EA199900352A1 - Композиции жидкого алендроната - Google Patents
Композиции жидкого алендронатаInfo
- Publication number
- EA199900352A1 EA199900352A1 EA199900352A EA199900352A EA199900352A1 EA 199900352 A1 EA199900352 A1 EA 199900352A1 EA 199900352 A EA199900352 A EA 199900352A EA 199900352 A EA199900352 A EA 199900352A EA 199900352 A1 EA199900352 A1 EA 199900352A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- liquid
- alandronate
- compositions
- composition
- hcl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
- A61K31/663—Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Physical Education & Sports Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Rheumatology (AREA)
- Epidemiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Жидкая композиция алендроновой кислоты или фармацевтически приемлемой соли имеет достаточные буферные свойства, так что рН композиции равняется 4-7,5, и 15 мл композиции может увеличить рН 50 мл 0,1 н HCl от 1 до, по крайней мере, 3, предпочтительно до 4.Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2676596P | 1996-10-04 | 1996-10-04 | |
GBGB9700541.7A GB9700541D0 (en) | 1997-01-13 | 1997-01-13 | Liquid alendronate formulation |
US3600297P | 1997-01-22 | 1997-01-22 | |
PCT/US1997/015740 WO1998014196A1 (en) | 1996-10-04 | 1997-10-02 | Liquid alendronate formulations |
Publications (2)
Publication Number | Publication Date |
---|---|
EA199900352A1 true EA199900352A1 (ru) | 1999-08-26 |
EA001213B1 EA001213B1 (ru) | 2000-12-25 |
Family
ID=27268667
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA199900352A EA001213B1 (ru) | 1996-10-04 | 1997-10-02 | Композиции жидкого алендроната |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP1007054A4 (ru) |
JP (1) | JP2001501222A (ru) |
CN (1) | CN1238691A (ru) |
AU (1) | AU723357B2 (ru) |
BG (1) | BG103306A (ru) |
BR (1) | BR9712197A (ru) |
CA (1) | CA2267370A1 (ru) |
CZ (1) | CZ116999A3 (ru) |
EA (1) | EA001213B1 (ru) |
EE (1) | EE03669B1 (ru) |
HU (1) | HUP0000125A3 (ru) |
IL (1) | IL129127A0 (ru) |
IS (1) | IS5012A (ru) |
NO (1) | NO991569L (ru) |
NZ (1) | NZ334836A (ru) |
PL (1) | PL332496A1 (ru) |
SK (1) | SK42999A3 (ru) |
TR (1) | TR199900730T2 (ru) |
WO (1) | WO1998014196A1 (ru) |
YU (1) | YU17499A (ru) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE297740T1 (de) | 2001-01-23 | 2005-07-15 | Gador Sa | Bisphosphonate-enthaltenden zusammensetzungen zur vorbeugung und/oder heilung von metabolischen knochenkrankheiten, verfahren zu ihren herstellung und benutzung dieser zusammensetzungen |
US7645460B2 (en) | 2004-05-24 | 2010-01-12 | The Procter & Gamble Company | Dosage forms of risedronate |
US20080286359A1 (en) | 2004-05-24 | 2008-11-20 | Richard John Dansereau | Low Dosage Forms Of Risedronate Or Its Salts |
US7645459B2 (en) | 2004-05-24 | 2010-01-12 | The Procter & Gamble Company | Dosage forms of bisphosphonates |
US20080287400A1 (en) | 2004-05-24 | 2008-11-20 | Richard John Dansereau | Low Dosage Forms Of Risedronate Or Its Salts |
NZ567200A (en) * | 2005-09-16 | 2010-08-27 | Selamine Ltd | Bisphosphonate formulation |
US7473684B2 (en) | 2005-09-16 | 2009-01-06 | Selamine Limited | Bisphosphonate formulation |
JP2010043119A (ja) * | 2009-10-16 | 2010-02-25 | Gador Sa | 骨の代謝病の予防および/または治療のための組成物、その組成物の調製方法およびその使用 |
US8568747B1 (en) | 2012-10-05 | 2013-10-29 | Silvergate Pharmaceuticals, Inc. | Enalapril compositions |
US9463183B1 (en) | 2015-10-30 | 2016-10-11 | Silvergate Pharmaceuticals, Inc. | Lisinopril formulations |
US9669008B1 (en) | 2016-03-18 | 2017-06-06 | Silvergate Pharmaceuticals, Inc. | Enalapril formulations |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4206209A (en) * | 1978-11-02 | 1980-06-03 | Kracauer Paul | Sublingual aspirin tablet |
IT1201087B (it) * | 1982-04-15 | 1989-01-27 | Gentili Ist Spa | Bifosfonati farmacologicamente attivi,procedimento per la loro preparazione e relative composizioni farmaceutiche |
US4922007A (en) * | 1989-06-09 | 1990-05-01 | Merck & Co., Inc. | Process for preparing 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid or salts thereof |
US5019651A (en) * | 1990-06-20 | 1991-05-28 | Merck & Co., Inc. | Process for preparing 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid (ABP) or salts thereof |
US5270365A (en) * | 1991-12-17 | 1993-12-14 | Merck & Co., Inc. | Prevention and treatment of periodontal disease with alendronate |
US5358941A (en) * | 1992-12-02 | 1994-10-25 | Merck & Co., Inc. | Dry mix formulation for bisphosphonic acids with lactose |
FR2703590B1 (fr) * | 1993-04-05 | 1995-06-30 | Sanofi Elf | Utilisation de derives d'acide bisphosphonique pour la preparation de medicaments destines a favoriser la reparation osseuse . |
US5510517A (en) * | 1993-08-25 | 1996-04-23 | Merck & Co., Inc. | Process for producing N-amino-1-hydroxy-alkylidene-1,1-bisphosphonic acids |
US5462932A (en) * | 1994-05-17 | 1995-10-31 | Merck & Co., Inc. | Oral liquid alendronate formulations |
US5780455A (en) * | 1994-08-24 | 1998-07-14 | Merck & Co., Inc. | Intravenous alendronate formulations |
US5616571A (en) * | 1995-06-06 | 1997-04-01 | Merck & Co., Inc. | Bisphosphonates prevent bone loss associated with immunosuppressive therapy |
-
1997
- 1997-10-02 SK SK429-99A patent/SK42999A3/sk unknown
- 1997-10-02 EE EEP199900113A patent/EE03669B1/xx not_active IP Right Cessation
- 1997-10-02 CN CN97180165A patent/CN1238691A/zh active Pending
- 1997-10-02 TR TR1999/00730T patent/TR199900730T2/xx unknown
- 1997-10-02 HU HU0000125A patent/HUP0000125A3/hu unknown
- 1997-10-02 BR BR9712197-5A patent/BR9712197A/pt unknown
- 1997-10-02 EP EP97945195A patent/EP1007054A4/en not_active Withdrawn
- 1997-10-02 PL PL97332496A patent/PL332496A1/xx unknown
- 1997-10-02 IL IL12912797A patent/IL129127A0/xx unknown
- 1997-10-02 WO PCT/US1997/015740 patent/WO1998014196A1/en not_active Application Discontinuation
- 1997-10-02 CA CA002267370A patent/CA2267370A1/en not_active Abandoned
- 1997-10-02 EA EA199900352A patent/EA001213B1/ru not_active IP Right Cessation
- 1997-10-02 NZ NZ334836A patent/NZ334836A/xx unknown
- 1997-10-02 CZ CZ991169A patent/CZ116999A3/cs unknown
- 1997-10-02 JP JP10516541A patent/JP2001501222A/ja active Pending
- 1997-10-02 AU AU46448/97A patent/AU723357B2/en not_active Ceased
-
1999
- 1999-03-26 IS IS5012A patent/IS5012A/is unknown
- 1999-03-30 NO NO991569A patent/NO991569L/no not_active Application Discontinuation
- 1999-03-31 YU YU17499A patent/YU17499A/sr unknown
- 1999-04-02 BG BG103306A patent/BG103306A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
YU17499A (en) | 1999-11-22 |
CZ116999A3 (cs) | 1999-09-15 |
AU4644897A (en) | 1998-04-24 |
EP1007054A1 (en) | 2000-06-14 |
WO1998014196A1 (en) | 1998-04-09 |
IS5012A (is) | 1999-03-26 |
EP1007054A4 (en) | 2000-07-19 |
PL332496A1 (en) | 1999-09-13 |
EE9900113A (et) | 1999-10-15 |
CN1238691A (zh) | 1999-12-15 |
EA001213B1 (ru) | 2000-12-25 |
HUP0000125A3 (en) | 2001-04-28 |
NO991569L (no) | 1999-06-04 |
SK42999A3 (en) | 2000-01-18 |
EE03669B1 (et) | 2002-04-15 |
BG103306A (en) | 2000-01-31 |
NO991569D0 (no) | 1999-03-30 |
JP2001501222A (ja) | 2001-01-30 |
CA2267370A1 (en) | 1998-04-09 |
AU723357B2 (en) | 2000-08-24 |
NZ334836A (en) | 2000-11-24 |
BR9712197A (pt) | 1999-08-31 |
IL129127A0 (en) | 2000-02-17 |
TR199900730T2 (xx) | 1999-07-21 |
HUP0000125A2 (hu) | 2000-06-28 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA199901100A1 (ru) | Фармацевтические композиции, содержащие гемисульфат элетриптана и кофеин | |
EA199800563A1 (ru) | Антагонисты гормона, высвобождающего гонадотропин | |
EA199900979A1 (ru) | Композиции активированного протеина | |
FI970825A (fi) | Farmaseuttiset koostumukset, jotka aktiivisen yhdisteen biologisen hyötyosuuden lisäämiseksi sisältävät sappisuolaa ja puskuria | |
TR200200706T2 (tr) | Nöropatik ağrı tedavisi için retigabin kullanımı. | |
EA199700285A1 (ru) | Препарат, содержащий мономерный аналог инсулина, кристаллический аналог инсулина, способ его получения | |
HU9602229D0 (en) | Novel mercaptoacetylamido 1,3,4,5-tetrahydro-benzo[c]azepin-3-one disulfide derivatives useful as inhibitors of enkephalinase and ace | |
EA200100412A1 (ru) | Замещенные 3-цианохинолины в качестве ингибиторов протеинтирозинкиназ | |
ES2125477T3 (es) | Composicion detergente lavavajillas concentrada, liquida o gelificada, que contiene xileno-sulfonato de calcio. | |
NZ240230A (en) | Mercaptoacetylamide derivatives; preparation, use and pharmaceutical compositions thereof | |
ES2158537T3 (es) | Derivados de acidos ciclopropilalcanoicos. | |
PT814782E (pt) | Composicao farmaceutica estabilizada com um agente basico | |
EA200400815A1 (ru) | Контролируемый синтез зипразидона и его композиции | |
CA2244785A1 (en) | Pentafluorobenzenesulfonamides and analogs | |
EA199900352A1 (ru) | Композиции жидкого алендроната | |
EA200200479A1 (ru) | Новые олигосахариды, их получение и содержащие их фармацевтические композиции | |
EA200100194A1 (ru) | КРИСТАЛЛИЧЕСКИЕ ФОРМЫ ETO2C-CH2-(R)Cgl-Aze-Pab-OH | |
EA200100354A1 (ru) | Фармацевтическая композиция, содержащая энтакапон или нитекапон, а также поперечно-сшитое производное целлюлозы | |
EA200100184A1 (ru) | Новые гидратные формы алендроната натрия, способы их получения и фармацевтические композиции | |
EA199901013A1 (ru) | Гели пролонгированного действия | |
BG103558A (en) | Sulphonic acid or sulphonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds | |
EA199700160A1 (ru) | Производные индола в качестве антагонистов eaa | |
ITRM910430A1 (it) | Composizioni farmaceutiche di somatostatina con assorbimento migliorato, loro preparazione e loro impiego | |
NO982229D0 (no) | Svovelholdige di-tert-butylfenol-forbindelser anvendbare som antiinflammatoriske midler | |
EA200000198A1 (ru) | 2-ациламинопропанамины в качестве антагонистов рецепторов тахикининов |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |