EA200900344A1 - Циклические ингибиторы 11-бета-гидроксистероиддегидрогеназы типа i - Google Patents
Циклические ингибиторы 11-бета-гидроксистероиддегидрогеназы типа iInfo
- Publication number
- EA200900344A1 EA200900344A1 EA200900344A EA200900344A EA200900344A1 EA 200900344 A1 EA200900344 A1 EA 200900344A1 EA 200900344 A EA200900344 A EA 200900344A EA 200900344 A EA200900344 A EA 200900344A EA 200900344 A1 EA200900344 A1 EA 200900344A1
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- EA
- Eurasian Patent Office
- Prior art keywords
- beta
- inhibitors
- hydroxysteroid dehydrogenase
- type
- dehydrogenase type
- Prior art date
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Abstract
Обеспечены новые соединения, которые являются ингибиторами 11-бета-гидроксистероиддегидрогеназы типа I. Ингибиторы 11-бета-гидроксистероиддегидрогеназы типа I являются полезными при лечении, профилактике или подавлении прогрессирования заболеваний, требующих терапию ингибитором 11-бета-гидроксистероиддегидрогеназы типа I. Указанные новые соединения имеют структуру (I), их энантиомеры, диастереомеры, сольваты или соли, где A, W, Х и Z являются теми, как определено в настоящем описании.
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US11/843,015 US7727978B2 (en) | 2006-08-24 | 2007-08-22 | Cyclic 11-beta hydroxysteroid dehydrogenase type I inhibitors |
PCT/US2007/076593 WO2008024892A2 (en) | 2006-08-24 | 2007-08-23 | Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors |
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EA200900344A1 true EA200900344A1 (ru) | 2009-10-30 |
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JP (2) | JP5268912B2 (ru) |
KR (1) | KR20090057038A (ru) |
CN (1) | CN103833544A (ru) |
AR (1) | AR062533A1 (ru) |
AU (1) | AU2007286629A1 (ru) |
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NO (1) | NO20090445L (ru) |
TW (1) | TW200817353A (ru) |
WO (1) | WO2008024892A2 (ru) |
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-
2007
- 2007-08-22 US US11/843,015 patent/US7727978B2/en active Active
- 2007-08-23 CN CN201410057480.5A patent/CN103833544A/zh active Pending
- 2007-08-23 BR BRPI0715839-4A patent/BRPI0715839A2/pt not_active IP Right Cessation
- 2007-08-23 EA EA200900344A patent/EA200900344A1/ru unknown
- 2007-08-23 WO PCT/US2007/076593 patent/WO2008024892A2/en active Application Filing
- 2007-08-23 JP JP2009525773A patent/JP5268912B2/ja not_active Expired - Fee Related
- 2007-08-23 KR KR1020097005903A patent/KR20090057038A/ko not_active Application Discontinuation
- 2007-08-23 CA CA002661401A patent/CA2661401A1/en not_active Abandoned
- 2007-08-23 EP EP20120181050 patent/EP2527317A1/en not_active Withdrawn
- 2007-08-23 AU AU2007286629A patent/AU2007286629A1/en not_active Abandoned
- 2007-08-23 MX MX2009001687A patent/MX2009001687A/es active IP Right Grant
- 2007-08-23 EP EP07814376.5A patent/EP2054368B1/en active Active
- 2007-08-24 AR ARP070103783A patent/AR062533A1/es not_active Application Discontinuation
- 2007-08-24 CL CL2007002492A patent/CL2007002492A1/es unknown
- 2007-08-24 TW TW096131558A patent/TW200817353A/zh unknown
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2009
- 2009-01-29 NO NO20090445A patent/NO20090445L/no not_active Application Discontinuation
- 2009-02-11 IL IL196989A patent/IL196989A0/en unknown
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2010
- 2010-04-14 US US12/759,867 patent/US8299054B2/en active Active
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Also Published As
Publication number | Publication date |
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CN103833544A (zh) | 2014-06-04 |
TW200817353A (en) | 2008-04-16 |
AR062533A1 (es) | 2008-11-12 |
US8299054B2 (en) | 2012-10-30 |
US7727978B2 (en) | 2010-06-01 |
JP2013173783A (ja) | 2013-09-05 |
IL196989A0 (en) | 2009-11-18 |
WO2008024892A3 (en) | 2008-12-11 |
EP2054368B1 (en) | 2015-09-16 |
KR20090057038A (ko) | 2009-06-03 |
CL2007002492A1 (es) | 2008-01-11 |
CA2661401A1 (en) | 2008-02-28 |
EP2527317A1 (en) | 2012-11-28 |
WO2008024892A2 (en) | 2008-02-28 |
MX2009001687A (es) | 2009-02-25 |
US20080234249A1 (en) | 2008-09-25 |
AU2007286629A1 (en) | 2008-02-28 |
US20100204199A1 (en) | 2010-08-12 |
NO20090445L (no) | 2009-02-26 |
BRPI0715839A2 (pt) | 2013-07-23 |
JP2010501589A (ja) | 2010-01-21 |
JP5268912B2 (ja) | 2013-08-21 |
EP2054368A2 (en) | 2009-05-06 |
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