GB1155529A - Imidazole derivatives, their Preparation and Compositions containing them - Google Patents
Imidazole derivatives, their Preparation and Compositions containing themInfo
- Publication number
- GB1155529A GB1155529A GB35039/68A GB3503968A GB1155529A GB 1155529 A GB1155529 A GB 1155529A GB 35039/68 A GB35039/68 A GB 35039/68A GB 3503968 A GB3503968 A GB 3503968A GB 1155529 A GB1155529 A GB 1155529A
- Authority
- GB
- United Kingdom
- Prior art keywords
- radical
- oxoalkyl
- imidazole derivatives
- acid
- aralkoxycarbonylalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000002460 imidazoles Chemical class 0.000 title abstract 4
- 229940079865 intestinal antiinfectives imidazole derivative Drugs 0.000 title abstract 3
- 239000000203 mixture Substances 0.000 title 1
- 125000005188 oxoalkyl group Chemical group 0.000 abstract 3
- SEULWJSKCVACTH-UHFFFAOYSA-N 1-phenylimidazole Chemical compound C1=NC=CN1C1=CC=CC=C1 SEULWJSKCVACTH-UHFFFAOYSA-N 0.000 abstract 2
- DTQVDTLACAAQTR-UHFFFAOYSA-N Trifluoroacetic acid Chemical compound OC(=O)C(F)(F)F DTQVDTLACAAQTR-UHFFFAOYSA-N 0.000 abstract 2
- 125000005078 alkoxycarbonylalkyl group Chemical group 0.000 abstract 2
- -1 5-nitroimidazol - 1 - yl Chemical group 0.000 abstract 1
- VYDWQPKRHOGLPA-UHFFFAOYSA-N 5-nitroimidazole Chemical compound [O-][N+](=O)C1=CN=CN1 VYDWQPKRHOGLPA-UHFFFAOYSA-N 0.000 abstract 1
- 208000004881 Amebiasis Diseases 0.000 abstract 1
- 206010001980 Amoebiasis Diseases 0.000 abstract 1
- 208000014085 Chronic respiratory disease Diseases 0.000 abstract 1
- QOSSAOTZNIDXMA-UHFFFAOYSA-N Dicylcohexylcarbodiimide Chemical compound C1CCCCC1N=C=NC1CCCCC1 QOSSAOTZNIDXMA-UHFFFAOYSA-N 0.000 abstract 1
- GRYLNZFGIOXLOG-UHFFFAOYSA-N Nitric acid Chemical compound O[N+]([O-])=O GRYLNZFGIOXLOG-UHFFFAOYSA-N 0.000 abstract 1
- 208000030852 Parasitic disease Diseases 0.000 abstract 1
- QAOWNCQODCNURD-UHFFFAOYSA-N Sulfuric acid Chemical compound OS(O)(=O)=O QAOWNCQODCNURD-UHFFFAOYSA-N 0.000 abstract 1
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical compound [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 239000011248 coating agent Substances 0.000 abstract 1
- 238000000576 coating method Methods 0.000 abstract 1
- 230000032050 esterification Effects 0.000 abstract 1
- 238000005886 esterification reaction Methods 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 239000003701 inert diluent Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 238000006396 nitration reaction Methods 0.000 abstract 1
- 125000006501 nitrophenyl group Chemical group 0.000 abstract 1
- IOVCWXUNBOPUCH-UHFFFAOYSA-O nitrosooxidanium Chemical compound [OH2+]N=O IOVCWXUNBOPUCH-UHFFFAOYSA-O 0.000 abstract 1
- 230000003647 oxidation Effects 0.000 abstract 1
- 238000007254 oxidation reaction Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 150000003333 secondary alcohols Chemical class 0.000 abstract 1
- 235000011149 sulphuric acid Nutrition 0.000 abstract 1
- 239000001117 sulphuric acid Substances 0.000 abstract 1
- 201000002311 trypanosomiasis Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/91—Nitro radicals
- C07D233/92—Nitro radicals attached in position 4 or 5
- C07D233/94—Nitro radicals attached in position 4 or 5 with hydrocarbon radicals, substituted by oxygen or sulfur atoms, attached to other ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/91—Nitro radicals
- C07D233/92—Nitro radicals attached in position 4 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Devices For Checking Fares Or Tickets At Control Points (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47023965A | 1965-07-07 | 1965-07-07 | |
| US55093266A | 1966-05-18 | 1966-05-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1155529A true GB1155529A (en) | 1969-06-18 |
Family
ID=27043018
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB35039/68A Expired GB1155529A (en) | 1965-07-07 | 1966-07-04 | Imidazole derivatives, their Preparation and Compositions containing them |
| GB29846/66A Expired GB1153347A (en) | 1965-07-07 | 1966-07-04 | Imidazole Derivatives, their preparation and Compositions containing them. |
| GB32952/68A Expired GB1155528A (en) | 1965-07-07 | 1966-07-04 | Imidazole derivatives, their Preparation and Compositions containing them |
| GB38884/68A Expired GB1155530A (en) | 1965-07-07 | 1966-07-04 | Imidazole Derivatives, their Preparation and Compositions containing them |
| GB35033/68A Expired GB1154290A (en) | 1965-07-07 | 1966-07-04 | Imidazole Derivatives, their preparation and compositions containing them |
Family Applications After (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB29846/66A Expired GB1153347A (en) | 1965-07-07 | 1966-07-04 | Imidazole Derivatives, their preparation and Compositions containing them. |
| GB32952/68A Expired GB1155528A (en) | 1965-07-07 | 1966-07-04 | Imidazole derivatives, their Preparation and Compositions containing them |
| GB38884/68A Expired GB1155530A (en) | 1965-07-07 | 1966-07-04 | Imidazole Derivatives, their Preparation and Compositions containing them |
| GB35033/68A Expired GB1154290A (en) | 1965-07-07 | 1966-07-04 | Imidazole Derivatives, their preparation and compositions containing them |
Country Status (18)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016156290A1 (en) * | 2015-04-02 | 2016-10-06 | Bayer Cropscience Aktiengesellschaft | Novel 5-substituted imidazole derivatives |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1280355A (en) * | 1969-06-20 | 1972-07-05 | Rech S Et D Applic Scient Et M | Substituted 5-nitro-imidazoles and their preparation |
| BE758145A (fr) * | 1969-10-29 | 1971-04-28 | Smith Kline French Lab | Iso-thio-urees et derives |
| US3678066A (en) * | 1970-03-06 | 1972-07-18 | Squibb & Sons Inc | Thiocyanic acid esters |
| US3968228A (en) * | 1973-11-13 | 1976-07-06 | Merck & Co., Inc. | 4-Nitro-5-cyanoimidazoles as coccidiostats |
| JPH02254965A (ja) * | 1989-03-28 | 1990-10-15 | Chiyoudendou Hatsuden Kanren Kiki Zairyo Gijutsu Kenkyu Kumiai | 超電導回転電機の回転子 |
| EP3519389A1 (en) | 2016-09-29 | 2019-08-07 | Bayer CropScience Aktiengesellschaft | Novel 5-substituted imidazolylmethyl derivatives |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5149436B2 (enrdf_load_stackoverflow) * | 1971-11-15 | 1976-12-27 |
-
1966
- 1966-06-08 IL IL25931A patent/IL25931A/en unknown
- 1966-07-04 GB GB35039/68A patent/GB1155529A/en not_active Expired
- 1966-07-04 GB GB29846/66A patent/GB1153347A/en not_active Expired
- 1966-07-04 GB GB32952/68A patent/GB1155528A/en not_active Expired
- 1966-07-04 GB GB38884/68A patent/GB1155530A/en not_active Expired
- 1966-07-04 GB GB35033/68A patent/GB1154290A/en not_active Expired
- 1966-07-05 IT IT6615338A patent/IT1061026B/it active
- 1966-07-05 AT AT559369A patent/AT291990B/de not_active IP Right Cessation
- 1966-07-05 AT AT643566A patent/AT284114B/de not_active IP Right Cessation
- 1966-07-05 AT AT559269A patent/AT291989B/de not_active IP Right Cessation
- 1966-07-05 AT AT545669A patent/AT294487B/de not_active IP Right Cessation
- 1966-07-05 AT AT551669A patent/AT291988B/de not_active IP Right Cessation
- 1966-07-05 ES ES0329085A patent/ES329085A1/es not_active Expired
- 1966-07-06 DE DE1966M0070135 patent/DE1620018B2/de active Granted
- 1966-07-06 DK DK348866AA patent/DK141287B/da unknown
- 1966-07-06 FR FR68482A patent/FR1502699A/fr not_active Expired
- 1966-07-06 FI FI661807A patent/FI46961C/fi active
- 1966-07-06 BR BR181050/66A patent/BR6681050D0/pt unknown
- 1966-07-06 SE SE9274/66A patent/SE343578B/xx unknown
- 1966-07-06 NO NO163800A patent/NO122186B/no unknown
- 1966-07-07 CH CH991771A patent/CH565769A5/xx not_active IP Right Cessation
- 1966-07-07 CH CH988566A patent/CH562806A5/xx not_active IP Right Cessation
- 1966-07-07 CH CH988566A patent/CH522651A/de not_active IP Right Cessation
- 1966-07-07 BE BE683796D patent/BE683796A/xx not_active IP Right Cessation
- 1966-07-07 JP JP41043868A patent/JPS5010865B1/ja active Pending
- 1966-07-07 NL NL666609552A patent/NL149793B/xx not_active IP Right Cessation
- 1966-10-05 FR FR78932A patent/FR5890M/fr not_active Expired
-
1970
- 1970-11-09 CY CY56570A patent/CY565A/xx unknown
- 1970-11-09 JP JP45097971A patent/JPS4843909B1/ja active Pending
- 1970-11-27 IL IL35748A patent/IL35748A0/xx unknown
-
1971
- 1971-12-31 MY MY197155A patent/MY7100055A/xx unknown
-
1974
- 1974-11-29 JP JP49136394A patent/JPS5138718B1/ja active Pending
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016156290A1 (en) * | 2015-04-02 | 2016-10-06 | Bayer Cropscience Aktiengesellschaft | Novel 5-substituted imidazole derivatives |
| CN107635968A (zh) * | 2015-04-02 | 2018-01-26 | 拜耳作物科学股份公司 | 新的5‑取代的咪唑衍生物 |
| US10231453B2 (en) | 2015-04-02 | 2019-03-19 | Bayer Cropscience Aktiengesellschaft | 5-substituted imidazole derivatives |
| US10568326B2 (en) | 2015-04-02 | 2020-02-25 | Bayer Cropscience Aktiengesellschaft | 5-substituted imidazole derivatives |
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