DK246878A - PROCEDURE FOR THE PREPARATION OF ACYLD DERIVATIVES - Google Patents

PROCEDURE FOR THE PREPARATION OF ACYLD DERIVATIVES

Info

Publication number
DK246878A
DK246878A DK246878A DK246878A DK246878A DK 246878 A DK246878 A DK 246878A DK 246878 A DK246878 A DK 246878A DK 246878 A DK246878 A DK 246878A DK 246878 A DK246878 A DK 246878A
Authority
DK
Denmark
Prior art keywords
acyld
derivatives
procedure
preparation
acyld derivatives
Prior art date
Application number
DK246878A
Other languages
Danish (da)
Inventor
M Montavon
R Reiner
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK246878A publication Critical patent/DK246878A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK246878A 1977-06-03 1978-06-02 PROCEDURE FOR THE PREPARATION OF ACYLD DERIVATIVES DK246878A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
LU77485 1977-06-03
CH314278 1978-03-22

Publications (1)

Publication Number Publication Date
DK246878A true DK246878A (en) 1978-12-04

Family

ID=25692293

Family Applications (1)

Application Number Title Priority Date Filing Date
DK246878A DK246878A (en) 1977-06-03 1978-06-02 PROCEDURE FOR THE PREPARATION OF ACYLD DERIVATIVES

Country Status (26)

Country Link
EP (1) EP0000005B1 (en)
JP (1) JPS5412394A (en)
AR (1) AR225134A1 (en)
AT (2) AT362501B (en)
AU (1) AU518648B2 (en)
BR (1) BR7803565A (en)
CA (1) CA1114808A (en)
CU (1) CU21118A (en)
DE (2) DE2824065A1 (en)
DK (1) DK246878A (en)
ES (2) ES470442A1 (en)
FI (1) FI781754A (en)
FR (1) FR2393000A1 (en)
GB (1) GB1599232A (en)
GR (1) GR73554B (en)
HU (1) HU182498B (en)
IE (1) IE46903B1 (en)
IL (1) IL54803A (en)
IT (1) IT1098306B (en)
MC (1) MC1195A1 (en)
NL (1) NL7805715A (en)
NO (1) NO781934L (en)
NZ (1) NZ187392A (en)
PH (1) PH14653A (en)
PT (1) PT68134A (en)
SE (1) SE7806465L (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4200745A (en) * 1977-12-20 1980-04-29 Eli Lilly And Company 7[2-(2-Aminothiazol-4-yl)-2-alkoxyimino]acetamido 3[4-alkyl-5-oxo-6-hydroxy-3,4 dihydro 1,2,4-triazin 3-yl]thio methyl cephalosporins
FR2432521A1 (en) * 1978-03-31 1980-02-29 Roussel Uclaf NOVEL O-SUBSTITUTED OXIMES DERIVED FROM 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC ACID, THEIR PREPARATION PROCESS AND THEIR USE AS MEDICAMENTS
MC1259A1 (en) * 1978-05-30 1980-01-14 Hoffmann La Roche ACYL DERIVATIVES
NO782998L (en) * 1978-07-19 1980-01-22 Hoffmann La Roche CEPHALOSPORINESTERS AND EATERS.
US4472574A (en) * 1981-05-22 1984-09-18 Hoffman-La Roche Inc. Process for the manufacture of a cephem carboxylic acid derivative
US4698338A (en) * 1986-02-19 1987-10-06 Eli Lilly And Company 7[2-(2-aminothiazol-4-yl)-2-benzyloximino]acetamido-3[4-alkyl-5-oxo-6-hydroxy-3,4-dihydro-1,2,4-triazin-3-yl]thiomethyl cephalosporins

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1399086A (en) * 1971-05-14 1975-06-25 Glaxo Lab Ltd Cephalosporin compounds
CH609989A5 (en) * 1974-06-21 1979-03-30 Hoffmann La Roche Process for the preparation of acyl derivatives
CA1100129A (en) * 1974-08-02 1981-04-28 William H.W. Lunn Cephalosporin compounds
GB1555471A (en) * 1975-06-19 1979-11-14 Glaxo Lab Ltd 7 carbamoylalkoxyimino acetamido 3 em 4 carboxylic acidsand derivatives thereof
GB1576625A (en) * 1976-04-12 1980-10-08 Fujisawa Pharmaceutical Co Syn isomer 3,7 disubstituted 3 cephem 4 carboxylic acid compounds and processes for the preparation thereof
GB1596278A (en) * 1976-11-30 1981-08-26 Glaxo Operations Ltd 7-(-oxyimino-acetamino)cephalosporin derivatives

Also Published As

Publication number Publication date
JPS5412394A (en) 1979-01-30
NO781934L (en) 1978-12-05
NL7805715A (en) 1978-12-05
IT7824165A0 (en) 1978-06-02
IE781056L (en) 1978-12-03
IT1098306B (en) 1985-09-07
EP0000005B1 (en) 1980-10-29
AT365197B (en) 1981-12-28
AU518648B2 (en) 1981-10-15
NZ187392A (en) 1984-05-31
PT68134A (en) 1978-07-01
AT362501B (en) 1981-05-25
IL54803A (en) 1982-01-31
CU21118A (en) 1983-04-06
SE7806465L (en) 1978-12-04
ATA345980A (en) 1981-05-15
IL54803A0 (en) 1978-07-31
HU182498B (en) 1984-01-30
GR73554B (en) 1984-03-14
PH14653A (en) 1981-10-14
ATA403578A (en) 1980-10-15
AU3658878A (en) 1979-12-06
IE46903B1 (en) 1983-11-02
FR2393000A1 (en) 1978-12-29
FI781754A (en) 1978-12-04
AR225134A1 (en) 1982-02-26
FR2393000B1 (en) 1982-10-29
MC1195A1 (en) 1979-02-23
ES478115A1 (en) 1979-06-01
EP0000005A1 (en) 1978-12-20
CA1114808A (en) 1981-12-22
GB1599232A (en) 1981-09-30
ES470442A1 (en) 1979-10-01
DE2860248D1 (en) 1981-01-29
BR7803565A (en) 1979-02-20
DE2824065A1 (en) 1978-12-14

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Legal Events

Date Code Title Description
AHS Application shelved for other reasons than non-payment
AHB Application shelved due to non-payment