ES513128A0 - Un procediniento para la preparacion de nuevos derivados de acido acetamido penicilanico. - Google Patents

Un procediniento para la preparacion de nuevos derivados de acido acetamido penicilanico.

Info

Publication number
ES513128A0
ES513128A0 ES513128A ES513128A ES513128A0 ES 513128 A0 ES513128 A0 ES 513128A0 ES 513128 A ES513128 A ES 513128A ES 513128 A ES513128 A ES 513128A ES 513128 A0 ES513128 A0 ES 513128A0
Authority
ES
Spain
Prior art keywords
penicilanic
procedure
preparation
new derivatives
acetamide acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES513128A
Other languages
English (en)
Other versions
ES8307815A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of ES8307815A1 publication Critical patent/ES8307815A1/es
Publication of ES513128A0 publication Critical patent/ES513128A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
ES513128A 1981-06-16 1982-06-15 Un procediniento para la preparacion de nuevos derivados de acido acetamido penicilanico. Granted ES513128A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8118552 1981-06-16

Publications (2)

Publication Number Publication Date
ES8307815A1 ES8307815A1 (es) 1983-08-01
ES513128A0 true ES513128A0 (es) 1983-08-01

Family

ID=10522555

Family Applications (1)

Application Number Title Priority Date Filing Date
ES513128A Granted ES513128A0 (es) 1981-06-16 1982-06-15 Un procediniento para la preparacion de nuevos derivados de acido acetamido penicilanico.

Country Status (6)

Country Link
US (1) US4447422A (es)
EP (1) EP0067610A1 (es)
JP (1) JPS5821681A (es)
AU (1) AU8493182A (es)
ES (1) ES513128A0 (es)
ZA (1) ZA824052B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3479731D1 (en) * 1983-07-07 1989-10-19 Beecham Group Plc Substituted phenylglycine derivatives of beta-lactam antibiotics
US4684643A (en) * 1983-08-22 1987-08-04 Eli Lilly And Company Pharmaceutical compositions for storage in plastic containers and process therefor
US4533542A (en) * 1983-08-22 1985-08-06 Eli Lilly And Company Pharmaceutical compositions for storage in plastic containers and process therefor
JPS62161123U (es) * 1986-04-02 1987-10-13
TWI618707B (zh) * 2009-10-16 2018-03-21 梅林塔療法公司 抗微生物性化合物,及製法及其用途
WO2011047323A2 (en) 2009-10-16 2011-04-21 Rib-X Pharmaceuticals, Inc. Antimicrobial compounds and methods of making and using the same
WO2013163159A2 (en) * 2012-04-24 2013-10-31 Board Of Trustees Of Northern Illinois University Design and synthesis of novel inhibitors of isoprenoid biosynthesis
SG11201601654TA (en) 2013-09-09 2016-04-28 Melinta Therapeutics Inc Antimicrobial compunds and methods of making and using the same
MX2016003046A (es) 2013-09-09 2016-09-08 Melinta Therapeutics Inc Compuestos antimicrobianos y métodos de fabricación y utilización de los mismos.
CA2979342A1 (en) 2015-03-11 2016-09-15 Melinta Therapeutics, Inc. Antimicrobial compounds and methods of making and using the same
WO2017193016A1 (en) 2016-05-06 2017-11-09 Melinta Therapeutics, Inc. Antimicrobials and methods of making and using same
US10155766B2 (en) 2016-06-14 2018-12-18 Board Of Trustees Of Northern Illinois University Pyrazolopyrimidine antibacterial agents

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR208171A1 (es) * 1972-09-29 1976-12-09 Ciba Geigy Ag Procedimiento para la obtencion de nuevos derivados del acido cef-3-em-4-carboxilico
ES477520A1 (es) * 1978-02-25 1979-06-01 Thomae Gmbh Dr K Procedimiento para la preparacion de nuevas penicilinas.
JPS5573686A (en) * 1978-11-28 1980-06-03 Mitsui Toatsu Chem Inc Novel penicillin
US4267180A (en) * 1979-03-12 1981-05-12 Warner-Lambert Company Novel antibacterial amide compounds and process means for producing the same
US4315933A (en) * 1980-09-24 1982-02-16 Warner-Lambert Company Antibacterial amide compounds and pharmaceutical compositions containing the same

Also Published As

Publication number Publication date
EP0067610A1 (en) 1982-12-22
JPS5821681A (ja) 1983-02-08
ES8307815A1 (es) 1983-08-01
AU8493182A (en) 1982-12-23
ZA824052B (en) 1983-03-30
US4447422A (en) 1984-05-08

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