EA199800535A1 - METHOD OF TREATMENT OF PAIN - Google Patents

METHOD OF TREATMENT OF PAIN

Info

Publication number
EA199800535A1
EA199800535A1 EA199800535A EA199800535A EA199800535A1 EA 199800535 A1 EA199800535 A1 EA 199800535A1 EA 199800535 A EA199800535 A EA 199800535A EA 199800535 A EA199800535 A EA 199800535A EA 199800535 A1 EA199800535 A1 EA 199800535A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pain
treatment
composition
compound
azabicyclic
Prior art date
Application number
EA199800535A
Other languages
Russian (ru)
Inventor
Чарлз Х. Митч
Харлан Э. Шэннон
Original Assignee
Эли Лилли Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эли Лилли Энд Компани filed Critical Эли Лилли Энд Компани
Publication of EA199800535A1 publication Critical patent/EA199800535A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Abstract

Данное изобретение представляет способ и композицию для лечения боли с использованием композиции, содержащей азабициклическое или тетрагидропиридиновое соединение и классическое анальгетическое соединение.Международная заявка была опубликована вместе с отчетом о международном поиске.The present invention provides a method and composition for treating pain using a composition comprising an azabicyclic or tetrahydropyridine compound and a classic analgesic compound. The international application was published along with an international search report.

EA199800535A 1995-12-07 1996-12-05 METHOD OF TREATMENT OF PAIN EA199800535A1 (en)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US831895P 1995-12-07 1995-12-07
US830695P 1995-12-07 1995-12-07
US829895P 1995-12-07 1995-12-07
US831295P 1995-12-07 1995-12-07
US831995P 1995-12-07 1995-12-07
US829595P 1995-12-07 1995-12-07
US831395P 1995-12-07 1995-12-07
PCT/US1996/019390 WO1997020556A1 (en) 1995-12-07 1996-12-05 Method for treating pain

Publications (1)

Publication Number Publication Date
EA199800535A1 true EA199800535A1 (en) 1998-12-24

Family

ID=27567403

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199800535A EA199800535A1 (en) 1995-12-07 1996-12-05 METHOD OF TREATMENT OF PAIN

Country Status (14)

Country Link
EP (1) EP0866702A4 (en)
JP (1) JP2000501711A (en)
KR (1) KR19990071977A (en)
CN (1) CN1208348A (en)
AU (1) AU715645B2 (en)
CA (1) CA2239732A1 (en)
CZ (1) CZ174598A3 (en)
EA (1) EA199800535A1 (en)
HU (1) HUP0000110A3 (en)
IL (1) IL124786A0 (en)
NO (1) NO982582L (en)
NZ (1) NZ324594A (en)
PL (1) PL327144A1 (en)
WO (1) WO1997020556A1 (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1189902B1 (en) 1999-06-04 2003-08-27 Eli Lilly And Company 7-oxo-2-azabicyclo[2.2.1]heptanes as selective muscarinic receptor antagonist
US10195153B2 (en) 2013-08-12 2019-02-05 Pharmaceutical Manufacturing Research Services, Inc. Extruded immediate release abuse deterrent pill
US10172797B2 (en) 2013-12-17 2019-01-08 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
US9492444B2 (en) 2013-12-17 2016-11-15 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
EP3169315B1 (en) 2014-07-17 2020-06-24 Pharmaceutical Manufacturing Research Services, Inc. Immediate release abuse deterrent liquid fill dosage form
US20160106737A1 (en) 2014-10-20 2016-04-21 Pharmaceutical Manufacturing Research Services, Inc. Extended Release Abuse Deterrent Liquid Fill Dosage Form
WO2021097427A1 (en) 2019-11-15 2021-05-20 Karuna Therapeutics, Inc. Xanomeline derivatives and methods for treating neurological disorders
CN115974863A (en) * 2021-10-14 2023-04-18 南京迈诺威医药科技有限公司 Malate of xanomeline derivative, crystal form A, preparation method of malate, and application of crystal form A

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5043345A (en) * 1989-02-22 1991-08-27 Novo Nordisk A/S Piperidine compounds and their preparation and use
US5527813A (en) * 1990-08-21 1996-06-18 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
US5376668A (en) * 1990-08-21 1994-12-27 Novo Nordisk A/S Heterocyclic compounds
DK198590D0 (en) * 1990-08-21 1990-08-21 Novo Nordisk As HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND USE
WO1993014089A1 (en) * 1992-01-13 1993-07-22 Novo Nordisk A/S Heterocyclic compounds and their preparation and use
US5605701A (en) * 1995-02-17 1997-02-25 Eli Lilly And Company Transdermal formulation

Also Published As

Publication number Publication date
PL327144A1 (en) 1998-11-23
HUP0000110A3 (en) 2000-09-28
WO1997020556A1 (en) 1997-06-12
AU715645B2 (en) 2000-02-10
CN1208348A (en) 1999-02-17
IL124786A0 (en) 1999-01-26
AU1147697A (en) 1997-06-27
HUP0000110A2 (en) 2000-06-28
EP0866702A4 (en) 2001-07-25
NO982582D0 (en) 1998-06-05
NZ324594A (en) 1999-09-29
KR19990071977A (en) 1999-09-27
EP0866702A1 (en) 1998-09-30
CZ174598A3 (en) 1999-01-13
CA2239732A1 (en) 1997-06-12
NO982582L (en) 1998-08-03
JP2000501711A (en) 2000-02-15

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