FI103509B1 - Menetelmä uusien terapeuttisesti käyttökelpoisten 5-(2,5-disubstituoitu fenyyli)-1,3-dialkyyli-1,6-dihydro-7H-pyratsolo[4,3-d]pyrimidin-7-onien valmistamiseksi - Google Patents

Menetelmä uusien terapeuttisesti käyttökelpoisten 5-(2,5-disubstituoitu fenyyli)-1,3-dialkyyli-1,6-dihydro-7H-pyratsolo[4,3-d]pyrimidin-7-onien valmistamiseksi

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Publication number
FI103509B1
FI103509B1 FI923157A FI923157A FI103509B1 FI 103509 B1 FI103509 B1 FI 103509B1 FI 923157 A FI923157 A FI 923157A FI 923157 A FI923157 A FI 923157A FI 103509 B1 FI103509 B1 FI 103509B1
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FI
Finland
Prior art keywords
optionally substituted
alkyl
alkyl optionally
cycloalkyl
co2r
Prior art date
Application number
FI923157A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI103509B (fi
FI923157A (fi
FI923157A0 (fi
Inventor
Andrew Simon Bell
Nicholas Kenneth Terrett
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10698038&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI103509(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of FI923157A0 publication Critical patent/FI923157A0/fi
Publication of FI923157A publication Critical patent/FI923157A/fi
Priority to FI980420A priority Critical patent/FI980420A/fi
Application granted granted Critical
Publication of FI103509B publication Critical patent/FI103509B/fi
Publication of FI103509B1 publication Critical patent/FI103509B1/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Materials For Medical Uses (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FI923157A 1991-07-09 1992-07-08 Menetelmä uusien terapeuttisesti käyttökelpoisten 5-(2,5-disubstituoitu fenyyli)-1,3-dialkyyli-1,6-dihydro-7H-pyratsolo[4,3-d]pyrimidin-7-onien valmistamiseksi FI103509B1 (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI980420A FI980420A (fi) 1991-07-09 1998-02-24 Antianginaaliset pyratsolopyrimidinoniyhdisteet

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919114760A GB9114760D0 (en) 1991-07-09 1991-07-09 Therapeutic agents

Publications (4)

Publication Number Publication Date
FI923157A0 FI923157A0 (fi) 1992-07-08
FI923157A FI923157A (fi) 1993-01-10
FI103509B FI103509B (fi) 1999-07-15
FI103509B1 true FI103509B1 (fi) 1999-07-15

Family

ID=10698038

Family Applications (1)

Application Number Title Priority Date Filing Date
FI923157A FI103509B1 (fi) 1991-07-09 1992-07-08 Menetelmä uusien terapeuttisesti käyttökelpoisten 5-(2,5-disubstituoitu fenyyli)-1,3-dialkyyli-1,6-dihydro-7H-pyratsolo[4,3-d]pyrimidin-7-onien valmistamiseksi

Country Status (27)

Country Link
US (2) US5272147A (fr)
EP (1) EP0526004B1 (fr)
JP (1) JP2554824B2 (fr)
KR (1) KR950011739B1 (fr)
CN (1) CN1034503C (fr)
AT (1) ATE159019T1 (fr)
AU (1) AU636816B2 (fr)
BR (2) BR9202525A (fr)
CA (1) CA2073226C (fr)
CZ (1) CZ281316B6 (fr)
DE (1) DE69222595T2 (fr)
DK (1) DK0526004T3 (fr)
EG (1) EG19978A (fr)
ES (1) ES2107506T3 (fr)
FI (1) FI103509B1 (fr)
GB (1) GB9114760D0 (fr)
GR (1) GR3025424T3 (fr)
HU (2) HU220046B (fr)
IE (1) IE922222A1 (fr)
IL (1) IL102368A (fr)
MX (1) MX9204021A (fr)
NO (1) NO180750C (fr)
NZ (1) NZ243472A (fr)
PL (2) PL170893B1 (fr)
RU (1) RU2114113C1 (fr)
TW (1) TW358096B (fr)
ZA (1) ZA925084B (fr)

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EP0526004B1 (fr) 1997-10-08
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NZ243472A (en) 1993-12-23
BR9202525A (pt) 1993-03-16
HU220046B (hu) 2001-10-28
NO922685D0 (no) 1992-07-08
TW358096B (en) 1999-05-11
IE922222A1 (en) 1993-01-13
CZ210992A3 (en) 1993-10-13
CN1034503C (zh) 1997-04-09
AU636816B2 (en) 1993-05-06
CZ281316B6 (cs) 1996-08-14
HU9202267D0 (en) 1992-10-28
CA2073226C (fr) 1999-03-16
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BR1100029A (pt) 2000-06-06
MX9204021A (es) 1993-07-01
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NO180750C (no) 1997-06-11
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CN1068329A (zh) 1993-01-27
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US5272147A (en) 1993-12-21
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EP0526004A1 (fr) 1993-02-03
ATE159019T1 (de) 1997-10-15
GB9114760D0 (en) 1991-08-28
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