FR2104765A1 - Diuretic 6-sulphamyl tetrahydroquinazolinones prodn - - from 5-halo-2-alkyl anilines - Google Patents
Diuretic 6-sulphamyl tetrahydroquinazolinones prodn - - from 5-halo-2-alkyl anilinesInfo
- Publication number
- FR2104765A1 FR2104765A1 FR7123420A FR7123420A FR2104765A1 FR 2104765 A1 FR2104765 A1 FR 2104765A1 FR 7123420 A FR7123420 A FR 7123420A FR 7123420 A FR7123420 A FR 7123420A FR 2104765 A1 FR2104765 A1 FR 2104765A1
- Authority
- FR
- France
- Prior art keywords
- alkyl
- halo
- tetrahydroquinazolinones
- sulphamyl
- prodn
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- ZMMSDXIZPARXPH-UHFFFAOYSA-N 2-oxo-3,4,4a,5-tetrahydro-1H-quinazoline-6-sulfonamide Chemical class S(N)(=O)(=O)C=1CC2CNC(NC2=CC=1)=O ZMMSDXIZPARXPH-UHFFFAOYSA-N 0.000 title 1
- 239000002934 diuretic Substances 0.000 title 1
- 230000001882 diuretic effect Effects 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 238000006243 chemical reaction Methods 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- KXDAEFPNCMNJSK-UHFFFAOYSA-N Benzamide Chemical compound NC(=O)C1=CC=CC=C1 KXDAEFPNCMNJSK-UHFFFAOYSA-N 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 229910006074 SO2NH2 Inorganic materials 0.000 abstract 1
- DHKHKXVYLBGOIT-UHFFFAOYSA-N acetaldehyde Diethyl Acetal Natural products CCOC(C)OCC DHKHKXVYLBGOIT-UHFFFAOYSA-N 0.000 abstract 1
- 125000002777 acetyl group Chemical class [H]C([H])([H])C(*)=O 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000005110 aryl thio group Chemical group 0.000 abstract 1
- 230000005494 condensation Effects 0.000 abstract 1
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 abstract 1
- 125000002485 formyl group Chemical class [H]C(*)=O 0.000 abstract 1
- 125000004995 haloalkylthio group Chemical group 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 150000002576 ketones Chemical class 0.000 abstract 1
- 230000003647 oxidation Effects 0.000 abstract 1
- 238000007254 oxidation reaction Methods 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 238000006798 ring closing metathesis reaction Methods 0.000 abstract 1
- 238000007363 ring formation reaction Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000000446 sulfanediyl group Chemical group *S* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
- C07D265/26—Two oxygen atoms, e.g. isatoic anhydride
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5089570A | 1970-06-29 | 1970-06-29 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2104765A1 true FR2104765A1 (en) | 1972-04-21 |
| FR2104765B1 FR2104765B1 (enExample) | 1975-10-10 |
Family
ID=21968132
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7123420A Granted FR2104765A1 (en) | 1970-06-29 | 1971-06-28 | Diuretic 6-sulphamyl tetrahydroquinazolinones prodn - - from 5-halo-2-alkyl anilines |
Country Status (5)
| Country | Link |
|---|---|
| CH (1) | CH546244A (enExample) |
| DE (1) | DE2131622A1 (enExample) |
| FR (1) | FR2104765A1 (enExample) |
| LU (1) | LU63414A1 (enExample) |
| NL (1) | NL7108861A (enExample) |
-
1971
- 1971-06-11 CH CH546244D patent/CH546244A/fr not_active IP Right Cessation
- 1971-06-25 LU LU63414D patent/LU63414A1/xx unknown
- 1971-06-25 DE DE19712131622 patent/DE2131622A1/de active Pending
- 1971-06-25 NL NL7108861A patent/NL7108861A/xx not_active Application Discontinuation
- 1971-06-28 FR FR7123420A patent/FR2104765A1/fr active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| DE2131622A1 (de) | 1972-01-05 |
| FR2104765B1 (enExample) | 1975-10-10 |
| NL7108861A (enExample) | 1971-12-31 |
| LU63414A1 (enExample) | 1971-09-24 |
| CH546244A (fr) | 1974-02-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TP | Transmission of property |