EA200500881A1 - N-арилсульфонил-3-замещенные индолы, обладающие афинностью к серотониновому рецептору, способ их получения и содержащая их фармацевтическая композиция - Google Patents

N-арилсульфонил-3-замещенные индолы, обладающие афинностью к серотониновому рецептору, способ их получения и содержащая их фармацевтическая композиция

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EA200500881A1
EA200500881A1 EA200500881A EA200500881A EA200500881A1 EA 200500881 A1 EA200500881 A1 EA 200500881A1 EA 200500881 A EA200500881 A EA 200500881A EA 200500881 A EA200500881 A EA 200500881A EA 200500881 A1 EA200500881 A1 EA 200500881A1
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arylsulphone
affinity
receiving
pharmaceutical composition
serotonin receptor
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EA200500881A
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English (en)
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EA011320B1 (ru
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Венката Сатья Нироги Рамакришна
Викас Шрикришна Ширсатх
Рама Састри Камбхампати
Венката Сатья Веерабхадра Вадламуди Рао
Венкатесварлу Джасти
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Сувен Лайф Сайенсиз Лимитед
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Publication of EA200500881A1 publication Critical patent/EA200500881A1/ru
Publication of EA011320B1 publication Critical patent/EA011320B1/ru

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Abstract

Настоящее изобретение относится к новым N-арилсульфонил-3-замещенным индольным соединениям, их производным, их аналогам, их таутомерным формам, их стереоизомерам, их геометрическим формам, их N-оксидам, их полиморфам, их фармацевтически приемлемым солям, их фармацевтически приемлемым сольватам и содержащим их фармацевтически приемлемым композициям. Настоящее изобретение, в частности, относится к новым N-арилсульфонил-3-замещенным индолам общей формулы (I), их производным, их аналогам, их таутомерным формам, их стереоизомерам, их геометрическим формам, их полиморфам, их фармацевтически приемлемым солям, их фармацевтически приемлемым сольватам и содержащим их фармацевтически приемлемым композициям. Настоящее изобретение также относится к способу получения соединений общей формулы (I), фармацевтических композиций, содержащих такие соединения, и к применению таких соединений и композиций в медицине. Настоящее изобретение также относится к новым используемым промежуточным соединениям и к способу их получения.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200500881A 2002-11-28 2003-06-05 N-арилсульфонил-3-замещенные индолы, обладающие афинностью к серотониновому рецептору, способ их получения и содержащая их фармацевтическая композиция EA011320B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN884MA2002 2002-11-28
PCT/IN2003/000209 WO2004048330A1 (en) 2002-11-28 2003-06-05 N-arylsulfonyl-3-substituted indoles having serotonin receptor affinity, process for their preparation and pharmaceutical composition containing them

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EA200500881A1 true EA200500881A1 (ru) 2005-12-29
EA011320B1 EA011320B1 (ru) 2009-02-27

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US (1) US7875605B2 (ru)
EP (1) EP1581492B1 (ru)
JP (1) JP4559230B2 (ru)
KR (1) KR100818508B1 (ru)
CN (2) CN1720225B (ru)
AT (1) ATE401307T1 (ru)
AU (1) AU2003237599B2 (ru)
BR (2) BRPI0318799B8 (ru)
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DK (1) DK1581492T3 (ru)
EA (1) EA011320B1 (ru)
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NO (2) NO330341B1 (ru)
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PT (1) PT1581492E (ru)
SI (1) SI1581492T1 (ru)
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