ES2074224T3 - Nuevos intermedios de cefalosporina y proceso para preparar los intermedios y sus productos finales. - Google Patents
Nuevos intermedios de cefalosporina y proceso para preparar los intermedios y sus productos finales.Info
- Publication number
- ES2074224T3 ES2074224T3 ES91302486T ES91302486T ES2074224T3 ES 2074224 T3 ES2074224 T3 ES 2074224T3 ES 91302486 T ES91302486 T ES 91302486T ES 91302486 T ES91302486 T ES 91302486T ES 2074224 T3 ES2074224 T3 ES 2074224T3
- Authority
- ES
- Spain
- Prior art keywords
- intermediates
- cephalosporin
- alkyl
- final products
- prepare
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
ESTA INVENCION PROPORCIONA NUEVOS DERIVADOS DE CEFALOSPORINA REPRESENTADOS POR LA SIGUIENTE FORMULA (1), QUE SON ESPECIALMENTE UTILES COMO INTERMEDIARIOS PARA LA PREPARACION DE COMPUESTOS DE CEFALOSPORINA DOTADOS CON UNAS ACTIVIDADES ANTIBACTERIANAS POTENTES Y AMPLIAS. DONDE: R ELEVADO 1 UN ALQUILO C SUB 1-4, ALQUENILO C SUB 3-4, CICLOALQUILO C SUB 3-4, AMINO OPCIONALMENTE SUSTITUIDO CON UN RADICAL ALQUILO C SUB 1-4, O GRUPO FENILO OPCIONALMENTE SUSTITUIDO EN SU POSICION 2-, 4 UN HALOGENO, ALQUILO C SUB 1-4, ALCOXI C SUB 1-3 O RADICAL HIDROXI; R (AL CUADRADO) ES HIDROGENO O UN GRUPO ALQUILO C SUB 1-4; Y N ES BIEN 0 O 1. LA INVENCION TAMBIEN SE REFIERE A UN PROCESO PARA PREPARAR ESTOS INTERMEDIARIOS Y SUS ANTIBIOTICOS FARMACOLOGICAMENTE ACTIVOS DE CEFALOSPORINA ACTIVA.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR1019900003994A KR920004822B1 (ko) | 1990-03-24 | 1990-03-24 | 세팔로스포린계 화합물 및 그의 제조방법 |
KR1019900022332A KR930001116B1 (ko) | 1990-12-29 | 1990-12-29 | 세팔로스포린 중간체의 제조방법 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2074224T3 true ES2074224T3 (es) | 1995-09-01 |
Family
ID=26628215
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES91302486T Expired - Lifetime ES2074224T3 (es) | 1990-03-24 | 1991-03-21 | Nuevos intermedios de cefalosporina y proceso para preparar los intermedios y sus productos finales. |
Country Status (7)
Country | Link |
---|---|
US (1) | US5142041A (es) |
EP (1) | EP0449515B1 (es) |
JP (1) | JPH04217987A (es) |
AT (1) | ATE123034T1 (es) |
DE (1) | DE69109913T2 (es) |
DK (1) | DK0449515T3 (es) |
ES (1) | ES2074224T3 (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5202315A (en) * | 1989-05-11 | 1993-04-13 | Lucky, Ltd. | Cephalosporin compounds |
KR930007264B1 (ko) * | 1990-08-17 | 1993-08-04 | 주식회사 럭키 | 신규한 세팔로스포린 화합물과 그의 제조방법 |
EP0508375A3 (en) * | 1991-04-12 | 1992-12-09 | Lucky Ltd. | Novel cephalosporin compounds and processes for preparation thereof |
KR970010069B1 (ko) * | 1992-08-24 | 1997-06-20 | 주식회사 럭키 | 신규 세팔로스포린계 항생제 및 이의 제조방법 |
KR970005896B1 (ko) * | 1993-07-23 | 1997-04-21 | 주식회사 엘지화학 | 신규 세팔로스포린계 항생제 및 그의 제조방법 |
EP0638573A1 (en) * | 1993-08-10 | 1995-02-15 | Lucky Ltd. | Crystalline hydrates of cephalosporin and process for preparation thereof |
AT403284B (de) * | 1996-04-23 | 1997-12-29 | Biochemie Gmbh | 3-methylimino-3-cephemderivate |
AT403283B (de) * | 1996-04-17 | 1997-12-29 | Biochemie Gmbh | 3-methylimino-3-cephemderivate |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2716677C2 (de) * | 1977-04-15 | 1985-10-10 | Hoechst Ag, 6230 Frankfurt | Cephemderivate und Verfahren zu ihrer Herstellung |
AR231986A1 (es) * | 1978-05-26 | 1985-04-30 | Glaxo Group Ltd | Procedimiento para preparar antibioticos de cefalosporina |
GB1604723A (en) * | 1978-05-26 | 1981-12-16 | Glaxo Operations Ltd | 7-(2-aminothiazol-4-yl)-2-oxyimino-acetamido)-cephem derivatives |
DE3006888A1 (de) * | 1980-02-23 | 1981-09-10 | Hoechst Ag, 6000 Frankfurt | Cephalosporinderivate und verfahren zu ihrer herstellung |
JPS59106492A (ja) * | 1982-11-24 | 1984-06-20 | グラクソ・グル−プ・リミテツド | セフアロスポリン抗生物質 |
JPS61267584A (ja) * | 1985-01-16 | 1986-11-27 | Fujisawa Pharmaceut Co Ltd | セフアロスポラン酸誘導体もしくはその薬理学的に許容しうる塩 |
JPS63107989A (ja) * | 1986-06-04 | 1988-05-12 | Tanabe Seiyaku Co Ltd | セファロスポリン化合物 |
US5202315A (en) * | 1989-05-11 | 1993-04-13 | Lucky, Ltd. | Cephalosporin compounds |
-
1991
- 1991-03-21 AT AT91302486T patent/ATE123034T1/de not_active IP Right Cessation
- 1991-03-21 ES ES91302486T patent/ES2074224T3/es not_active Expired - Lifetime
- 1991-03-21 EP EP91302486A patent/EP0449515B1/en not_active Expired - Lifetime
- 1991-03-21 DK DK91302486.5T patent/DK0449515T3/da active
- 1991-03-21 DE DE69109913T patent/DE69109913T2/de not_active Expired - Fee Related
- 1991-03-22 US US07/673,673 patent/US5142041A/en not_active Expired - Fee Related
- 1991-03-22 JP JP3058790A patent/JPH04217987A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
DE69109913T2 (de) | 1995-12-07 |
DK0449515T3 (da) | 1995-10-16 |
EP0449515A3 (en) | 1992-06-17 |
JPH04217987A (ja) | 1992-08-07 |
US5142041A (en) | 1992-08-25 |
DE69109913D1 (de) | 1995-06-29 |
ATE123034T1 (de) | 1995-06-15 |
EP0449515A2 (en) | 1991-10-02 |
EP0449515B1 (en) | 1995-05-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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