FI941644A0 - Antifungala triatzolföreningar - Google Patents

Antifungala triatzolföreningar

Info

Publication number
FI941644A0
FI941644A0 FI941644A FI941644A FI941644A0 FI 941644 A0 FI941644 A0 FI 941644A0 FI 941644 A FI941644 A FI 941644A FI 941644 A FI941644 A FI 941644A FI 941644 A0 FI941644 A0 FI 941644A0
Authority
FI
Finland
Prior art keywords
pct
image
date apr
compounds against
triazole compounds
Prior art date
Application number
FI941644A
Other languages
English (en)
Finnish (fi)
Other versions
FI108131B (sv
FI941644A (sv
Inventor
Andrew Simon Bell
Kenneth Richardson
Peter John Whittle
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI941644A publication Critical patent/FI941644A/sv
Publication of FI941644A0 publication Critical patent/FI941644A0/sv
Application granted granted Critical
Publication of FI108131B publication Critical patent/FI108131B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62Oxygen or sulfur atoms
    • C07D213/70Sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cephalosporin Compounds (AREA)
FI941644A 1991-10-10 1994-04-08 Förfarande för framställning av ett terapeutiskt användbart triazolderivat och en ny mellanprodukt FI108131B (sv)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB919121456A GB9121456D0 (en) 1991-10-10 1991-10-10 Triazole antifungal agents
GB9121456 1991-10-10
EP9202278 1992-10-01
PCT/EP1992/002278 WO1993007139A1 (en) 1991-10-10 1992-10-01 Triazole antifungal agents

Publications (3)

Publication Number Publication Date
FI941644A FI941644A (sv) 1994-04-08
FI941644A0 true FI941644A0 (sv) 1994-04-08
FI108131B FI108131B (sv) 2001-11-30

Family

ID=10702663

Family Applications (1)

Application Number Title Priority Date Filing Date
FI941644A FI108131B (sv) 1991-10-10 1994-04-08 Förfarande för framställning av ett terapeutiskt användbart triazolderivat och en ny mellanprodukt

Country Status (13)

Country Link
US (1) US5541203A (sv)
EP (1) EP0607193B1 (sv)
JP (1) JPH07502022A (sv)
AT (1) ATE196293T1 (sv)
CA (1) CA2118937C (sv)
DE (1) DE69231445T2 (sv)
DK (1) DK0607193T3 (sv)
ES (1) ES2149777T3 (sv)
FI (1) FI108131B (sv)
GB (1) GB9121456D0 (sv)
GR (1) GR3034769T3 (sv)
PT (1) PT100942B (sv)
WO (1) WO1993007139A1 (sv)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9317491D0 (en) * 1993-08-23 1993-10-06 Fujisawa Pharmaceutical Co New compound and a process for preparation thereof
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
GB9512961D0 (en) * 1995-06-26 1995-08-30 Pfizer Ltd Antifungal agents
GB9605705D0 (en) * 1996-03-19 1996-05-22 Pfizer Ltd Therapeutic agents
KR100889937B1 (ko) * 2007-08-06 2009-03-20 한미약품 주식회사 보리코나졸의 제조방법
GB2452049A (en) * 2007-08-21 2009-02-25 Alpharma Aps Process for the preparation of voriconazole
KR101912850B1 (ko) * 2011-06-19 2018-10-30 비아멧 파마슈티컬즈(엔씨), 인코포레이티드 금속효소 억제제 화합물
EP2721022B1 (en) * 2011-06-19 2019-03-06 Viamet Pharmaceuticals (NC), Inc. Metalloenzyme inhibitor compounds
CN104136427B (zh) * 2012-01-20 2017-03-01 威尔金制药有限公司 金属酶抑制剂化合物
TWI561515B (en) * 2012-03-16 2016-12-11 Viamet Pharmaceuticals Inc Metalloenzyme inhibitor compounds
WO2016187201A2 (en) 2015-05-18 2016-11-24 Viamet Pharmaceuticals, Inc. Antifungal compounds
EP3544427A4 (en) * 2016-11-22 2020-04-29 Dow Agrosciences Llc FUNGICIDE COMPOUNDS AND MIXTURES FOR CONTROLLING MUSHROOMS IN CEREALS
RU2019118631A (ru) * 2016-11-22 2020-12-24 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Применение соединения дифтор-(2-гидроксипропил)пиридина в качестве фунгицида для борьбы с фитопатогенным грибком ячменя
AR110210A1 (es) * 2016-11-22 2019-03-06 Viamet Pharmaceuticals Inc Uso de un compuesto de difluoro-(2-hidroxipropil)piridina como fungicida para el control de la mancha foliar en remolacha azucarera
CA3044386A1 (en) * 2016-11-22 2018-05-31 Dow Agrosciences Llc Use of a difluoro-(2-hydroxypropyl)pyridine compound as a fungicide for control of phytopathogenic fungi of corn
CN110290705A (zh) * 2016-11-22 2019-09-27 美国陶氏益农公司 用于谷物中的杀真菌防治的杀真菌化合物和混合物
BR112019010038A2 (pt) * 2016-11-22 2019-09-03 Dow Agrosciences Llc uso de um composto de difluoro-(2-hidroxipropildpiridina como fungicida para controle de fungos fitopatogênicos do arroz
MA46075B1 (fr) * 2016-11-22 2020-05-29 Dow Agrosciences Llc Composés et mélanges fongicides destinés à lutter contre les champignons dans les céréales
CA3044383A1 (en) * 2016-11-22 2018-05-31 Dow Agrosciences Llc Use of a difluoro-(2-hydroxypropyl)pyridine compound as a fungicide for control of phytopathogenic fungi of wheat
AU2017363226A1 (en) * 2016-11-22 2019-06-20 Corteva Agriscience Llc Fungicidal compounds and mixtures for fungal control in cereals
AU2017365179B2 (en) 2016-11-22 2021-09-02 Corteva Agriscience Llc Fungicidal compounds and mixtures for fungal control in cereals

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE322526C (de) * 1918-08-31 1920-07-01 Hermann Meyer Sicherheitskettenverschluss fuer Korridortueren u. dgl.
EP0158741A3 (en) * 1980-11-19 1986-02-12 Imperial Chemical Industries Plc Intermediates for fungicidal triazole and imidazole compounds
ES523184A0 (es) * 1982-06-17 1985-04-01 Pfizer Un procedimiento para la preparacion de un compuesto dotado de propiedades fungicidas
DE3245504A1 (de) * 1982-12-09 1984-06-14 Bayer Ag, 5090 Leverkusen Fungizide mittel, deren herstellung und verwendung
US4952232A (en) * 1987-04-29 1990-08-28 E. I. Du Pont De Nemours And Company Antifungal carbinols
DE3813841A1 (de) * 1987-06-03 1988-12-15 Bayer Ag Heterocyclische hydroxyethylazole
DE3732385A1 (de) * 1987-09-25 1989-04-06 Bayer Ag Hydroxyalkylcyclopropyl1-1,2,4-triazolyl- oder -imidazolyl-derivate und ihre verwendung als antimykotische mittel
WO1989005801A1 (en) * 1987-12-17 1989-06-29 E.I. Du Pont De Nemours And Company Antifungal carbinols
FI97382C (sv) * 1988-03-04 1996-12-10 Sankyo Co Förfarande för framställning av som läkemedel användbara 1,2,4-triazolderivat
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
GB9002375D0 (en) * 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents

Also Published As

Publication number Publication date
CA2118937A1 (en) 1993-04-15
FI108131B (sv) 2001-11-30
GB9121456D0 (en) 1991-11-27
FI941644A (sv) 1994-04-08
WO1993007139A1 (en) 1993-04-15
US5541203A (en) 1996-07-30
CA2118937C (en) 1998-04-28
DE69231445T2 (de) 2001-01-11
GR3034769T3 (en) 2001-02-28
EP0607193B1 (en) 2000-09-13
EP0607193A1 (en) 1994-07-27
DE69231445D1 (de) 2000-10-19
JPH07502022A (ja) 1995-03-02
PT100942A (pt) 1993-10-29
PT100942B (pt) 1999-07-30
ES2149777T3 (es) 2000-11-16
DK0607193T3 (da) 2000-10-09
ATE196293T1 (de) 2000-09-15

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