DK108500C - Fremgangsmåde til fremstilling af 1-glykosyl-5-azacytosiner. - Google Patents

Fremgangsmåde til fremstilling af 1-glykosyl-5-azacytosiner.

Info

Publication number
DK108500C
DK108500C DK620664AA DK620664A DK108500C DK 108500 C DK108500 C DK 108500C DK 620664A A DK620664A A DK 620664AA DK 620664 A DK620664 A DK 620664A DK 108500 C DK108500 C DK 108500C
Authority
DK
Denmark
Prior art keywords
azacytosines
glycosyl
preparation
Prior art date
Application number
DK620664AA
Other languages
Danish (da)
English (en)
Original Assignee
Ceskoslovenska Akademie Ved
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ceskoslovenska Akademie Ved filed Critical Ceskoslovenska Akademie Ved
Application granted granted Critical
Publication of DK108500C publication Critical patent/DK108500C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/12—Triazine radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK620664AA 1963-12-22 1964-12-18 Fremgangsmåde til fremstilling af 1-glykosyl-5-azacytosiner. DK108500C (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CS709363 1963-12-22

Publications (1)

Publication Number Publication Date
DK108500C true DK108500C (da) 1967-12-27

Family

ID=5419399

Family Applications (1)

Application Number Title Priority Date Filing Date
DK620664AA DK108500C (da) 1963-12-22 1964-12-18 Fremgangsmåde til fremstilling af 1-glykosyl-5-azacytosiner.

Country Status (13)

Country Link
US (1) US3350388A (lt)
AT (1) AT252458B (lt)
BE (1) BE657451A (lt)
BR (1) BR6465569D0 (lt)
CH (1) CH479595A (lt)
DE (1) DE1245384B (lt)
DK (1) DK108500C (lt)
ES (1) ES307376A1 (lt)
FI (1) FI46389C (lt)
FR (1) FR1450440A (lt)
GB (1) GB1050899A (lt)
IT (1) IT1043755B (lt)
NL (1) NL6414959A (lt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1030970A (en) * 1964-05-15 1966-05-25 Inst Mikrobiologii Im Akad D K Method for the preparation of 2', 3', 5'-tri-o-acyl-6-azacytidines
DE2012888C3 (de) * 1970-03-14 1981-04-02 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden
US7038038B2 (en) * 2003-03-17 2006-05-02 Pharmion Corporation Synthesis of 5-azacytidine
US6887855B2 (en) * 2003-03-17 2005-05-03 Pharmion Corporation Forms of 5-azacytidine
US6943249B2 (en) * 2003-03-17 2005-09-13 Ash Stevens, Inc. Methods for isolating crystalline Form I of 5-azacytidine
US20060014949A1 (en) * 2004-07-13 2006-01-19 Supergen Inc. Compositions and formulations of decitabine polymorphs and methods of use thereof
WO2009042064A2 (en) 2007-09-21 2009-04-02 Nektar Therapeutics Al, Corporation Oligomer-nucleoside phosphate conjugates
BRPI0817269A2 (pt) * 2007-09-26 2014-10-07 Sinai School Medicine Análogos de azacitidina e usos dos mesmos
CN103479586B (zh) 2008-05-15 2017-03-01 细胞基因公司 胞苷类似物的口服制剂和其使用方法
WO2010014883A2 (en) * 2008-08-01 2010-02-04 Dr. Reddy's Laboratories Ltd. Azacitidine process and polymorphs
JP5650643B2 (ja) * 2008-08-08 2015-01-07 サイノファーム タイワン リミテッド ５−アザシトシンヌクレオシド及びその誘導体の製造方法
CA2755976C (en) * 2009-03-23 2020-04-07 Ambit Biosciences Corporation Methods of treatment using combination therapy
IT1399195B1 (it) 2010-03-30 2013-04-11 Chemi Spa Processo per la sintesi di azacitidina e decitabina
WO2012135405A1 (en) 2011-03-31 2012-10-04 Pharmion Llc Systhesis of 5-azacytidine
EA031986B1 (ru) 2012-04-04 2019-03-29 Галозим, Инк. Способ и комбинация для лечения солидной раковой опухоли и набор, содержащий комбинацию
CN108239128B (zh) 2016-12-23 2019-03-29 江苏奥赛康药业股份有限公司 β-核苷类化合物的制备方法
US20190351031A1 (en) 2018-05-16 2019-11-21 Halozyme, Inc. Methods of selecting subjects for combination cancer therapy with a polymer-conjugated soluble ph20

Also Published As

Publication number Publication date
FR1450440A (fr) 1966-06-24
ES307376A1 (es) 1965-05-01
FI46389C (fi) 1973-03-12
US3350388A (en) 1967-10-31
IT1043755B (it) 1980-02-29
FI46389B (lt) 1972-11-30
GB1050899A (lt)
AT252458B (de) 1967-02-27
CH479595A (de) 1969-10-15
BE657451A (lt) 1965-04-16
BR6465569D0 (pt) 1973-08-02
DE1245384B (de) 1967-07-27
NL6414959A (lt) 1965-06-23

Similar Documents

Publication Publication Date Title
DK108500C (da) Fremgangsmåde til fremstilling af 1-glykosyl-5-azacytosiner.
DK114837B (da) Fremgangsmåde til fremstilling af mitosanforbindelser.
DK127726B (da) Analogifremgangsmåde til fremstilling af 1-halogenbenzoylaminomethyl-2-phenyl-cyclopropan-forbindelser.
DK112736B (da) Fremgangsmåde til fremstilling af N-(3-aminopyrazinoyl)-benzamidiner.
DK111889B (da) Fremgangsmåde til fremstilling af 3-N-substituerede tricycloundecaner.
DK116292B (da) Fremgangsmåde til fremstilling af phenylalkanolaminderivater.
DK106185C (da) Fremgangsmåde til fremstilling af 17α-acyloxy-4,6-pregnadien-20-oner.
DK120596B (da) Fremgangsmåde til fremstilling af acetoxymethylbenzylpenicillinat.
DK116443B (da) Fremgangsmåde til fremstilling af 3-amino-N-carbamylpyrazolderivater.
DK106240C (da) Fremgangsmåde til fremstilling af et jern-pectin-kompleks.
DK104461C (da) Fremgangsmåde til fremstilling af 3-amino-isoxazoler.
DK107031C (da) Fremgangsmåde til fremstilling af 2-halogenmethyl-quinazolin-3-oxider.
DK105592C (da) Fremgangsmåde til fremstilling af substituerede 5-fluor-pyrimidiner.
DK112321B (da) Fremgangsmåde til fremstilling af 2-methyl-2-alkenyl-chromanderivater.
DK104571C (da) Fremgangsmåde til fremstilling af trans-2-phenyl-3-methylmorpholin.
DK115327B (da) Fremgangsmåde til fremstilling af hydroxyphenylalkylphosphonater.
DK113991B (da) Fremgangsmåde til fremstilling af 2-chlor-3-oxo-butanamider.
DK122883B (da) Fremgangsmåde til fremstilling af ω-lactamer.
DK108153C (da) Fremgangsmåde til fremstilling af 1-alkyl-5-nitroimidazol-2-carboxylater.
DK120764B (da) Fremgangsmåde til fremstilling af 2-amino-5-nitro-benzophenoner.
DK104629C (da) Fremgangsmåde til fremstilling af 7-oxodesacetamidocolchicinderivater.
DK114126B (da) Fremgangsmåde til fremstilling af substituereded benzamider.
DK129243B (da) Fremgangsmåde til fremstilling af 6-demetyltetracykliner.
DK119157B (da) Fremgangsmåde til fremstilling af 17α-acyl-16α-hydroxy-pregnen-derivater.
DK105983C (da) Fremgangsmåde til fremstilling af 2-alkoxy-5-aryl-3H-1,4-benzodiazepin-4-oxider.