DK3573611T3 - Amidforbindelser og anvendelse deraf - Google Patents

Amidforbindelser og anvendelse deraf Download PDF

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Publication number
DK3573611T3
DK3573611T3 DK18745107.5T DK18745107T DK3573611T3 DK 3573611 T3 DK3573611 T3 DK 3573611T3 DK 18745107 T DK18745107 T DK 18745107T DK 3573611 T3 DK3573611 T3 DK 3573611T3
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amide compounds
amide
compounds
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DK18745107.5T
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English (en)
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Cheng-Ho Chung
Shi-Liang Tseng
Yung-Ning Yang
Yen-Fu Chen
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Alphala Co Ltd
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    • C07—ORGANIC CHEMISTRY
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    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
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    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
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    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/107—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with two aryl or substituted aryl radicals attached in positions 2 and 5
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK18745107.5T 2017-01-24 2018-01-22 Amidforbindelser og anvendelse deraf DK3573611T3 (da)

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US20230355591A1 (en) * 2020-01-10 2023-11-09 Alphala Co., Ltd. Pharmaceutical composition and use thereof
BR112022015507A2 (pt) * 2020-03-06 2022-09-27 Alphala Co Ltd Processos para produzir compostos de amida, e sua forma cristalina e salina
JP7368548B2 (ja) * 2021-07-02 2023-10-24 昊運股▲フン▼有限公司 薬学的組成物及びその使用

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US6524619B2 (en) * 2000-01-27 2003-02-25 Chronorx, Inc. Dosage forms useful for modifying conditions and functions associated with hearing loss and/or tinnitus
US6774111B1 (en) * 2000-03-14 2004-08-10 Abbott Laboratories Carbohydrate system and a method for providing nutrition to a diabetic
MXPA02011609A (es) * 2000-05-26 2003-03-27 Nippon Shinyaku Co Ltd Compuestos heterociclicos.
CA2446161A1 (en) * 2001-05-04 2002-11-14 Emanuele Sher Use of an ampa receptor potentiator for the manufacture of a medicament for the treatment of type 2 diabetes
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EP3573611A4 (en) 2020-09-09
US20190337915A1 (en) 2019-11-07
CA3048911C (en) 2021-11-09
EP3573611A1 (en) 2019-12-04
NZ755328A (en) 2021-06-25
CA3048911A1 (en) 2018-08-02
LT3573611T (lt) 2022-03-25
EP3573611B1 (en) 2022-01-12
SG11201905965QA (en) 2019-08-27
KR20190099048A (ko) 2019-08-23
CN110234318A (zh) 2019-09-13
TW201838967A (zh) 2018-11-01
PH12019501566A1 (en) 2020-03-09
BR112019015191A2 (pt) 2020-03-24
AU2018212473B2 (en) 2020-06-11
TWI676621B (zh) 2019-11-11
MX2019008728A (es) 2019-09-18
EA039455B1 (ru) 2022-01-28
RS63068B1 (sr) 2022-04-29
ZA201904383B (en) 2020-12-23
HUE058153T2 (hu) 2022-07-28
KR102378883B1 (ko) 2022-03-25
AU2018212473A1 (en) 2019-07-18
PL3573611T3 (pl) 2022-06-13
TW201838977A (zh) 2018-11-01
IL267937B (en) 2022-09-01
US10882837B2 (en) 2021-01-05
PT3573611T (pt) 2022-03-15
ES2907746T3 (es) 2022-04-26
SA519402283B1 (ar) 2022-12-25
WO2018140338A1 (en) 2018-08-02
JP2020506226A (ja) 2020-02-27
US11384060B2 (en) 2022-07-12
HRP20220232T1 (hr) 2022-05-13
TWI753995B (zh) 2022-02-01
SI3573611T1 (sl) 2022-05-31
US20190345118A1 (en) 2019-11-14
EA201991570A1 (ru) 2019-12-30
WO2018140339A1 (en) 2018-08-02
IL267937A (en) 2019-09-26
JP6937524B2 (ja) 2021-09-22

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