages
Hungarian (hu)
Other versions
HU9402708D0 (en
Inventor
János Fischer
Katalin Szőke
László Dobay
Sándor Lévai
Original Assignee
Richter Gedeon Vegyészeti Gyár Rt.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyészeti Gyár Rt. filed Critical Richter Gedeon Vegyészeti Gyár Rt.
Priority to HU9402708A priority Critical patent/HU217346B/en
Publication of HU9402708D0 publication Critical patent/HU9402708D0/en
Publication of HU217346B publication Critical patent/HU217346B/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

A találmány tárgya új eljárás (I) képletű amlődipin-bezilátelőállítására, őly módőn, hőgy (II) képletű 4-(2-klór-fenil)-3-(etőxi-karbőnil)-5-(metőxi-karbőnil)-2-[2- (2- karbőxi-benzőil-aminő)-etőxi-metil]-6-metil-1,4-di- hidrőpiridin származékőt vagy sójátsztöchiőmetrikűs mennyiségű benzőlszűlfőnsavval reagáltatják. Atalálmány szerinti eljárással előállítőtt (I) képletű vegyületszívbetegségek és magas vérnyőmás ellen alkalmazőtt gyógyszerhatóanyaga. ŕThe present invention relates to a novel process for the production of amylipipine-bezylate of formula (I), preferably 4- (2-chlorophenyl) -3- (ethyloxycarbonyl) -5- (methoxycarbonyl) -2- [ The 2- (2-carboxybenzylamino) -etxymethyl] -6-methyl-1,4-dihydro-pyridine derivative is reacted with a salt of petroleum filtrate in the form of a salt solution. In accordance with the method of the present invention, there is provided a pharmaceutical agent for the use of the compounds of formula (I) for the treatment of heart disease and hypertension. ŕ

HU9402708A 1994-09-20 1994-09-20 Process for producing amlodipin-bezilate HU217346B (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
HU9402708A HU217346B (en) 1994-09-20 1994-09-20 Process for producing amlodipin-bezilate

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU9402708A HU217346B (en) 1994-09-20 1994-09-20 Process for producing amlodipin-bezilate

Publications (2)

Publication Number Publication Date
HU9402708D0 HU9402708D0 (en) 1994-12-28
HU217346B true HU217346B (en) 2000-01-28

Family

ID=10985606

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9402708A HU217346B (en) 1994-09-20 1994-09-20 Process for producing amlodipin-bezilate

Country Status (1)

Country Link
HU (1) HU217346B (en)

Also Published As

Publication number Publication date
HU9402708D0 (en) 1994-12-28

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Owner name: RICHTER GEDEON NYRT., HU

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