DE3163803D1 - 2-methyl-5-thiazole-methylamine and carboxamide derivatives - Google Patents

2-methyl-5-thiazole-methylamine and carboxamide derivatives

Info

Publication number
DE3163803D1
DE3163803D1 DE8181300599T DE3163803T DE3163803D1 DE 3163803 D1 DE3163803 D1 DE 3163803D1 DE 8181300599 T DE8181300599 T DE 8181300599T DE 3163803 T DE3163803 T DE 3163803T DE 3163803 D1 DE3163803 D1 DE 3163803D1
Authority
DE
Germany
Prior art keywords
methylamine
thiazole
methyl
carboxamide derivatives
tranquilising
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE8181300599T
Other languages
English (en)
Inventor
Ronald Ernest The Queen Grigg
Kitti The Queen S U Amornraksa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Application granted granted Critical
Publication of DE3163803D1 publication Critical patent/DE3163803D1/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/28—Radicals substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE8181300599T 1980-02-14 1981-02-13 2-methyl-5-thiazole-methylamine and carboxamide derivatives Expired DE3163803D1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8004985 1980-02-14

Publications (1)

Publication Number Publication Date
DE3163803D1 true DE3163803D1 (en) 1984-07-05

Family

ID=10511348

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8181300599T Expired DE3163803D1 (en) 1980-02-14 1981-02-13 2-methyl-5-thiazole-methylamine and carboxamide derivatives

Country Status (4)

Country Link
EP (1) EP0034481B1 (de)
JP (1) JPS56131571A (de)
AT (1) ATE7694T1 (de)
DE (1) DE3163803D1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4492597A (en) * 1981-05-25 1985-01-08 Kureha Kagaku Kogyo Kabushiki Kaisha 1,5-Diphenyl derivative of 1,2,4-triazole-3-carboxamide and herbicide containing the same
DE3316300A1 (de) * 1982-05-07 1983-11-24 Kureha Kagaku Kogyo K.K., Tokyo Heribizide zusammensetzung mit einem gehalt an einem derivat des 1,2,4-triazols als wirkstoff
IL84093A (en) * 1986-10-09 1992-09-06 Ciba Geigy Ag Aralkyl-4h-1,2,4-triazole derivatives,their preparation and pharmaceutical compositions containing them
CN112480090B (zh) * 2020-11-25 2023-07-21 浙江工业大学 一种含有吲哚啉和5-芳基呋喃骨架的化合物及其制备与应用

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2640828A (en) * 1949-04-13 1953-06-02 Smith Kline French Lab Nu, nu-disubstituted beta-haloethylamines
FR1219869A (fr) * 1958-04-12 1960-05-20 Hoechst Ag Procédé de préparation d'acides thiophène-carboxyliques et de leurs dérivés
FR1481686A (fr) * 1965-06-08 1967-05-19 Merck & Co Inc Procédé de fabrication de nu-(méthyl substitué)-anilines et thioanilides et leurs sels d'addition d'acides
GB1112128A (en) * 1965-12-22 1968-05-01 Bellon Labor Sa Roger New thiazolyl-diphenylmethane derivatives
GB1174411A (en) * 1966-03-02 1969-12-17 Aspro Nicholas Ltd Novel Benzothiophen Compounds, Compositions containing them and processes for their manufacture
GB1166364A (en) * 1966-11-25 1969-10-08 American Cyanamid Co N-(Tert-Aminoalkyl) Amide Derivatives and Process for Preparing the Same
FR1546183A (fr) * 1966-12-07 1968-11-15 Uniroyal Inc Carboxamidothiazoles, leurs substituants et dérivés, leurs procédés de fabrication ainsi que leurs applications et procédés d'application agriculturaux
FR1563735A (de) * 1967-12-08 1969-04-18
US4054585A (en) * 1972-03-06 1977-10-18 Uniroyal, Inc. Furan-3-carboxamide derivatives and method of preparing same
FR2176528B1 (de) * 1972-03-22 1975-04-25 Roussel Uclaf
JPS5749552B2 (de) * 1972-06-07 1982-10-22
FR2209557A1 (en) * 1972-12-12 1974-07-05 Roussel Uclaf Piperazo alkyl thiazolyl ketones/ethers - adrenolytics and antihypertensives prepd. from a piperazine and a halo alkyl thiazole
AR205339A1 (es) * 1973-03-12 1976-04-30 Icn Pharmaceuticals Sintesis de 1,2,4-triazolo-3-carboxamidas utiles como agentes antivirales
FR2323383A1 (fr) * 1975-09-12 1977-04-08 Roussel Uclaf Nouveaux derives de 5-thiazole methane amine, un procede pour leur preparation, leur application a titre de medicaments
SE7609666L (sv) * 1975-09-12 1977-03-13 Roussel Uclaf Sett att framstella nya 5-aminometyltiazolderivat
US4097265A (en) * 1975-12-30 1978-06-27 Chevron Research Company 3,5-Dimethyl-2-thienylcarboxanilide and 3,5-dimethyl-2-thienyl-(N-haloalkylthiocarboxanilide) herbicides
FR2361111A1 (fr) * 1976-08-11 1978-03-10 Roussel Uclaf Nouveaux derives de 5-thiazole alkylamine, un procede pour leur preparation et leur application comme medicaments
FR2382445A1 (fr) * 1977-03-03 1978-09-29 Philagro Sa Nouveaux derives de l'oxadiazole-1, 3, 4 et compositions fongicides les contenant
US4140698A (en) * 1977-07-25 1979-02-20 Syntex (Usa) Inc. 1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
US4199506A (en) * 1978-05-15 1980-04-22 Monsanto Company 2,4-Disubstituted-5-thiazolecarboxylic acids and derivatives

Also Published As

Publication number Publication date
EP0034481A1 (de) 1981-08-26
EP0034481B1 (de) 1984-05-30
JPS56131571A (en) 1981-10-15
ATE7694T1 (de) 1984-06-15

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Legal Events

Date Code Title Description
8339 Ceased/non-payment of the annual fee