DK0476682T3 - Isoprenoid phospholipase A2-inhibitorer og præparater indeholende disse - Google Patents
Isoprenoid phospholipase A2-inhibitorer og præparater indeholende disseInfo
- Publication number
- DK0476682T3 DK0476682T3 DK91116015.8T DK91116015T DK0476682T3 DK 0476682 T3 DK0476682 T3 DK 0476682T3 DK 91116015 T DK91116015 T DK 91116015T DK 0476682 T3 DK0476682 T3 DK 0476682T3
- Authority
- DK
- Denmark
- Prior art keywords
- phospholipase
- isoprenoid
- inhibitors
- preparations containing
- chem
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C63/00—Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings
- C07C63/64—Monocyclic acids with unsaturation outside the aromatic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C403/00—Derivatives of cyclohexane or of a cyclohexene or of cyclohexadiene, having a side-chain containing an acyclic unsaturated part of at least four carbon atoms, this part being directly attached to the cyclohexane or cyclohexene or cyclohexadiene rings, e.g. vitamin A, beta-carotene, beta-ionone
- C07C403/20—Derivatives of cyclohexane or of a cyclohexene or of cyclohexadiene, having a side-chain containing an acyclic unsaturated part of at least four carbon atoms, this part being directly attached to the cyclohexane or cyclohexene or cyclohexadiene rings, e.g. vitamin A, beta-carotene, beta-ionone having side-chains substituted by carboxyl groups or halides, anhydrides, or (thio)esters thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/09—Geometrical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pain & Pain Management (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Enzymes And Modification Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Immobilizing And Processing Of Enzymes And Microorganisms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/586,159 US5141959A (en) | 1990-09-21 | 1990-09-21 | Isoprenoid phospholipase a2 inhibitors and preparations comprising same |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0476682T3 true DK0476682T3 (da) | 1995-04-03 |
Family
ID=24344545
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK91116015.8T DK0476682T3 (da) | 1990-09-21 | 1991-09-20 | Isoprenoid phospholipase A2-inhibitorer og præparater indeholende disse |
Country Status (18)
Country | Link |
---|---|
US (1) | US5141959A (da) |
EP (1) | EP0476682B1 (da) |
JP (1) | JP2943089B2 (da) |
AT (1) | ATE117979T1 (da) |
AU (1) | AU637756B2 (da) |
CA (1) | CA2051766A1 (da) |
DE (1) | DE69107153T2 (da) |
DK (1) | DK0476682T3 (da) |
ES (1) | ES2067822T3 (da) |
FI (1) | FI104168B (da) |
GR (1) | GR3014944T3 (da) |
IE (1) | IE66745B1 (da) |
IL (1) | IL99536A (da) |
MX (1) | MX9101163A (da) |
NZ (1) | NZ239844A (da) |
OA (1) | OA09514A (da) |
PT (1) | PT99014B (da) |
ZA (1) | ZA917531B (da) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7189737B2 (en) | 1991-08-09 | 2007-03-13 | Research Triangle Institute | Cocaine receptor binding ligands |
US5688781A (en) | 1994-08-19 | 1997-11-18 | Bristol-Myers Squibb Company | Method for treating vascular leak syndrome |
FR2735371B1 (fr) * | 1995-06-19 | 1997-07-18 | Cird Galderma | Procede pour identifier des composes antagonistes des recepteurs rars |
US6900228B1 (en) | 1998-03-10 | 2005-05-31 | Research Triangle Institute | Opiate compounds, methods of making and methods of use |
US6267945B1 (en) * | 1998-12-18 | 2001-07-31 | Neuromed Technologies, Inc. | Farnesol-related calcium channel blockers |
US6538010B1 (en) * | 2000-11-08 | 2003-03-25 | Research Triangle Institute | Compounds and methods for promoting smoking cessation |
US8026280B2 (en) | 2001-03-27 | 2011-09-27 | Errant Gene Therapeutics, Llc | Histone deacetylase inhibitors |
US7312247B2 (en) | 2001-03-27 | 2007-12-25 | Errant Gene Therapeutics, Llc | Histone deacetylase inhibitors |
US7842727B2 (en) * | 2001-03-27 | 2010-11-30 | Errant Gene Therapeutics, Llc | Histone deacetylase inhibitors |
US6495719B2 (en) * | 2001-03-27 | 2002-12-17 | Circagen Pharmaceutical | Histone deacetylase inhibitors |
CA2486303C (en) * | 2002-05-22 | 2013-04-30 | Errant Gene Therapeutics, Llc | Histone deacetylase inhibitors based on alpha-ketoepoxide compounds |
WO2003101177A2 (en) * | 2002-06-04 | 2003-12-11 | Sequenom, Inc. | Diagnosing predisposition to fat deposition and therapeutic methods for reducing fat deposition and treatment of associated conditions |
JP2006508642A (ja) * | 2002-06-27 | 2006-03-16 | ハークネス ファーマシューティカルズ,インコーポレイティド | 脂肪の蓄積を減少させる方法と、関連疾患を治療するための方法 |
AU2003248793A1 (en) * | 2002-06-27 | 2004-01-19 | Sequenom, Inc | Diagnosing predisposition to fat deposition and associated condition |
AU2003291097A1 (en) * | 2002-11-20 | 2004-06-15 | Errant Gene Therapeutics, Llc | Treatment of lung cells with histone deacetylase inhibitors |
US20060160902A1 (en) * | 2004-11-08 | 2006-07-20 | Wiech Norbert L | Histone deacetylase inhibitors |
US7872023B2 (en) * | 2005-02-17 | 2011-01-18 | Research Triangle Institute | Kappa opioid receptor ligands |
US7399762B2 (en) * | 2005-04-25 | 2008-07-15 | Research Triangle Institute | Opioid receptor agonist compounds and their use in treatment of pain |
US7476679B2 (en) * | 2005-07-26 | 2009-01-13 | Research Triangle Institute | Octahydroisoquinoline compounds as opioid receptor modulators |
BRPI0810063A2 (pt) * | 2007-04-20 | 2014-10-14 | Acucela Inc | Composto, composição farmacêutica, e, métodos para modular fluxo de cromóforo em um ciclo retinóide, para tratar uma doença ou distúrbio oftálmico em um indivíduo, para inibir adaptação ao escuro em uma célula fotorreceptora de bastão da retina, para inibir regeneração de rodopsina em uma célula fotoreceptora de bastão da retina, para reduzir isquemia em um olho de um indivíduo, para inibir neovascularização na retina de um olho de um indivíduo, e para inibir degeneração de uma célula da retina em uma retina |
US8048895B2 (en) * | 2008-04-18 | 2011-11-01 | Research Triangle Institute | Kappa opioid receptor ligands |
AU2010346633B2 (en) | 2010-02-24 | 2015-12-03 | Research Triangle Institute | Arylpiperazine opioid receptor antagonists |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4194007A (en) * | 1978-01-13 | 1980-03-18 | Scott Eugene J Van | α-Hydroxyretinoic acid, α-ketoretinoic acid and mixtures and their use in treating skin conditions |
US4456618A (en) * | 1982-10-15 | 1984-06-26 | Sri International | Naphthenic and heterocyclic retinoic acid analogues |
US4568757A (en) * | 1984-01-30 | 1986-02-04 | Research Triangle Institute | Configurationally locked retinoids |
-
1990
- 1990-09-21 US US07/586,159 patent/US5141959A/en not_active Expired - Fee Related
-
1991
- 1991-09-18 NZ NZ239844A patent/NZ239844A/xx unknown
- 1991-09-18 CA CA002051766A patent/CA2051766A1/en not_active Abandoned
- 1991-09-19 OA OA60073A patent/OA09514A/en unknown
- 1991-09-19 MX MX9101163A patent/MX9101163A/es not_active IP Right Cessation
- 1991-09-19 PT PT99014A patent/PT99014B/pt not_active IP Right Cessation
- 1991-09-19 FI FI914405A patent/FI104168B/fi active
- 1991-09-20 IE IE331891A patent/IE66745B1/en not_active IP Right Cessation
- 1991-09-20 AU AU84626/91A patent/AU637756B2/en not_active Ceased
- 1991-09-20 JP JP3313021A patent/JP2943089B2/ja not_active Expired - Fee Related
- 1991-09-20 EP EP91116015A patent/EP0476682B1/en not_active Expired - Lifetime
- 1991-09-20 IL IL9953691A patent/IL99536A/en active IP Right Grant
- 1991-09-20 ZA ZA917531A patent/ZA917531B/xx unknown
- 1991-09-20 AT AT91116015T patent/ATE117979T1/de not_active IP Right Cessation
- 1991-09-20 ES ES91116015T patent/ES2067822T3/es not_active Expired - Lifetime
- 1991-09-20 DK DK91116015.8T patent/DK0476682T3/da active
- 1991-09-20 DE DE69107153T patent/DE69107153T2/de not_active Expired - Fee Related
-
1995
- 1995-02-02 GR GR940403510T patent/GR3014944T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
EP0476682A1 (en) | 1992-03-25 |
FI914405A (fi) | 1992-03-22 |
AU8462691A (en) | 1992-03-26 |
FI104168B1 (fi) | 1999-11-30 |
IE913318A1 (en) | 1992-02-25 |
IE66745B1 (en) | 1996-02-07 |
PT99014B (pt) | 1999-02-26 |
IL99536A0 (en) | 1992-08-18 |
CA2051766A1 (en) | 1992-03-22 |
EP0476682B1 (en) | 1995-02-01 |
JP2943089B2 (ja) | 1999-08-30 |
GR3014944T3 (en) | 1995-05-31 |
DE69107153T2 (de) | 1995-05-24 |
FI104168B (fi) | 1999-11-30 |
FI914405A0 (fi) | 1991-09-19 |
ES2067822T3 (es) | 1995-04-01 |
NZ239844A (en) | 1993-04-28 |
DE69107153D1 (de) | 1995-03-16 |
IL99536A (en) | 1995-10-31 |
AU637756B2 (en) | 1993-06-03 |
US5141959A (en) | 1992-08-25 |
PT99014A (pt) | 1992-08-31 |
MX9101163A (es) | 1992-05-04 |
JPH04270261A (ja) | 1992-09-25 |
ATE117979T1 (de) | 1995-02-15 |
ZA917531B (en) | 1992-07-29 |
OA09514A (en) | 1992-11-15 |
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