FI810991A7 - Kolesterolin biosynteesin inhibiitit, niiden valmistus ja käyttö. - Google Patents

Kolesterolin biosynteesin inhibiitit, niiden valmistus ja käyttö. Download PDF

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Publication number
FI810991A7
FI810991A7 FI810991A FI810991A FI810991A7 FI 810991 A7 FI810991 A7 FI 810991A7 FI 810991 A FI810991 A FI 810991A FI 810991 A FI810991 A FI 810991A FI 810991 A7 FI810991 A7 FI 810991A7
Authority
FI
Finland
Prior art keywords
preparation
biosynthesis inhibitors
cholesterol biosynthesis
cholesterol
inhibitors
Prior art date
Application number
FI810991A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI810991L (fi
Inventor
Aiya Sato
Akira Terahara
Yoshio Tsujita
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=12604367&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI810991(A7) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of FI810991L publication Critical patent/FI810991L/fi
Publication of FI810991A7 publication Critical patent/FI810991A7/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • A61K31/366Lactones having six-membered rings, e.g. delta-lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30Oxygen atoms, e.g. delta-lactones
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/02Oxygen as only ring hetero atoms
    • C12P17/06Oxygen as only ring hetero atoms containing a six-membered hetero ring, e.g. fluorescein

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
FI810991A 1980-03-31 1981-03-31 Kolesterolin biosynteesin inhibiitit, niiden valmistus ja käyttö. FI810991A7 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP55041292A JPH0692381B2 (ja) 1980-03-31 1980-03-31 Mb−530a誘導体

Publications (2)

Publication Number Publication Date
FI810991L FI810991L (fi) 1981-10-01
FI810991A7 true FI810991A7 (fi) 1981-10-01

Family

ID=12604367

Family Applications (1)

Application Number Title Priority Date Filing Date
FI810991A FI810991A7 (fi) 1980-03-31 1981-03-31 Kolesterolin biosynteesin inhibiitit, niiden valmistus ja käyttö.

Country Status (15)

Country Link
JP (1) JPH0692381B2 (enrdf_load_stackoverflow)
AT (1) ATA150781A (enrdf_load_stackoverflow)
AU (1) AU6893281A (enrdf_load_stackoverflow)
BE (1) BE888214A (enrdf_load_stackoverflow)
CH (1) CH646966A5 (enrdf_load_stackoverflow)
DE (2) DE3112566A1 (enrdf_load_stackoverflow)
DK (3) DK151273C (enrdf_load_stackoverflow)
FI (1) FI810991A7 (enrdf_load_stackoverflow)
FR (1) FR2479222A1 (enrdf_load_stackoverflow)
GB (1) GB2073193A (enrdf_load_stackoverflow)
IE (1) IE52367B1 (enrdf_load_stackoverflow)
IT (1) IT1144325B (enrdf_load_stackoverflow)
MX (1) MX9203567A (enrdf_load_stackoverflow)
NL (1) NL8101592A (enrdf_load_stackoverflow)
SE (1) SE461590B (enrdf_load_stackoverflow)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4472426A (en) * 1982-12-22 1984-09-18 Merck & Co., Inc. Antihypercholesterolemic compounds
EP0215665B1 (en) * 1985-09-13 1991-11-21 Sankyo Company Limited Hydroxy-ml-236b derivatives, their preparation and use
US4997848A (en) 1987-10-27 1991-03-05 Sankyo Company, Limited Octahydronaphthalene oxime derivatives for cholesterol synthesis inhibition
US5075327A (en) * 1988-08-10 1991-12-24 Hoffmann-La Roche Inc. Antipsoriatic agents
US5073568A (en) * 1988-11-14 1991-12-17 Hoffmann-La Roche Inc. Antipsoriatic agents
US5200549A (en) * 1988-11-14 1993-04-06 Hoffman-La Roche Inc. Antipsoriatic agents
US5021451A (en) * 1988-11-14 1991-06-04 Hoffman-La Roche Inc. Method for inhibiting hyperproliferative diseases
US5159104A (en) * 1991-05-01 1992-10-27 Merck & Co., Inc. Process to simvastatin ester
FR2937537A1 (fr) 2008-10-29 2010-04-30 Centre Nat Rech Scient Nanoparticules de statine
KR101820099B1 (ko) 2013-01-18 2018-01-18 에스프린팅솔루션 주식회사 저항 발열체, 이를 채용한 가열 부재, 및 정착 장치
AU2019207625A1 (en) * 2018-01-09 2020-07-30 Ligand Pharmaceuticals, Inc. Acetal compounds and therapeutic uses thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5612114B2 (enrdf_load_stackoverflow) * 1974-06-07 1981-03-18
JPS5925599B2 (ja) * 1979-02-20 1984-06-19 三共株式会社 新生理活性物質モナコリンkおよびその製造法
GR69216B (enrdf_load_stackoverflow) * 1979-06-15 1982-05-07 Merck & Co Inc
US4231938A (en) * 1979-06-15 1980-11-04 Merck & Co., Inc. Hypocholesteremic fermentation products and process of preparation
ZA81703B (en) * 1980-02-04 1982-09-29 Merck & Co Inc New antihypercholesterolemic compounds,intermediates and processes
PT72394B (en) * 1980-02-04 1982-09-06 Merck & Co Inc Process for preparing dihydro and tetrahydromevinoline hypocholesterolimics
AU548996B2 (en) * 1980-02-04 1986-01-09 Merck & Co., Inc. Tetrahydro-2h-pyran-2-one derivatives
US4282155A (en) * 1980-02-04 1981-08-04 Merck & Co., Inc. Antihypercholesterolemic compounds

Also Published As

Publication number Publication date
GB2073193A (en) 1981-10-14
SE8102047L (sv) 1981-10-01
JPH0692381B2 (ja) 1994-11-16
IE52367B1 (en) 1987-09-30
DK32290A (da) 1990-02-07
IT1144325B (it) 1986-10-29
FR2479222B1 (enrdf_load_stackoverflow) 1983-08-26
DK145481A (da) 1981-10-01
DK32190D0 (da) 1990-02-07
SE461590B (sv) 1990-03-05
MX9203567A (es) 1992-09-01
DK151273B (da) 1987-11-16
IT8167438A0 (it) 1981-03-30
DE3153666C2 (de) 1993-11-11
DK167805B1 (da) 1993-12-20
AU6893281A (en) 1981-10-08
DE3112566C2 (enrdf_load_stackoverflow) 1990-04-05
JPS56138181A (en) 1981-10-28
DK151273C (da) 1988-07-04
DK32190A (da) 1990-02-07
BE888214A (fr) 1981-09-30
FR2479222A1 (fr) 1981-10-02
DK32290D0 (da) 1990-02-07
IE810698L (en) 1981-09-30
CH646966A5 (de) 1984-12-28
ATA150781A (de) 1983-03-15
DE3112566A1 (de) 1982-03-11
FI810991L (fi) 1981-10-01
NL8101592A (nl) 1981-10-16

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Legal Events

Date Code Title Description
FA Application withdrawn [patent]

Owner name: SANKYO COMPANY LIMITED