GB1198941A - Benzimidazole Derivatives - Google Patents
Benzimidazole DerivativesInfo
- Publication number
- GB1198941A GB1198941A GB5259/68A GB525968A GB1198941A GB 1198941 A GB1198941 A GB 1198941A GB 5259/68 A GB5259/68 A GB 5259/68A GB 525968 A GB525968 A GB 525968A GB 1198941 A GB1198941 A GB 1198941A
- Authority
- GB
- United Kingdom
- Prior art keywords
- compound
- benzimidazole
- reacting
- give
- appropriate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- E—FIXED CONSTRUCTIONS
- E21—EARTH OR ROCK DRILLING; MINING
- E21D—SHAFTS; TUNNELS; GALLERIES; LARGE UNDERGROUND CHAMBERS
- E21D11/00—Lining tunnels, galleries or other underground cavities, e.g. large underground chambers; Linings therefor; Making such linings in situ, e.g. by assembling
- E21D11/14—Lining predominantly with metal
- E21D11/28—Longitudinal struts, i.e. longitudinal connections between adjoining arches
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Health & Medical Sciences (AREA)
- Mining & Mineral Resources (AREA)
- Life Sciences & Earth Sciences (AREA)
- Geology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Life Sciences & Earth Sciences (AREA)
- Geochemistry & Mineralogy (AREA)
- Civil Engineering (AREA)
- Architecture (AREA)
- Medicinal Chemistry (AREA)
- Structural Engineering (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US61374667A | 1967-02-03 | 1967-02-03 | |
| US69649668A | 1968-01-09 | 1968-01-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1198941A true GB1198941A (en) | 1970-07-15 |
Family
ID=27087090
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB46573/69A Expired GB1198942A (en) | 1967-02-03 | 1968-02-01 | Benzimidazole Derivatives |
| GB5259/68A Expired GB1198941A (en) | 1967-02-03 | 1968-02-01 | Benzimidazole Derivatives |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB46573/69A Expired GB1198942A (en) | 1967-02-03 | 1968-02-01 | Benzimidazole Derivatives |
Country Status (19)
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3853894A (en) * | 1972-06-02 | 1974-12-10 | Squibb & Sons Inc | Isothiocyanobenzimidazoles |
| USB486280I5 (enrdf_load_html_response) * | 1972-06-02 | 1976-02-03 | ||
| US3985755A (en) * | 1972-06-02 | 1976-10-12 | E. R. Squibb & Sons, Inc. | Pyridine containing isothiocyanobenzoxazoles |
| WO2005042513A1 (en) * | 2003-10-23 | 2005-05-12 | Sterix Limited | Phenyl carboxamide and sulfonamide derivatives for use as 11-beta-hydroxysteroid dehydrogenase |
| JP2006513159A (ja) * | 2002-11-01 | 2006-04-20 | メルク エンド カムパニー インコーポレーテッド | アンドロゲン受容体モジュレーターとしてのカルボニルアミノ−ベンズイミダゾール誘導体 |
| US7230020B2 (en) | 2003-10-23 | 2007-06-12 | Sterix Limited | 11β-hydroxysteroid dehydrogenase inhibitors |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3711608A (en) * | 1971-04-13 | 1973-01-16 | Merck & Co Inc | The treatment of pain, fever and inflammation with benzimidazoles |
| MA19290A1 (fr) * | 1980-05-22 | 1982-04-01 | Ciba Geigy Ag | Derives du benzole,leur preparaton et leur utilisations therapeutiques . |
| SE8604566D0 (sv) * | 1986-10-27 | 1986-10-27 | Haessle Ab | Novel compunds |
| CA2548657A1 (en) * | 2003-12-18 | 2005-06-30 | Tibotec Pharmaceuticals Ltd. | Aminobenzimidazoles and benzimidazoles as inhibitors of respiratory syncytial virus replication |
| RU2410382C2 (ru) * | 2005-03-17 | 2011-01-27 | Тиботек Фармасьютикалз Лтд | 1, 3-дигидробензимидазол-2-илиденовые амины в качестве ингибиторов репликации респираторного синцитиального вируса |
-
1968
- 1968-01-16 IE IE48/68A patent/IE31812B1/xx unknown
- 1968-01-30 BE BE710081D patent/BE710081A/xx not_active IP Right Cessation
- 1968-01-30 FI FI680234A patent/FI52859C/fi active
- 1968-01-31 SE SE1277/68A patent/SE346321B/xx unknown
- 1968-02-01 GB GB46573/69A patent/GB1198942A/en not_active Expired
- 1968-02-01 GB GB5259/68A patent/GB1198941A/en not_active Expired
- 1968-02-01 IT IT34575/68A patent/IT1044176B/it active
- 1968-02-01 NL NL6801482.A patent/NL157015B/xx not_active IP Right Cessation
- 1968-02-02 AT AT545070A patent/AT289828B/de not_active IP Right Cessation
- 1968-02-02 CH CH159768A patent/CH509318A/de not_active IP Right Cessation
- 1968-02-02 CH CH184271A patent/CH545796A/xx not_active IP Right Cessation
- 1968-02-02 CH CH184071A patent/CH545294A/de not_active IP Right Cessation
- 1968-02-02 CH CH183971A patent/CH545293A/de not_active IP Right Cessation
- 1968-02-02 ES ES350083A patent/ES350083A1/es not_active Expired
- 1968-02-02 AT AT544970A patent/AT289835B/de not_active IP Right Cessation
- 1968-02-02 DE DE1695545A patent/DE1695545C3/de not_active Expired
- 1968-02-02 NO NO413/68*[A patent/NO126484B/no unknown
- 1968-02-02 AT AT104468A patent/AT293378B/de active
- 1968-02-02 CH CH184171A patent/CH545295A/de not_active IP Right Cessation
- 1968-02-02 FR FR1580153D patent/FR1580153A/fr not_active Expired
- 1968-02-02 DK DK41168AA patent/DK139940B/da not_active IP Right Cessation
- 1968-02-02 AT AT545170A patent/AT289833B/de not_active IP Right Cessation
- 1968-02-02 AT AT545270A patent/AT301244B/de not_active IP Right Cessation
- 1968-02-02 DE DE1795711A patent/DE1795711C3/de not_active Expired
- 1968-02-02 CS CS815A patent/CS162651B2/cs unknown
- 1968-02-03 SU SU1215532A patent/SU540569A3/ru active
- 1968-02-08 OA OA53178A patent/OA04036A/xx unknown
- 1968-08-15 YU YU212/68A patent/YU33831B/xx unknown
-
1969
- 1969-02-17 ES ES363760A patent/ES363760A1/es not_active Expired
- 1969-02-17 ES ES363761A patent/ES363761A1/es not_active Expired
- 1969-02-17 ES ES363762A patent/ES363762A1/es not_active Expired
- 1969-06-27 BE BE735281D patent/BE735281A/xx not_active IP Right Cessation
-
1972
- 1972-08-31 CY CY65372A patent/CY653A/xx unknown
Cited By (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3853894A (en) * | 1972-06-02 | 1974-12-10 | Squibb & Sons Inc | Isothiocyanobenzimidazoles |
| USB486280I5 (enrdf_load_html_response) * | 1972-06-02 | 1976-02-03 | ||
| US3983130A (en) | 1972-06-02 | 1976-09-28 | E. R. Squibb & Sons, Inc. | Anthelmintic isothiocyanobenzoxazoles |
| US3985755A (en) * | 1972-06-02 | 1976-10-12 | E. R. Squibb & Sons, Inc. | Pyridine containing isothiocyanobenzoxazoles |
| JP2006513159A (ja) * | 2002-11-01 | 2006-04-20 | メルク エンド カムパニー インコーポレーテッド | アンドロゲン受容体モジュレーターとしてのカルボニルアミノ−ベンズイミダゾール誘導体 |
| EP1581217A4 (en) * | 2002-11-01 | 2007-07-11 | Merck & Co Inc | CARBONYLAMINO-BENZIMIDAZOLE DERIVATIVES AS MODULATORS OF ANDROGENIC RECEPTORS |
| AU2003286757B2 (en) * | 2002-11-01 | 2009-06-04 | Merck Sharp & Dohme Corp. | Carbonylamino-benzimidazole derivatives as androgen receptor modulators |
| US7622592B2 (en) | 2002-11-01 | 2009-11-24 | Merck & Co., Inc. | Carbonylamino-benzimidazole derivatives as androgen receptor modulators |
| WO2005042513A1 (en) * | 2003-10-23 | 2005-05-12 | Sterix Limited | Phenyl carboxamide and sulfonamide derivatives for use as 11-beta-hydroxysteroid dehydrogenase |
| US7230020B2 (en) | 2003-10-23 | 2007-06-12 | Sterix Limited | 11β-hydroxysteroid dehydrogenase inhibitors |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed | ||
| 48S | Specification amended (sect. 8/1949) | ||
| PCNP | Patent ceased through non-payment of renewal fee |