DK1423108T3 - C-2'-methylerede derivater af paclitaxel til brug som antitumorpræparater - Google Patents

C-2'-methylerede derivater af paclitaxel til brug som antitumorpræparater

Info

Publication number
DK1423108T3
DK1423108T3 DK02764753T DK02764753T DK1423108T3 DK 1423108 T3 DK1423108 T3 DK 1423108T3 DK 02764753 T DK02764753 T DK 02764753T DK 02764753 T DK02764753 T DK 02764753T DK 1423108 T3 DK1423108 T3 DK 1423108T3
Authority
DK
Denmark
Prior art keywords
sub
paclitaxel
methylated derivatives
formula
antitumor preparations
Prior art date
Application number
DK02764753T
Other languages
Danish (da)
English (en)
Inventor
Ezio Bombardelli
Gabriele Fontana
Arturo Battaglia
Samanta Cimitan
Original Assignee
Indena Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Indena Spa filed Critical Indena Spa
Application granted granted Critical
Publication of DK1423108T3 publication Critical patent/DK1423108T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/12Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epoxy Compounds (AREA)
DK02764753T 2001-08-07 2002-07-23 C-2'-methylerede derivater af paclitaxel til brug som antitumorpræparater DK1423108T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT2001MI001734A ITMI20011734A1 (it) 2001-08-07 2001-08-07 Derivanti tassanici e procedimenti per la loro preparazione
PCT/EP2002/008185 WO2003013503A1 (en) 2001-08-07 2002-07-23 C-2' methylated derivatives of paclitaxel for use as antitumour agents

Publications (1)

Publication Number Publication Date
DK1423108T3 true DK1423108T3 (da) 2007-10-01

Family

ID=11448252

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02764753T DK1423108T3 (da) 2001-08-07 2002-07-23 C-2'-methylerede derivater af paclitaxel til brug som antitumorpræparater

Country Status (21)

Country Link
US (1) US7153884B2 (ru)
EP (1) EP1423108B1 (ru)
KR (1) KR100894580B1 (ru)
CN (1) CN100370980C (ru)
AT (1) ATE363901T1 (ru)
AU (1) AU2002328942B2 (ru)
BR (1) BR0211770A (ru)
CA (1) CA2456523A1 (ru)
DE (1) DE60220524T2 (ru)
DK (1) DK1423108T3 (ru)
ES (1) ES2287310T3 (ru)
HK (1) HK1066483A1 (ru)
HU (1) HUP0401275A3 (ru)
IL (1) IL160233A0 (ru)
IT (1) ITMI20011734A1 (ru)
MX (1) MXPA04001234A (ru)
NO (1) NO20040535L (ru)
PL (1) PL194975B1 (ru)
PT (1) PT1423108E (ru)
RU (1) RU2287528C2 (ru)
WO (1) WO2003013503A1 (ru)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2460769C (en) * 2007-11-30 2011-09-07 Applied Genomics Inc TLE3 as a marker for chemotherapy
CN101851231A (zh) * 2010-05-27 2010-10-06 东北林业大学 一种多西紫杉醇新衍生物的合成方法及其在制备抗肿瘤药物中的应用
CN104650012A (zh) * 2013-11-22 2015-05-27 天士力控股集团有限公司 一种紫杉烷类化合物

Also Published As

Publication number Publication date
AU2002328942B2 (en) 2007-08-30
US20040242674A1 (en) 2004-12-02
CA2456523A1 (en) 2003-02-20
RU2287528C2 (ru) 2006-11-20
EP1423108A1 (en) 2004-06-02
HK1066483A1 (en) 2005-03-24
EP1423108B1 (en) 2007-06-06
WO2003013503A1 (en) 2003-02-20
KR20040030926A (ko) 2004-04-09
DE60220524D1 (de) 2007-07-19
NO20040535L (no) 2004-04-26
RU2004103481A (ru) 2005-06-10
PL367868A1 (en) 2005-03-07
CN100370980C (zh) 2008-02-27
CN1538841A (zh) 2004-10-20
KR100894580B1 (ko) 2009-04-24
US7153884B2 (en) 2006-12-26
BR0211770A (pt) 2004-07-27
ES2287310T3 (es) 2007-12-16
MXPA04001234A (es) 2004-05-27
HUP0401275A2 (hu) 2004-10-28
IL160233A0 (en) 2004-07-25
ITMI20011734A0 (it) 2001-08-07
ITMI20011734A1 (it) 2003-02-07
HUP0401275A3 (en) 2007-05-29
PL194975B1 (pl) 2007-07-31
PT1423108E (pt) 2007-08-28
DE60220524T2 (de) 2008-02-07
ATE363901T1 (de) 2007-06-15

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