DK155283C - METHOD OF ANALOGUE FOR THE PREPARATION OF 1- (BETA- (R-THIO) -PHENETHYL) -IMIDAZOLES OR ACID ADDITION SALTS THEREOF - Google Patents

METHOD OF ANALOGUE FOR THE PREPARATION OF 1- (BETA- (R-THIO) -PHENETHYL) -IMIDAZOLES OR ACID ADDITION SALTS THEREOF

Info

Publication number
DK155283C
DK155283C DK427075A DK427075A DK155283C DK 155283 C DK155283 C DK 155283C DK 427075 A DK427075 A DK 427075A DK 427075 A DK427075 A DK 427075A DK 155283 C DK155283 C DK 155283C
Authority
DK
Denmark
Prior art keywords
imidazoles
phenethyl
thio
analogue
beta
Prior art date
Application number
DK427075A
Other languages
Danish (da)
Other versions
DK427075A (en
DK155283B (en
Inventor
Keith A M Walker
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of DK427075A publication Critical patent/DK427075A/en
Publication of DK155283B publication Critical patent/DK155283B/en
Application granted granted Critical
Publication of DK155283C publication Critical patent/DK155283C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK427075A 1974-09-23 1975-09-23 METHOD OF ANALOGUE FOR THE PREPARATION OF 1- (BETA- (R-THIO) -PHENETHYL) -IMIDAZOLES OR ACID ADDITION SALTS THEREOF DK155283C (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US50838474A 1974-09-23 1974-09-23
US50838474 1974-09-23
US59362075A 1975-07-07 1975-07-07
US59362075 1975-07-07

Publications (3)

Publication Number Publication Date
DK427075A DK427075A (en) 1976-03-24
DK155283B DK155283B (en) 1989-03-20
DK155283C true DK155283C (en) 1989-07-24

Family

ID=27056177

Family Applications (1)

Application Number Title Priority Date Filing Date
DK427075A DK155283C (en) 1974-09-23 1975-09-23 METHOD OF ANALOGUE FOR THE PREPARATION OF 1- (BETA- (R-THIO) -PHENETHYL) -IMIDAZOLES OR ACID ADDITION SALTS THEREOF

Country Status (19)

Country Link
JP (1) JPS5910344B2 (en)
AR (1) AR224222A1 (en)
AU (1) AU496881B2 (en)
CA (1) CA1064040A (en)
CH (1) CH623813A5 (en)
DE (1) DE2541833A1 (en)
DK (1) DK155283C (en)
FI (1) FI64583C (en)
FR (1) FR2285126A1 (en)
GB (1) GB1485719A (en)
HK (1) HK8380A (en)
IE (1) IE43267B1 (en)
IL (1) IL47885A (en)
MX (1) MX4832E (en)
MY (1) MY8000270A (en)
NL (1) NL174462C (en)
NO (1) NO144345C (en)
SE (1) SE428471B (en)
YU (3) YU39746B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA755100B (en) * 1974-09-23 1977-03-30 Syntex Inc 1-(b-(r-thio) phenethyl) imidazoles and derivatives thereof
EP0013786B1 (en) * 1979-01-22 1982-10-06 Syntex (U.S.A.) Inc. Imidazole derivatives, pharmaceutical compositions containing them and their preparation
JPS63156228U (en) * 1987-04-01 1988-10-13
DE3939525A1 (en) * 1989-11-30 1991-06-06 Hoechst Ag ARYL-ALKYL-AZOLES SUBSTITUTED WITH MULTIPLE UNSATURATED REMAINS, METHOD FOR THEIR PRODUCTION AND THEIR USE
IT1303672B1 (en) * 1998-07-28 2001-02-23 Nicox Sa NITRATED SALTS OF DRUGS ACTIVE IN BONE DISORDERS
CN116063234B (en) * 2022-12-29 2023-11-24 山东京卫制药有限公司 Preparation method of sulconazole nitrate

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU557755A3 (en) * 1968-08-19 1977-05-05 Янссен Фармасьютика Н.В. (Фирма) Method for preparing imidazole derivatives
US3658813A (en) * 1970-01-13 1972-04-25 Janssen Pharmaceutica Nv 1-(beta-aryl-beta-(r-oxy)-ethyl)-imidazoles
DE2041771C3 (en) * 1970-08-22 1979-07-26 Bayer Ag, 5090 Leverkusen derivatives
SE364275B (en) * 1971-06-17 1974-02-18 Janssen Pharmaceutica Nv
DE2242454A1 (en) * 1972-08-29 1974-03-07 Bayer Ag 1-AETHYL-IMIDAZOLE, METHOD FOR MANUFACTURING IT AND ITS USE AS A MEDICINAL PRODUCT

Also Published As

Publication number Publication date
NO144345B (en) 1981-05-04
JPS5910344B2 (en) 1984-03-08
IL47885A0 (en) 1975-11-25
IE43267B1 (en) 1981-01-28
YU227081A (en) 1982-02-28
DK427075A (en) 1976-03-24
AR224222A1 (en) 1981-11-13
NO753048L (en) 1976-03-24
FR2285126A1 (en) 1976-04-16
JPS5157828A (en) 1976-05-20
IL47885A (en) 1979-01-31
FI752614A (en) 1976-03-24
GB1485719A (en) 1977-09-14
FI64583C (en) 1983-12-12
DE2541833A1 (en) 1976-04-01
SE428471B (en) 1983-07-04
YU226981A (en) 1982-02-28
FR2285126B1 (en) 1979-09-14
DE2541833C2 (en) 1989-09-14
MY8000270A (en) 1980-12-31
YU224475A (en) 1982-02-28
NL174462B (en) 1984-01-16
MX4832E (en) 1982-10-26
NL174462C (en) 1984-06-18
NL7510224A (en) 1976-03-25
CH623813A5 (en) 1981-06-30
FI64583B (en) 1983-08-31
AU496881B2 (en) 1978-11-09
AU8408175A (en) 1977-02-24
SE7510595L (en) 1976-03-24
CA1064040A (en) 1979-10-09
HK8380A (en) 1980-03-14
DK155283B (en) 1989-03-20
YU39746B (en) 1985-04-30
NO144345C (en) 1981-08-12
IE43267L (en) 1976-03-23

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