Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Темпест Терапьютикс, Инк.filedCriticalТемпест Терапьютикс, Инк.
Priority claimed from PCT/US2019/027992external-prioritypatent/WO2019204523A1/en
Publication of EA202092273A1publicationCriticalpatent/EA202092273A1/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
Соединения, композиции и способы представлены для модуляции активности рецепторов EP2 и EP4 и для лечения, предупреждения и облегчения одного или более симптомов заболеваний или нарушений, связанных с активностью рецепторов EP2 и EP4. Согласно некоторым вариантам осуществления соединения представляют собой антагонисты обоих рецепторов EP2 и EP4.Compounds, compositions and methods are provided for modulating the activity of EP2 and EP4 receptors and for treating, preventing and ameliorating one or more symptoms of diseases or disorders associated with the activity of EP2 and EP4 receptors. In some embodiments, the compounds are antagonists of both EP2 and EP4 receptors.
EA202092273A2018-10-172019-04-17
BICYCLIC CARBOXAMIDES AND METHODS OF THEIR APPLICATION
EA202092273A1
(en)