FR2553408B1 - 1- (4-ACETYLAMINOPHENYL) -2-AMINO-PROPANONE DERIVATIVES, THEIR USE IN THERAPEUTICS AND THEIR PREPARATION PROCESS - Google Patents

1- (4-ACETYLAMINOPHENYL) -2-AMINO-PROPANONE DERIVATIVES, THEIR USE IN THERAPEUTICS AND THEIR PREPARATION PROCESS

Info

Publication number
FR2553408B1
FR2553408B1 FR8316408A FR8316408A FR2553408B1 FR 2553408 B1 FR2553408 B1 FR 2553408B1 FR 8316408 A FR8316408 A FR 8316408A FR 8316408 A FR8316408 A FR 8316408A FR 2553408 B1 FR2553408 B1 FR 2553408B1
Authority
FR
France
Prior art keywords
acetylaminophenyl
therapeutics
amino
preparation process
propanone derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR8316408A
Other languages
French (fr)
Other versions
FR2553408A1 (en
Inventor
Louis Lafon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Cephalon France SAS
Original Assignee
Laboratoire L Lafon SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratoire L Lafon SA filed Critical Laboratoire L Lafon SA
Priority to FR8316408A priority Critical patent/FR2553408B1/en
Priority to MA20470A priority patent/MA20246A1/en
Priority to CA000464759A priority patent/CA1250838A/en
Priority to IE2555/84A priority patent/IE57807B1/en
Priority to PT79328A priority patent/PT79328B/en
Priority to AU34092/84A priority patent/AU570076B2/en
Priority to DK484884A priority patent/DK164900C/en
Priority to ES536969A priority patent/ES536969A0/en
Priority to NO844072A priority patent/NO164650C/en
Priority to NZ209871A priority patent/NZ209871A/en
Priority to DE8484402064T priority patent/DE3463764D1/en
Priority to AT84402064T priority patent/ATE27267T1/en
Priority to OA58410A priority patent/OA07833A/en
Priority to GR80636A priority patent/GR80636B/en
Priority to FI844030A priority patent/FI83509C/en
Priority to EP84402064A priority patent/EP0138714B1/en
Priority to HU843837A priority patent/HU194847B/en
Priority to YU1747/84A priority patent/YU43859B/en
Priority to IL73231A priority patent/IL73231A/en
Priority to JP59217207A priority patent/JPS60120845A/en
Priority to ZA848021A priority patent/ZA848021B/en
Publication of FR2553408A1 publication Critical patent/FR2553408A1/en
Application granted granted Critical
Publication of FR2553408B1 publication Critical patent/FR2553408B1/en
Priority to US07/038,981 priority patent/US4877812A/en
Priority to US07/375,987 priority patent/US4933442A/en
Priority to US07/376,635 priority patent/US4963570A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/10—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms
    • C07D295/104—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/108—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
FR8316408A 1983-10-14 1983-10-14 1- (4-ACETYLAMINOPHENYL) -2-AMINO-PROPANONE DERIVATIVES, THEIR USE IN THERAPEUTICS AND THEIR PREPARATION PROCESS Expired FR2553408B1 (en)

Priority Applications (24)

Application Number Priority Date Filing Date Title
FR8316408A FR2553408B1 (en) 1983-10-14 1983-10-14 1- (4-ACETYLAMINOPHENYL) -2-AMINO-PROPANONE DERIVATIVES, THEIR USE IN THERAPEUTICS AND THEIR PREPARATION PROCESS
MA20470A MA20246A1 (en) 1983-10-14 1984-10-04 Process for the preparation of new derivatives of 1- (acetylaminophenyl) -2 aminopropanone.
CA000464759A CA1250838A (en) 1983-10-14 1984-10-04 Process for preparing 1-(acetylaminophenyl)-2-amino-propanone derivatives; derivatives thus obtained
IE2555/84A IE57807B1 (en) 1983-10-14 1984-10-05 1-(acetylaminophenyl)-2-aminopropanone derivatives,their use in therapy and process for their preparation
PT79328A PT79328B (en) 1983-10-14 1984-10-09 PROCESS FOR PREPARING NOVEL 1- (ACETYLAMINOPHENYL) -2-AMINO-PROPANONE DERIVATIVES
AU34092/84A AU570076B2 (en) 1983-10-14 1984-10-10 1-(acetylaminophenyl)-2-amino-propanones
DK484884A DK164900C (en) 1983-10-14 1984-10-10 DERIVATIVES OF 1- (ACETYLAMINOPHENYL) -2-AMINOPROPANON, A THERAPEUTIC AGENT CONTAINING THESE AND THEIR PREPARATION
NO844072A NO164650C (en) 1983-10-14 1984-10-11 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 1- (ACETYLAMINOPHENYL) -2-AMINOPROPANON DERIVATIVES.
ES536969A ES536969A0 (en) 1983-10-14 1984-10-11 PROCEDURE FOR THE PREPARATION OF NEW DERIVATIVES OF 1- (ACETILAMINOFENIL) -2-AMINO-PROPANONA
GR80636A GR80636B (en) 1983-10-14 1984-10-12 Method for the preparation of novel 1-(acetylaminophenyl)-2-amino-propanone derivatives
AT84402064T ATE27267T1 (en) 1983-10-14 1984-10-12 1-(ACETYLAMINOPHENYL)-2-AMINO-PROPANONE DERIVATIVES THEIR THERAPEUTIC USE AND PROCESS FOR THEIR MANUFACTURE.
OA58410A OA07833A (en) 1983-10-14 1984-10-12 Process for the preparation of new derivatives of 1- (acetylamino) -2-amino-propanone.
NZ209871A NZ209871A (en) 1983-10-14 1984-10-12 1-(acetylaminophenyl)-2-aminopropanone derivatives and pharmaceutical compositions
FI844030A FI83509C (en) 1983-10-14 1984-10-12 FOR EXAMINATION OF THE PHARMACEUTICAL PROCEDURE 1- (ACETYLAMINOPHENYL) -2-AMINOPROPANONDERIVAT.
EP84402064A EP0138714B1 (en) 1983-10-14 1984-10-12 1-(acetylaminophenyl)-2-amino-propanone derivatives, their therapeutical use and process for their preparation
HU843837A HU194847B (en) 1983-10-14 1984-10-12 Process for producing 1-/acetyl-amino-phenyl/-2-amino-propanone derivatives and salts and pharmaceutical compositions containing them as active components
YU1747/84A YU43859B (en) 1983-10-14 1984-10-12 Process for obtaining derivatives of 1-(acetyl-aminophenyl)-2-amino propanone
DE8484402064T DE3463764D1 (en) 1983-10-14 1984-10-12 1-(acetylaminophenyl)-2-amino-propanone derivatives, their therapeutical use and process for their preparation
IL73231A IL73231A (en) 1983-10-14 1984-10-14 1-acetylaminophenyl-2-amino-propanone derivatives,their preparation and pharmaceutical compositions containing them
JP59217207A JPS60120845A (en) 1983-10-14 1984-10-15 1-(acetylaminophenyl)-2-aminopropanone derivative, manufacture and therapeutical composition
ZA848021A ZA848021B (en) 1983-10-14 1984-10-15 1-(acetylaminophenyl)-2-amino-propanone derivatives useful as pharmaceuticals
US07/038,981 US4877812A (en) 1983-10-14 1987-04-16 1-(acetylaminophenyl)-2-aminopropanone derivatives and antidepressant compositions thereof
US07/375,987 US4933442A (en) 1983-10-14 1989-07-06 1-(acetylaminophenyl)-2-aminopropanone derivatives and central nervous system antidepressant compositions
US07/376,635 US4963570A (en) 1983-10-14 1989-07-07 1-(acetylaminophenyl)-2-aminopropanone derivatives and pharmaceutical compositions thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8316408A FR2553408B1 (en) 1983-10-14 1983-10-14 1- (4-ACETYLAMINOPHENYL) -2-AMINO-PROPANONE DERIVATIVES, THEIR USE IN THERAPEUTICS AND THEIR PREPARATION PROCESS

Publications (2)

Publication Number Publication Date
FR2553408A1 FR2553408A1 (en) 1985-04-19
FR2553408B1 true FR2553408B1 (en) 1986-11-28

Family

ID=9293165

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8316408A Expired FR2553408B1 (en) 1983-10-14 1983-10-14 1- (4-ACETYLAMINOPHENYL) -2-AMINO-PROPANONE DERIVATIVES, THEIR USE IN THERAPEUTICS AND THEIR PREPARATION PROCESS

Country Status (3)

Country Link
JP (1) JPS60120845A (en)
FR (1) FR2553408B1 (en)
ZA (1) ZA848021B (en)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1262965A (en) * 1969-03-21 1972-02-09 Ferrosan As Butyrophenones
FR2430933A1 (en) * 1978-07-13 1980-02-08 Synthelabo PROPIOPHENONE DERIVATIVES AND THEIR THERAPEUTIC APPLICATION

Also Published As

Publication number Publication date
FR2553408A1 (en) 1985-04-19
ZA848021B (en) 1985-06-26
JPS60120845A (en) 1985-06-28
JPH058696B2 (en) 1993-02-02

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Legal Events

Date Code Title Description
ST Notification of lapse