GB1368233A - Penicillin 1-oxides - Google Patents
Penicillin 1-oxidesInfo
- Publication number
- GB1368233A GB1368233A GB5228570A GB5228570A GB1368233A GB 1368233 A GB1368233 A GB 1368233A GB 5228570 A GB5228570 A GB 5228570A GB 5228570 A GB5228570 A GB 5228570A GB 1368233 A GB1368233 A GB 1368233A
- Authority
- GB
- United Kingdom
- Prior art keywords
- group
- formula
- penicillin
- amino group
- oxides
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229930182555 Penicillin Natural products 0.000 title abstract 3
- JGSARLDLIJGVTE-MBNYWOFBSA-N Penicillin G Chemical compound N([C@H]1[C@H]2SC([C@@H](N2C1=O)C(O)=O)(C)C)C(=O)CC1=CC=CC=C1 JGSARLDLIJGVTE-MBNYWOFBSA-N 0.000 title abstract 3
- 229940049954 penicillin Drugs 0.000 title abstract 3
- QTBSBXVTEAMEQO-UHFFFAOYSA-N Acetic acid Chemical compound CC(O)=O QTBSBXVTEAMEQO-UHFFFAOYSA-N 0.000 abstract 6
- 125000003277 amino group Chemical group 0.000 abstract 4
- -1 azide salt Chemical class 0.000 abstract 3
- 238000006243 chemical reaction Methods 0.000 abstract 3
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000007062 hydrolysis Effects 0.000 abstract 2
- 238000006460 hydrolysis reaction Methods 0.000 abstract 2
- 230000008707 rearrangement Effects 0.000 abstract 2
- JWGZDJNUMPJRAP-BAFYGKSASA-N (5R)-2-isocyanato-4-thia-1-azabicyclo[3.2.0]heptan-7-one Chemical compound N(=C=O)C1CS[C@H]2N1C(C2)=O JWGZDJNUMPJRAP-BAFYGKSASA-N 0.000 abstract 1
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- ISWSIDIOOBJBQZ-UHFFFAOYSA-N Phenol Chemical compound OC1=CC=CC=C1 ISWSIDIOOBJBQZ-UHFFFAOYSA-N 0.000 abstract 1
- 230000002378 acidificating effect Effects 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 125000004442 acylamino group Chemical group 0.000 abstract 1
- 229910052783 alkali metal Inorganic materials 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 150000008064 anhydrides Chemical class 0.000 abstract 1
- 239000011260 aqueous acid Substances 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 238000006114 decarboxylation reaction Methods 0.000 abstract 1
- 239000000428 dust Substances 0.000 abstract 1
- 238000005886 esterification reaction Methods 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 238000007327 hydrogenolysis reaction Methods 0.000 abstract 1
- 230000003647 oxidation Effects 0.000 abstract 1
- 238000007254 oxidation reaction Methods 0.000 abstract 1
- OJMIONKXNSYLSR-UHFFFAOYSA-N phosphorous acid Chemical compound OP(O)O OJMIONKXNSYLSR-UHFFFAOYSA-N 0.000 abstract 1
- 229910052698 phosphorus Inorganic materials 0.000 abstract 1
- 239000011574 phosphorus Substances 0.000 abstract 1
- 238000006722 reduction reaction Methods 0.000 abstract 1
- JOYRKODLDBILNP-UHFFFAOYSA-N urethane group Chemical group NC(=O)OCC JOYRKODLDBILNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Cephalosporin Compounds (AREA)
Priority Applications (14)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB5228570A GB1368233A (en) | 1970-07-31 | 1970-11-03 | Penicillin 1-oxides |
| AU31843/71A AU467354B2 (en) | 1970-07-31 | 1971-07-30 | Penicillin i-oxides |
| ES393800A ES393800A1 (es) | 1970-07-31 | 1971-07-30 | Un procedimiento para la preparacion de penicilin-1-oxidos. |
| NL7110612A NL7110612A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1970-07-31 | 1971-07-30 | |
| CH1129471A CH592097A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1970-07-31 | 1971-07-30 | |
| DE19712138323 DE2138323A1 (de) | 1970-07-31 | 1971-07-30 | Chemische Verbindungen |
| BE770727A BE770727A (fr) | 1970-07-31 | 1971-07-30 | Nouveaux composes intermediaires pour la synthese de cephalosporines, penicillines et antibiotiques analogues |
| DE19712166022 DE2166022A1 (de) | 1970-07-31 | 1971-07-30 | Chemische Verbindungen. Ausscheidung aus: 2138323 |
| FR7128114A FR2104819B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1970-07-31 | 1971-07-30 | |
| AT571174*1A AT324566B (de) | 1970-07-31 | 1971-07-30 | Verfahren zur herstellung von neuen penicillin-1-oxiden |
| JP5788271A JPS554113B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1970-07-31 | 1971-07-30 | |
| AT281473A AT329073B (de) | 1970-07-31 | 1973-03-30 | Verfahren zur herstellung von neuen 4,7-diaza -2- thia-bicyclo (3.2.0) -hept-3-enderivaten |
| CH352876A CH591504A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1970-07-31 | 1976-03-22 | |
| CH551077A CH594679A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1970-07-31 | 1977-05-03 |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB3718970 | 1970-07-31 | ||
| GB5228570A GB1368233A (en) | 1970-07-31 | 1970-11-03 | Penicillin 1-oxides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1368233A true GB1368233A (en) | 1974-09-25 |
Family
ID=26263366
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB5228570A Expired GB1368233A (en) | 1970-07-31 | 1970-11-03 | Penicillin 1-oxides |
Country Status (10)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4115383A (en) | 1976-02-23 | 1978-09-19 | Eli Lilly And Company | Alkoxycarbonyl-ethylthio-azetidinones and process for their preparation |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4036846A (en) * | 1976-04-26 | 1977-07-19 | Pfizer Inc. | 3-Hydroxy and 3-acetoxy-6-triphenyl-methylaminopenams |
-
1970
- 1970-11-03 GB GB5228570A patent/GB1368233A/en not_active Expired
-
1971
- 1971-07-30 DE DE19712138323 patent/DE2138323A1/de active Pending
- 1971-07-30 ES ES393800A patent/ES393800A1/es not_active Expired
- 1971-07-30 AT AT571174*1A patent/AT324566B/de not_active IP Right Cessation
- 1971-07-30 FR FR7128114A patent/FR2104819B1/fr not_active Expired
- 1971-07-30 AU AU31843/71A patent/AU467354B2/en not_active Expired
- 1971-07-30 CH CH1129471A patent/CH592097A5/xx not_active IP Right Cessation
- 1971-07-30 DE DE19712166022 patent/DE2166022A1/de active Pending
- 1971-07-30 NL NL7110612A patent/NL7110612A/xx unknown
- 1971-07-30 BE BE770727A patent/BE770727A/xx unknown
- 1971-07-30 JP JP5788271A patent/JPS554113B1/ja active Pending
-
1973
- 1973-03-30 AT AT281473A patent/AT329073B/de not_active IP Right Cessation
-
1976
- 1976-03-22 CH CH352876A patent/CH591504A5/xx not_active IP Right Cessation
-
1977
- 1977-05-03 CH CH551077A patent/CH594679A5/xx not_active IP Right Cessation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4115383A (en) | 1976-02-23 | 1978-09-19 | Eli Lilly And Company | Alkoxycarbonyl-ethylthio-azetidinones and process for their preparation |
Also Published As
| Publication number | Publication date |
|---|---|
| CH591504A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-09-30 |
| AT324566B (de) | 1975-09-10 |
| ATA281473A (de) | 1975-07-15 |
| DE2166022A1 (de) | 1972-09-28 |
| DE2138323A1 (de) | 1972-02-10 |
| FR2104819B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1975-08-01 |
| BE770727A (fr) | 1972-01-31 |
| FR2104819A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1972-04-21 |
| AU3184371A (en) | 1973-02-01 |
| AT329073B (de) | 1976-04-26 |
| AU467354B2 (en) | 1975-11-27 |
| JPS554113B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1980-01-29 |
| ES393800A1 (es) | 1974-07-16 |
| NL7110612A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1972-02-02 |
| CH594679A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1978-01-13 |
| CH592097A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-10-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed | ||
| PCNP | Patent ceased through non-payment of renewal fee |