EP1922072A4 - Melanocortin receptor-specific piperazine compounds with diamine groups - Google Patents
Melanocortin receptor-specific piperazine compounds with diamine groupsInfo
- Publication number
- EP1922072A4 EP1922072A4 EP06813393A EP06813393A EP1922072A4 EP 1922072 A4 EP1922072 A4 EP 1922072A4 EP 06813393 A EP06813393 A EP 06813393A EP 06813393 A EP06813393 A EP 06813393A EP 1922072 A4 EP1922072 A4 EP 1922072A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- melanocortin receptor
- piperazine compounds
- diamine groups
- specific piperazine
- specific
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/04—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Gynecology & Obstetrics (AREA)
- Neurosurgery (AREA)
- Nutrition Science (AREA)
- Neurology (AREA)
- Pregnancy & Childbirth (AREA)
- Biomedical Technology (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70748805P | 2005-08-11 | 2005-08-11 | |
PCT/US2006/031472 WO2007021990A2 (en) | 2005-08-11 | 2006-08-11 | Melanocortin receptor-specific piperazine compounds with diamine groups |
Publications (2)
Publication Number | Publication Date |
---|---|
EP1922072A2 EP1922072A2 (en) | 2008-05-21 |
EP1922072A4 true EP1922072A4 (en) | 2010-12-29 |
Family
ID=37758229
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP06813394A Withdrawn EP1919479A4 (en) | 2005-08-11 | 2006-08-11 | Melanocortin receptor-specific piperazine and keto-piperazine compounds |
EP06813393A Withdrawn EP1922072A4 (en) | 2005-08-11 | 2006-08-11 | Melanocortin receptor-specific piperazine compounds with diamine groups |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP06813394A Withdrawn EP1919479A4 (en) | 2005-08-11 | 2006-08-11 | Melanocortin receptor-specific piperazine and keto-piperazine compounds |
Country Status (4)
Country | Link |
---|---|
EP (2) | EP1919479A4 (en) |
JP (2) | JP2009504671A (en) |
CN (2) | CN101272788A (en) |
WO (2) | WO2007021990A2 (en) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7727991B2 (en) | 2003-05-01 | 2010-06-01 | Palatin Technologies, Inc. | Substituted melanocortin receptor-specific single acyl piperazine compounds |
WO2007021990A2 (en) * | 2005-08-11 | 2007-02-22 | Palatin Technologies, Inc. | Melanocortin receptor-specific piperazine compounds with diamine groups |
WO2008090357A2 (en) * | 2007-01-24 | 2008-07-31 | Palatin Technologies, Inc. | N, n; -substituted piperazines binding to melanocortin receptor |
WO2009144432A1 (en) * | 2008-05-30 | 2009-12-03 | Palatin Technologies, Inc. | Mc4-r agonists for the treatment of obesity |
ES2869229T3 (en) * | 2015-11-27 | 2021-10-25 | Mitsubishi Tanabe Pharma Corp | 2 - (((pyrrolidin-3-yl) carbonyl) amino) -1H-imidazole derivatives as melanocortin receptor 1 (MCR1) agonists to treat rheumatoid arthritis |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20040157264A1 (en) * | 2001-08-10 | 2004-08-12 | Palatin Technologies, Inc. | Piperazine melanocortin-specific compounds |
US20050130988A1 (en) * | 2001-08-10 | 2005-06-16 | Palatin Technologies, Inc. | Naphthalene-containing melanocortin receptor-specific small molecule |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7456184B2 (en) * | 2003-05-01 | 2008-11-25 | Palatin Technologies Inc. | Melanocortin receptor-specific compounds |
WO2004078716A1 (en) * | 2003-03-03 | 2004-09-16 | Merck & Co. Inc. | Acylated piperazine derivatives as melanocortin-4 receptor agonists |
WO2007021990A2 (en) * | 2005-08-11 | 2007-02-22 | Palatin Technologies, Inc. | Melanocortin receptor-specific piperazine compounds with diamine groups |
-
2006
- 2006-08-11 WO PCT/US2006/031472 patent/WO2007021990A2/en active Application Filing
- 2006-08-11 EP EP06813394A patent/EP1919479A4/en not_active Withdrawn
- 2006-08-11 JP JP2008526249A patent/JP2009504671A/en active Pending
- 2006-08-11 JP JP2008526250A patent/JP2009504672A/en active Pending
- 2006-08-11 CN CNA2006800353276A patent/CN101272788A/en active Pending
- 2006-08-11 EP EP06813393A patent/EP1922072A4/en not_active Withdrawn
- 2006-08-11 WO PCT/US2006/031474 patent/WO2007021991A2/en active Application Filing
- 2006-08-11 CN CNA2006800353810A patent/CN101272789A/en active Pending
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20040157264A1 (en) * | 2001-08-10 | 2004-08-12 | Palatin Technologies, Inc. | Piperazine melanocortin-specific compounds |
US20050130988A1 (en) * | 2001-08-10 | 2005-06-16 | Palatin Technologies, Inc. | Naphthalene-containing melanocortin receptor-specific small molecule |
Also Published As
Publication number | Publication date |
---|---|
CN101272788A (en) | 2008-09-24 |
JP2009504671A (en) | 2009-02-05 |
JP2009504672A (en) | 2009-02-05 |
WO2007021990A2 (en) | 2007-02-22 |
CN101272789A (en) | 2008-09-24 |
EP1919479A2 (en) | 2008-05-14 |
EP1919479A4 (en) | 2010-11-17 |
EP1922072A2 (en) | 2008-05-21 |
WO2007021991A2 (en) | 2007-02-22 |
WO2007021990A3 (en) | 2007-08-09 |
WO2007021991A3 (en) | 2007-07-12 |
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Legal Events
Date | Code | Title | Description |
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PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
17P | Request for examination filed |
Effective date: 20080222 |
|
AK | Designated contracting states |
Kind code of ref document: A2 Designated state(s): AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR |
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REG | Reference to a national code |
Ref country code: HK Ref legal event code: DE Ref document number: 1117062 Country of ref document: HK |
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A4 | Supplementary search report drawn up and despatched |
Effective date: 20101130 |
|
RIC1 | Information provided on ipc code assigned before grant |
Ipc: C07D 241/14 20060101ALI20101124BHEP Ipc: A61P 15/10 20060101ALI20101124BHEP Ipc: C07D 241/04 20060101ALI20101124BHEP Ipc: A61K 31/496 20060101AFI20080318BHEP |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
18D | Application deemed to be withdrawn |
Effective date: 20110301 |
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REG | Reference to a national code |
Ref country code: HK Ref legal event code: WD Ref document number: 1117062 Country of ref document: HK |