ES2341510T3 - Microemulsiones como formas farmaceuticas solidas para la administracion oral. - Google Patents
Microemulsiones como formas farmaceuticas solidas para la administracion oral. Download PDFInfo
- Publication number
- ES2341510T3 ES2341510T3 ES99941159T ES99941159T ES2341510T3 ES 2341510 T3 ES2341510 T3 ES 2341510T3 ES 99941159 T ES99941159 T ES 99941159T ES 99941159 T ES99941159 T ES 99941159T ES 2341510 T3 ES2341510 T3 ES 2341510T3
- Authority
- ES
- Spain
- Prior art keywords
- microemulsion
- drug
- solid
- pharmaceutical form
- solid pharmaceutical
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0007—Effervescent
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/143—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with inorganic compounds
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Dispersion Chemistry (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9634798P | 1998-08-13 | 1998-08-13 | |
| US96347P | 1998-08-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2341510T3 true ES2341510T3 (es) | 2010-06-21 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES99941159T Expired - Lifetime ES2341510T3 (es) | 1998-08-13 | 1999-08-13 | Microemulsiones como formas farmaceuticas solidas para la administracion oral. |
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|---|---|
| US (1) | US6280770B1 (https=) |
| EP (2) | EP2127642A3 (https=) |
| JP (1) | JP4815053B2 (https=) |
| AT (1) | ATE462417T1 (https=) |
| AU (1) | AU5486899A (https=) |
| CA (1) | CA2339991C (https=) |
| DE (1) | DE69942205D1 (https=) |
| ES (1) | ES2341510T3 (https=) |
| WO (1) | WO2000009093A1 (https=) |
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| US6350470B1 (en) * | 1998-04-29 | 2002-02-26 | Cima Labs Inc. | Effervescent drug delivery system for oral administration |
| US6793934B1 (en) | 1999-12-08 | 2004-09-21 | Shire Laboratories, Inc. | Solid oral dosage form |
| AUPQ573300A0 (en) | 2000-02-21 | 2000-03-16 | Australian Nuclear Science & Technology Organisation | Controlled release ceramic particles, compositions thereof, processes of preparation and methods of use |
| GB0008785D0 (en) * | 2000-04-10 | 2000-05-31 | Novartis Ag | Organic compounds |
| EP1318790A4 (en) * | 2000-09-19 | 2006-02-01 | Cima Labs Inc | PHARMACEUTICAL COMPOSITIONS FOR RECTAL AND VAGINAL ADMINISTRATION |
| US7799342B2 (en) * | 2000-12-06 | 2010-09-21 | Wyeth Llc | Fast dissolving tablet |
| WO2002083102A1 (en) * | 2001-02-23 | 2002-10-24 | Cima Labs Inc. | Emulsions as solid dosage forms for oral administration |
| US6692771B2 (en) | 2001-02-23 | 2004-02-17 | Cima Labs Inc. | Emulsions as solid dosage forms for oral administration |
| EE200400034A (et) * | 2001-06-22 | 2004-06-15 | Pfizer Products Inc. | Amorfse ravimaine adsorbaatide farmatseutilised kompositsioonid |
| US20030068356A1 (en) | 2001-07-10 | 2003-04-10 | Pather S. Indiran | Sequential drug delivery systems |
| ITMI20011756A1 (it) * | 2001-08-09 | 2003-02-09 | Remedia S R L | Composizione farmaceutica comprendente una microemulsione doppia acqua/olio/acqua incorporata in un supporto solido |
| US20030083286A1 (en) * | 2001-08-22 | 2003-05-01 | Ching-Leou Teng | Bioadhesive compositions and methods for enhanced intestinal drug absorption |
| US20030124196A1 (en) * | 2001-08-22 | 2003-07-03 | Susan Weinbach | Pulsatile release compositions and methods for enhanced intestinal drug absorption |
| BR0214679A (pt) * | 2001-12-03 | 2004-12-14 | Novacea Inc | Composições farmacêuticas compreendendo compostos a base de vitamina d ativa |
| ITMI20012694A1 (it) * | 2001-12-19 | 2003-06-19 | Remedia S R L | Composizione farmaceutica comprendente una microemulsione doppia olio/acqua/olio incorporata in un supporto solido |
| ATE395044T1 (de) | 2002-02-01 | 2008-05-15 | Pfizer Prod Inc | Pharmazeutische zusammensetzungen amorpher dispersionen von wirkstoffen und lipophiler mikrophasenbildender materialien |
| ITMI20021392A1 (it) * | 2002-06-25 | 2003-12-29 | Nicox Sa | Forme farmaceutiche per la somministrazione orale di farmaci liquidi a temperatura ambiente dotate di migliore biodisponibilita' |
| WO2004002443A1 (en) * | 2002-06-26 | 2004-01-08 | Tuo Jin | Solid dosage forms for rapid dissolution of poorly soluble drugs |
| US20040115226A1 (en) * | 2002-12-12 | 2004-06-17 | Wenji Li | Free-flowing solid formulations with improved bio-availability of poorly water soluble drugs and process for making the same |
| FR2851918B1 (fr) * | 2003-03-06 | 2006-06-16 | Poudre impregnee ameliorant la biodisponibilite et/ou la solubilite et procede de fabrication | |
| JP2007501218A (ja) * | 2003-08-04 | 2007-01-25 | ファイザー・プロダクツ・インク | 非晶質薬物の吸着物および親油性ミクロ相形成物質の医薬組成物 |
| US7390503B1 (en) | 2003-08-22 | 2008-06-24 | Barr Laboratories, Inc. | Ondansetron orally disintegrating tablets |
| JP5179757B2 (ja) * | 2004-02-17 | 2013-04-10 | トランセプト ファーマシューティカルズ， インコーポレイティド | 口腔粘膜を介して催眠剤をデリバリーするための組成物及びその使用方法 |
| US20050220866A1 (en) * | 2004-04-02 | 2005-10-06 | Dr. Reddy's Laboratories Limited | Novel capsule formulations of etoposide for oral use |
| WO2005105040A2 (en) * | 2004-04-26 | 2005-11-10 | Micelle Products, Inc. | Water-soluble formulations of fat soluble vitamins and pharmaceutical agents and their applications |
| US20060014677A1 (en) * | 2004-07-19 | 2006-01-19 | Isotechnika International Inc. | Method for maximizing efficacy and predicting and minimizing toxicity of calcineurin inhibitor compounds |
| ATE533473T1 (de) | 2004-09-24 | 2011-12-15 | Boehringer Ingelheim Pharma | Neue klasse von surfuctantähnlichen materialien mit vitamin-e-tpgs und wasserlöslichem polymer |
| WO2006085217A2 (en) * | 2005-02-08 | 2006-08-17 | Pfizer Products Inc. | Solid adsorbates of hydrophobic drugs |
| US8492369B2 (en) | 2010-04-12 | 2013-07-23 | Clarus Therapeutics Inc | Oral testosterone ester formulations and methods of treating testosterone deficiency comprising same |
| CA2604943C (en) | 2005-04-15 | 2013-09-17 | Clarus Therapeutics, Inc. | Pharmaceutical delivery systems for hydrophobic drugs and compositions comprising same |
| US20070225322A1 (en) * | 2005-05-25 | 2007-09-27 | Transoral Pharmaceuticals, Inc. | Compositions and methods for treating middle-of-the night insomnia |
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| EP1883408A4 (en) * | 2005-05-25 | 2009-11-11 | Transcept Pharmaceuticals Inc | SOLID COMPOSITIONS AND METHODS FOR TREATMENT OF INSOMNIA IN THE NIGHT |
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-
1999
- 1999-08-13 EP EP09011793A patent/EP2127642A3/en not_active Withdrawn
- 1999-08-13 DE DE69942205T patent/DE69942205D1/de not_active Expired - Lifetime
- 1999-08-13 CA CA002339991A patent/CA2339991C/en not_active Expired - Fee Related
- 1999-08-13 JP JP2000564596A patent/JP4815053B2/ja not_active Expired - Fee Related
- 1999-08-13 AU AU54868/99A patent/AU5486899A/en not_active Abandoned
- 1999-08-13 EP EP99941159A patent/EP1104290B1/en not_active Expired - Lifetime
- 1999-08-13 ES ES99941159T patent/ES2341510T3/es not_active Expired - Lifetime
- 1999-08-13 AT AT99941159T patent/ATE462417T1/de not_active IP Right Cessation
- 1999-08-13 US US09/374,393 patent/US6280770B1/en not_active Expired - Lifetime
- 1999-08-13 WO PCT/US1999/018552 patent/WO2000009093A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| ATE462417T1 (de) | 2010-04-15 |
| CA2339991A1 (en) | 2000-02-24 |
| EP1104290B1 (en) | 2010-03-31 |
| JP4815053B2 (ja) | 2011-11-16 |
| EP1104290A1 (en) | 2001-06-06 |
| WO2000009093A1 (en) | 2000-02-24 |
| US6280770B1 (en) | 2001-08-28 |
| EP2127642A3 (en) | 2010-02-24 |
| AU5486899A (en) | 2000-03-06 |
| JP2002522473A (ja) | 2002-07-23 |
| DE69942205D1 (de) | 2010-05-12 |
| CA2339991C (en) | 2007-01-02 |
| EP1104290A4 (en) | 2006-01-18 |
| EP2127642A2 (en) | 2009-12-02 |
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