FI94761C - 4- och 6-substituerade 1,2,3,3a,8,8a-hexahydro-1,3a,8-trimetylpyrrolo/2,3-b/indolderivat - Google Patents

4- och 6-substituerade 1,2,3,3a,8,8a-hexahydro-1,3a,8-trimetylpyrrolo/2,3-b/indolderivat Download PDF

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Publication number
FI94761C
FI94761C FI933119A FI933119A FI94761C FI 94761 C FI94761 C FI 94761C FI 933119 A FI933119 A FI 933119A FI 933119 A FI933119 A FI 933119A FI 94761 C FI94761 C FI 94761C
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FI
Finland
Prior art keywords
hexahydro
cis
added
trimethylpyrrolo
indol
Prior art date
Application number
FI933119A
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English (en)
Finnish (fi)
Other versions
FI94761B (sv
FI933119A0 (sv
FI933119A (sv
Inventor
Edward J Glamkowski
Barbara E Kurys
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Priority claimed from US07/431,103 external-priority patent/US5081117A/en
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of FI933119A0 publication Critical patent/FI933119A0/sv
Publication of FI933119A publication Critical patent/FI933119A/sv
Publication of FI94761B publication Critical patent/FI94761B/sv
Application granted granted Critical
Publication of FI94761C publication Critical patent/FI94761C/sv

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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)

Claims (4)

  1. 33 94761 L Patenttivaatimus 4- ja 6-substituoidut l,2,3,3a,8,8a-heksahydro-1,3a,8-trimetyylipyrrolo[2,3-b]indolijohdannaiset, joilla 5 on kaava III
  2. 4 CH3 , Jp-XJ
  3. 10 X 1 H * A ch3 CH3 jossa R3 on vety tai metyyli ja X on vety tai halogeeni sekä niiden optiset isomeerit 3aS-cis- ja 3aR-cis-isomee-15 rit mukaan luettuna, isomeerien raseemiset seokset ja näiden happoadditiosuolat. 20 4- och 6-substituerade l,2,3,3a,8,8a-hexahydro- l,3a,8-trimetylpyrrolo[2,3-b]indolderivat med formeln III
  4. 4 CH3 vPrP Ä ch3 CH3 väri R3 är väte eller metyl och X är väte eller halogen 30 samt deras optiska isomerer inkluderande 3aS-cis- och 3aR-cis-isomererna, racemiska blandningar av isomerer och sy-raadditionssalter därav.
FI933119A 1989-11-03 1993-07-07 4- och 6-substituerade 1,2,3,3a,8,8a-hexahydro-1,3a,8-trimetylpyrrolo/2,3-b/indolderivat FI94761C (sv)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US07/431,103 US5081117A (en) 1989-09-28 1989-11-03 4- and 6-carbamates related to physostigmine and intermediates for the preparation thereof
US43110389 1989-11-03
FI905418 1990-11-01
FI905418A FI92701C (sv) 1989-09-28 1990-11-01 Förfarande för framställning av terapeutiskt användbara 4- eller 6-substituerade trimetylpyrrolo/2,3-b/indolkarbamater

Publications (4)

Publication Number Publication Date
FI933119A0 FI933119A0 (sv) 1993-07-07
FI933119A FI933119A (sv) 1993-07-07
FI94761B FI94761B (sv) 1995-07-14
FI94761C true FI94761C (sv) 1995-10-25

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Family Applications (1)

Application Number Title Priority Date Filing Date
FI933119A FI94761C (sv) 1989-11-03 1993-07-07 4- och 6-substituerade 1,2,3,3a,8,8a-hexahydro-1,3a,8-trimetylpyrrolo/2,3-b/indolderivat

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FI (1) FI94761C (sv)

Also Published As

Publication number Publication date
FI94761B (sv) 1995-07-14
FI933119A0 (sv) 1993-07-07
FI933119A (sv) 1993-07-07

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Owner name: HOECHST MARION ROUSSEL, INC.