GB1580402A - Processes for the manufacture of steroid carboxylic acids and the esters thereof - Google Patents

Processes for the manufacture of steroid carboxylic acids and the esters thereof Download PDF

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Publication number
GB1580402A
GB1580402A GB15779/77A GB1577977A GB1580402A GB 1580402 A GB1580402 A GB 1580402A GB 15779/77 A GB15779/77 A GB 15779/77A GB 1577977 A GB1577977 A GB 1577977A GB 1580402 A GB1580402 A GB 1580402A
Authority
GB
United Kingdom
Prior art keywords
process according
hydroxyl group
acid
starting materials
carboxylic acids
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB15779/77A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of GB1580402A publication Critical patent/GB1580402A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J3/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0033Androstane derivatives substituted in position 17 alfa and 17 beta
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008Expansion of ring D by one atom, e.g. D homo steroids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J7/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C07J7/008Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21
    • C07J7/009Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21 by only one oxygen atom doubly bound
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • C07J71/0026Oxygen-containing hetero ring cyclic ketals
    • C07J71/0031Oxygen-containing hetero ring cyclic ketals at positions 16, 17

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
GB15779/77A 1976-04-15 1977-04-15 Processes for the manufacture of steroid carboxylic acids and the esters thereof Expired GB1580402A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH484876A CH614960A5 (US20040152965A1-20040805-M00009.png) 1976-04-15 1976-04-15

Publications (1)

Publication Number Publication Date
GB1580402A true GB1580402A (en) 1980-12-03

Family

ID=4283605

Family Applications (1)

Application Number Title Priority Date Filing Date
GB15779/77A Expired GB1580402A (en) 1976-04-15 1977-04-15 Processes for the manufacture of steroid carboxylic acids and the esters thereof

Country Status (9)

Country Link
US (1) US4119625A (US20040152965A1-20040805-M00009.png)
JP (1) JPS52128363A (US20040152965A1-20040805-M00009.png)
CA (1) CA1091223A (US20040152965A1-20040805-M00009.png)
CH (1) CH614960A5 (US20040152965A1-20040805-M00009.png)
DE (1) DE2715863A1 (US20040152965A1-20040805-M00009.png)
FR (1) FR2348226A1 (US20040152965A1-20040805-M00009.png)
GB (1) GB1580402A (US20040152965A1-20040805-M00009.png)
IL (1) IL51879A (US20040152965A1-20040805-M00009.png)
NL (1) NL7704105A (US20040152965A1-20040805-M00009.png)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7275462B2 (en) 2002-06-20 2007-10-02 Aktiebolaget Skf Tensioning device for prestressing a rod, and related tensioning method
US7429133B2 (en) 2002-07-02 2008-09-30 Aktiebolaget Skf Instrumented antifriction bearing and electrical motor equipped therewith

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4198336A (en) * 1978-04-05 1980-04-15 Syntex (U.S.A.) Inc. Chemical process for preparing androsta-4-ene 17α-carboxylic acids
DE3024008C2 (de) * 1980-06-24 1982-04-15 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 17α-Hydroxy-etiocarbonsäuren
SE8306370D0 (sv) * 1983-11-18 1983-11-18 Draco Ab Novel androstane-17beta-carboxylic acid esters, a process and intermediates for their preparation, compositions and method for the treatment of inflammatory conditions
EP1848897A1 (fr) * 2005-02-15 2007-10-31 Aktiebolaget SKF (publ) Dispositif de roulement codeur et machine tournante
FR2902699B1 (fr) * 2006-06-26 2010-10-22 Skf Ab Dispositif de butee de suspension et jambe de force.
FR2906587B1 (fr) * 2006-10-03 2009-07-10 Skf Ab Dispositif de galet tendeur.
FR2906858B1 (fr) * 2006-10-04 2008-12-05 Skf Ab Dispositif de poulie debrayable.
FR2910129B1 (fr) * 2006-12-15 2009-07-10 Skf Ab Dispositif de palier a roulement instrumente
FR2913081B1 (fr) * 2007-02-27 2009-05-15 Skf Ab Dispositif de poulie debrayable

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3636010A (en) * 1968-12-23 1972-01-18 Ciba Geigy Corp Esters of steroid-17-carboxylic acids
DE2260303C2 (de) * 1972-12-06 1983-12-15 Schering AG, 1000 Berlin und 4709 Bergkamen Verfahren zur Herstellung von Pregnansäurederivaten
GB1514476A (en) * 1974-08-30 1978-06-14 Glaxo Lab Ltd Alkyl and haloalkyl androst-4-ene and androsta-1,4-diene-17beta-carboxylates

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7275462B2 (en) 2002-06-20 2007-10-02 Aktiebolaget Skf Tensioning device for prestressing a rod, and related tensioning method
US7429133B2 (en) 2002-07-02 2008-09-30 Aktiebolaget Skf Instrumented antifriction bearing and electrical motor equipped therewith

Also Published As

Publication number Publication date
NL7704105A (nl) 1977-10-18
DE2715863A1 (de) 1977-11-03
US4119625A (en) 1978-10-10
CH614960A5 (US20040152965A1-20040805-M00009.png) 1979-12-28
FR2348226A1 (fr) 1977-11-10
FR2348226B1 (US20040152965A1-20040805-M00009.png) 1980-07-04
CA1091223A (en) 1980-12-09
JPS52128363A (en) 1977-10-27
IL51879A0 (en) 1977-06-30
IL51879A (en) 1981-06-29

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Legal Events

Date Code Title Description
PS Patent sealed [section 19, patents act 1949]
PCNP Patent ceased through non-payment of renewal fee