FR2317929A1 - Derives d'acide azanaphtaleneacetique et leur utilisation comme agents anti-inflammatoires - Google Patents

Derives d'acide azanaphtaleneacetique et leur utilisation comme agents anti-inflammatoires

Info

Publication number
FR2317929A1
FR2317929A1 FR7621673A FR7621673A FR2317929A1 FR 2317929 A1 FR2317929 A1 FR 2317929A1 FR 7621673 A FR7621673 A FR 7621673A FR 7621673 A FR7621673 A FR 7621673A FR 2317929 A1 FR2317929 A1 FR 2317929A1
Authority
FR
France
Prior art keywords
azanaphtaleneacetic
acid derivatives
inflammatory agents
inflammatory
agents
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7621673A
Other languages
English (en)
Other versions
FR2317929B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GD Searle LLC
Original Assignee
GD Searle LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by GD Searle LLC filed Critical GD Searle LLC
Publication of FR2317929A1 publication Critical patent/FR2317929A1/fr
Application granted granted Critical
Publication of FR2317929B1 publication Critical patent/FR2317929B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • C07D215/227Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Quinoline Compounds (AREA)
FR7621673A 1975-07-16 1976-07-15 Derives d'acide azanaphtaleneacetique et leur utilisation comme agents anti-inflammatoires Granted FR2317929A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/596,509 US3991061A (en) 1975-07-16 1975-07-16 Azanaphthaleneacetic acid derivatives

Publications (2)

Publication Number Publication Date
FR2317929A1 true FR2317929A1 (fr) 1977-02-11
FR2317929B1 FR2317929B1 (fr) 1979-10-12

Family

ID=24387582

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7621673A Granted FR2317929A1 (fr) 1975-07-16 1976-07-15 Derives d'acide azanaphtaleneacetique et leur utilisation comme agents anti-inflammatoires

Country Status (10)

Country Link
US (1) US3991061A (fr)
JP (1) JPS5212177A (fr)
AU (1) AU499163B2 (fr)
BE (1) BE844204A (fr)
CA (1) CA1082711A (fr)
DE (1) DE2631735A1 (fr)
FR (1) FR2317929A1 (fr)
GB (1) GB1508923A (fr)
SE (1) SE7608081L (fr)
ZA (1) ZA764209B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH628892A5 (it) * 1977-06-22 1982-03-31 Simes Procedimento per la preparazione di acidi chinolinici ad attivita antiinfiammatoria.
JPS5587771A (en) * 1978-12-27 1980-07-02 Teikoku Hormone Mfg Co Ltd 1-phenylisoquinoline derivative
AU778306B2 (en) 1999-10-22 2004-11-25 Sanofi-Aventis Phenyl- and pyridyl-tetrahydro-pyridines having TNF inhibiting activity
WO2007146838A2 (fr) * 2006-06-09 2007-12-21 Icos Corporation Acides phénylacétiques substitués utilisés en tant qu'antagonistes de dp-2

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2181801A1 (fr) * 1972-03-10 1973-12-07 Ciba Geigy Ag

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2921939A (en) * 1955-11-28 1960-01-19 Metal & Thermit Corp Process for preparing alpha-substituted acetic acids

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2181801A1 (fr) * 1972-03-10 1973-12-07 Ciba Geigy Ag

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
JOURNAL OF MEDICINAL CHEMISTRY, 18, PAGES 395-99, 1975 *

Also Published As

Publication number Publication date
CA1082711A (fr) 1980-07-29
AU1591476A (en) 1978-01-19
AU499163B2 (en) 1979-04-05
US3991061A (en) 1976-11-09
DE2631735A1 (de) 1977-02-03
ZA764209B (en) 1978-02-22
BE844204A (fr) 1977-01-17
FR2317929B1 (fr) 1979-10-12
SE7608081L (sv) 1977-01-17
JPS5212177A (en) 1977-01-29
GB1508923A (en) 1978-04-26

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Legal Events

Date Code Title Description
ST Notification of lapse