GB1416281A - N-benzene-sulphonyl-erythromycylamine derivatives - Google Patents
N-benzene-sulphonyl-erythromycylamine derivativesInfo
- Publication number
- GB1416281A GB1416281A GB224274A GB224274A GB1416281A GB 1416281 A GB1416281 A GB 1416281A GB 224274 A GB224274 A GB 224274A GB 224274 A GB224274 A GB 224274A GB 1416281 A GB1416281 A GB 1416281A
- Authority
- GB
- United Kingdom
- Prior art keywords
- sulphonyl
- benzene
- jan
- erythromycylamine
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- IEDVJHCEMCRBQM-UHFFFAOYSA-N trimethoprim Chemical compound COC1=C(OC)C(OC)=CC(CC=2C(=NC(N)=NC=2)N)=C1 IEDVJHCEMCRBQM-UHFFFAOYSA-N 0.000 abstract 2
- XCLJRCAJSCMIND-JCTYMORFSA-N (9S)-erythromycyclamine Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)[C@@H](N)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 XCLJRCAJSCMIND-JCTYMORFSA-N 0.000 abstract 1
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 229940088710 antibiotic agent Drugs 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- QZIQJVCYUQZDIR-UHFFFAOYSA-N mechlorethamine hydrochloride Chemical compound Cl.ClCCN(C)CCCl QZIQJVCYUQZDIR-UHFFFAOYSA-N 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
- 229960001082 trimethoprim Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
1416281 Medicines comprising antibiotics PLIVA PHARMACEUTICAL & CHEMICAL WORKS 17 Jan 1974 [19 Jan 1973] 2242/74 Heading A5B [Also in Division C2] Erythromycylamine derivatives of the general formula wherein R is a C 1-5 alkyl group, a halogen atom or a -NHCOR' group, in which R' is a C 1-3 alkyl or phenyl group, having antibiotic activity, exhibit synergism when used in combination with trimethoprim(2, 4-diamino-5-(3', 4', 5'-trimethoxybenzyl)pyrimidine).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| YU15173A YU35369B (en) | 1973-01-19 | 1973-01-19 | Process for preparing n-(benzenesulfonyl)-erythromycilamine derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1416281A true GB1416281A (en) | 1975-12-03 |
Family
ID=25548575
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB224274A Expired GB1416281A (en) | 1973-01-19 | 1974-01-17 | N-benzene-sulphonyl-erythromycylamine derivatives |
Country Status (5)
| Country | Link |
|---|---|
| AT (1) | AT327388B (en) |
| CA (1) | CA1014147A (en) |
| DE (1) | DE2402200C2 (en) |
| GB (1) | GB1416281A (en) |
| YU (1) | YU35369B (en) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006127252A1 (en) | 2005-05-24 | 2006-11-30 | Pfizer, Inc. | Motilide compounds |
| WO2008068593A2 (en) | 2006-12-05 | 2008-06-12 | Pfizer Inc. | Motilide polymorphs |
-
1973
- 1973-01-19 YU YU15173A patent/YU35369B/en unknown
-
1974
- 1974-01-15 AT AT29474A patent/AT327388B/en not_active IP Right Cessation
- 1974-01-17 GB GB224274A patent/GB1416281A/en not_active Expired
- 1974-01-17 DE DE19742402200 patent/DE2402200C2/en not_active Expired
- 1974-01-18 CA CA190,512A patent/CA1014147A/en not_active Expired
Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006127252A1 (en) | 2005-05-24 | 2006-11-30 | Pfizer, Inc. | Motilide compounds |
| US7582611B2 (en) | 2005-05-24 | 2009-09-01 | Pfizer Inc. | Motilide compounds |
| WO2008068593A2 (en) | 2006-12-05 | 2008-06-12 | Pfizer Inc. | Motilide polymorphs |
| US7872109B2 (en) | 2006-12-05 | 2011-01-18 | Licari Peter J | Motilide polymorphs |
| US8030282B2 (en) | 2006-12-05 | 2011-10-04 | Licari Peter J | Motilide polymorphs |
Also Published As
| Publication number | Publication date |
|---|---|
| ATA29474A (en) | 1975-04-15 |
| YU15173A (en) | 1980-06-30 |
| YU35369B (en) | 1980-12-31 |
| AT327388B (en) | 1976-01-26 |
| CA1014147A (en) | 1977-07-19 |
| DE2402200A1 (en) | 1974-07-25 |
| DE2402200C2 (en) | 1982-03-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed | ||
| PCNP | Patent ceased through non-payment of renewal fee |