DE1940572A1 - Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung - Google Patents

Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung

Info

Publication number
DE1940572A1
DE1940572A1 DE19691940572 DE1940572A DE1940572A1 DE 1940572 A1 DE1940572 A1 DE 1940572A1 DE 19691940572 DE19691940572 DE 19691940572 DE 1940572 A DE1940572 A DE 1940572A DE 1940572 A1 DE1940572 A1 DE 1940572A1
Authority
DE
Germany
Prior art keywords
thieno
pyrimidine
morpholino
radicals
general formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19691940572
Other languages
German (de)
English (en)
Inventor
Narr Dipl-Chem Dr Berthold
Woitun Dipl-Chem Dr Eberhard
Schroeter Dr Ludwig
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to BE754606D priority Critical patent/BE754606A/xx
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Priority to DE19691940572 priority patent/DE1940572A1/de
Priority to BG17335A priority patent/BG17969A3/xx
Priority to BG015244A priority patent/BG17591A3/xx
Priority to RO69224A priority patent/RO60647A/ro
Priority to RO69223A priority patent/RO60600A/ro
Priority to SU1669420A priority patent/SU428607A3/ru
Priority to SU701469618D priority patent/SU419032A3/ru
Priority to US00060933A priority patent/US3838121A/en
Priority to PH11712*UA priority patent/PH9574A/en
Priority to NL7011592A priority patent/NL7011592A/xx
Priority to CH1185070A priority patent/CH547299A/xx
Priority to CH341073A priority patent/CH546251A/xx
Priority to CH341173A priority patent/CH547304A/xx
Priority to CH340973A priority patent/CH547301A/xx
Priority to SE7010832A priority patent/SE386449B/xx
Priority to FI702170A priority patent/FI51939C/fi
Priority to CH340873A priority patent/CH547300A/xx
Priority to ES382549A priority patent/ES382549A1/es
Priority to ZA705482A priority patent/ZA705482B/xx
Priority to AT725170A priority patent/AT304531B/de
Priority to IL35078A priority patent/IL35078A/xx
Priority to GB3815070A priority patent/GB1311499A/en
Priority to ES382548A priority patent/ES382548A1/es
Priority to PL1970175151A priority patent/PL84258B1/pl
Priority to NO3045/70A priority patent/NO130538C/no
Priority to ES382552A priority patent/ES382552A1/es
Priority to PL1970142706A priority patent/PL83617B1/pl
Priority to ES382550A priority patent/ES382550A1/es
Priority to IE1025/70A priority patent/IE34687B1/xx
Priority to FR7029316A priority patent/FR2068478B1/fr
Priority to ES382551A priority patent/ES382551A1/es
Priority to PL1970175153A priority patent/PL84246B1/pl
Priority to JP45069666A priority patent/JPS519759B1/ja
Publication of DE1940572A1 publication Critical patent/DE1940572A1/de
Priority to US499460A priority patent/US3883651A/en
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DE19691940572 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung Pending DE1940572A1 (de)

Priority Applications (35)

Application Number Priority Date Filing Date Title
BE754606D BE754606A (fr) 1969-08-08 Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication
DE19691940572 DE1940572A1 (de) 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
BG17335A BG17969A3 (ru) 1969-08-08 1970-07-21
BG015244A BG17591A3 (bg) 1969-08-08 1970-07-21 Метод за получаване на нови 2- аминоалкил амино- тиено /3,2-д пиримидини
RO69224A RO60647A (ru) 1969-08-08 1970-07-28
RO69223A RO60600A (ru) 1969-08-08 1970-07-28
SU1669420A SU428607A3 (ru) 1969-08-08 1970-07-30
SU701469618D SU419032A3 (ru) 1969-08-08 1970-07-30 СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ 2-А!\\ИНО- АЛ КИЛАМИ НОТИЕНО-[3,2сг]-ПИРИЛ1ИДИ НА
US00060933A US3838121A (en) 1969-08-08 1970-08-04 2-(aminoalkyl-amino)-4-amino thieno(3,2-d)pyrimidines
PH11712*UA PH9574A (en) 1969-08-08 1970-08-04 2-(aminoalkyl-amino)-4-amino thieno(3,2-d)-pyrimidines
NL7011592A NL7011592A (ru) 1969-08-08 1970-08-05
CH340873A CH547300A (de) 1969-08-08 1970-08-06 Verfahren zur herstellung neuer 2-aminoalkylamino-thieno(3,2-d)pyrimidine.
CH341073A CH546251A (de) 1969-08-08 1970-08-06 Verfahren zur herstellung neuer 2-aminoalkylamino-thieno(3,2-d) pyrimidine.
CH341173A CH547304A (de) 1969-08-08 1970-08-06 Verfahren zur herstellung neuer 2-aminoalkylamino-thieno(3,2-d)pyrimidine.
CH340973A CH547301A (de) 1969-08-08 1970-08-06 Verfahren zur herstellung neuer 2-aminoalkylamino-thieno(3,2-d)pyrimidine.
SE7010832A SE386449B (sv) 1969-08-08 1970-08-06 Forfarande for framstellning av nya 2-aminoalkylamino-tieno(3,2-d)-pyrimidiner
FI702170A FI51939C (fi) 1969-08-08 1970-08-06 Menetelmä uusien verihiutaleiden kasautumista estävien 2-aminoalkyylia mino-tieno(3,2-d)pyrimidiinien valmistamiseksi
CH1185070A CH547299A (de) 1969-08-08 1970-08-06 Verfahren zur herstellung neuer 2-aminoalkylamino-thieno(3,2-d)pyrimidine.
PL1970175151A PL84258B1 (ru) 1969-08-08 1970-08-07
PL1970142706A PL83617B1 (ru) 1969-08-08 1970-08-07
AT725170A AT304531B (de) 1969-08-08 1970-08-07 Verfahren zur Herstellung von neuen 2-Aminoalkylamino-thieno[3,2-d]pyrimidinen und ihren Salzen
IL35078A IL35078A (en) 1969-08-08 1970-08-07 2-aminoalkylamino-thieno (3,2-d) pyrimidines and their salts,their preparation and pharmaceutical compositions containing them
GB3815070A GB1311499A (en) 1969-08-08 1970-08-07 Aminoalkylaminothienopyrimidines
ES382548A ES382548A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)piridinas.
ES382549A ES382549A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)piridinas.
NO3045/70A NO130538C (ru) 1969-08-08 1970-08-07
ES382552A ES382552A1 (es) 1969-08-08 1970-08-07 Procedimiento para la preparacion de nuevas 2-aminoalcohi- lamino tieno (3,2-d) pirimidinas.
ZA705482A ZA705482B (en) 1969-08-08 1970-08-07 Improvements relating to 2-aminoalkyl-amino-thieno(3,2-d)pyrimidines
ES382550A ES382550A1 (es) 1969-08-08 1970-08-07 Procedimiento para la preparacion de nuevas 2-aminoalcohi- lamino-tieno (3,2-d) pirimidinas.
IE1025/70A IE34687B1 (en) 1969-08-08 1970-08-07 Aminoalkylaminothieno-pyrimidines
FR7029316A FR2068478B1 (ru) 1969-08-08 1970-08-07
ES382551A ES382551A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)pirimidinas.
PL1970175153A PL84246B1 (ru) 1969-08-08 1970-08-07
JP45069666A JPS519759B1 (ru) 1969-08-08 1970-08-08
US499460A US3883651A (en) 1969-08-08 1974-08-22 Pharmaceutical compositions containing a 2-(aminoalkylamino)-4-amino-thieno{8 3,2-d{9 pyrimidine and method of use

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19691940572 DE1940572A1 (de) 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung

Publications (1)

Publication Number Publication Date
DE1940572A1 true DE1940572A1 (de) 1971-02-11

Family

ID=5742362

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19691940572 Pending DE1940572A1 (de) 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung

Country Status (6)

Country Link
BG (1) BG17969A3 (ru)
DE (1) DE1940572A1 (ru)
PL (3) PL84246B1 (ru)
RO (2) RO60647A (ru)
SU (2) SU428607A3 (ru)
ZA (1) ZA705482B (ru)

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1571146A1 (en) * 2002-12-10 2005-09-07 Ono Pharmaceutical Co., Ltd. Nitrogen-containing heterocyclic compounds and medicinal use thereof
WO2006111549A1 (de) * 2005-04-21 2006-10-26 Boehringer Ingelheim International Gmbh Dihydrothienopyrimidine zur behandlung von entzündlichen erkrankungen
US8604039B2 (en) 2006-04-19 2013-12-10 Boehringer Ingelheim International Gmbh Dihydrothienopyrimidines for the treatment of inflammatory diseases
US8637519B2 (en) 2007-10-19 2014-01-28 Boehringer Ingelheim International Gmbh Heterocycle-substituted piperazino-dihydrothienopyrimidines
US8754073B2 (en) 2007-10-19 2014-06-17 Boehringer Ingelheim International Gmbh Substituted piperazino-dihydrothienopyrimidines
US9090626B2 (en) 2007-10-19 2015-07-28 Boehringer Ingelheim International Gmbh Piperazino-dihydrothienopyrimidine derivatives
US9150586B2 (en) 2011-08-24 2015-10-06 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US10745411B2 (en) 2011-08-24 2020-08-18 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma

Cited By (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8153625B2 (en) 2002-12-10 2012-04-10 Ono Pharmaceutical Co., Ltd. Nitrogen-containing heterocyclic compounds and medicinal use thereof
EP1571146A1 (en) * 2002-12-10 2005-09-07 Ono Pharmaceutical Co., Ltd. Nitrogen-containing heterocyclic compounds and medicinal use thereof
EP1571146A4 (en) * 2002-12-10 2010-09-01 Ono Pharmaceutical Co NITROGENIC HETEROCYCLIC COMPOUNDS AND THEIR MEDICAL USE
US7723341B2 (en) 2005-04-21 2010-05-25 Boehringer Ingelheim International Gmbh Compounds for the treatment of inflammatory diseases
WO2006111549A1 (de) * 2005-04-21 2006-10-26 Boehringer Ingelheim International Gmbh Dihydrothienopyrimidine zur behandlung von entzündlichen erkrankungen
US8354531B2 (en) 2005-04-21 2013-01-15 Boehringer Ingelheim International Gmbh Compounds for the treatment of inflammatory diseases
EP2060575A1 (de) * 2006-04-19 2009-05-20 Boehringer Ingelheim International GmbH Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
EA013108B1 (ru) * 2006-04-19 2010-02-26 Бёрингер Ингельхайм Интернациональ Гмбх Дигидротиенопиримидины для лечения воспалительных заболеваний
US7511045B2 (en) 2006-04-19 2009-03-31 Boehringer Ingelheim International Gmbh Compounds for the treatment of inflammatory diseases
TWI380984B (zh) * 2006-04-19 2013-01-01 Boehringer Ingelheim Int 用於治療炎性疾病之新穎化合物
JP2008536890A (ja) * 2006-04-19 2008-09-11 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 炎症性疾患の治療用新規化合物
US8604039B2 (en) 2006-04-19 2013-12-10 Boehringer Ingelheim International Gmbh Dihydrothienopyrimidines for the treatment of inflammatory diseases
US8637519B2 (en) 2007-10-19 2014-01-28 Boehringer Ingelheim International Gmbh Heterocycle-substituted piperazino-dihydrothienopyrimidines
US8754073B2 (en) 2007-10-19 2014-06-17 Boehringer Ingelheim International Gmbh Substituted piperazino-dihydrothienopyrimidines
US9090626B2 (en) 2007-10-19 2015-07-28 Boehringer Ingelheim International Gmbh Piperazino-dihydrothienopyrimidine derivatives
US9115142B2 (en) 2007-10-19 2015-08-25 Boehringer Ingelheim International Gmbh Heterocycle-substituted piperazino-dihydrothienopyrimidines
US9150586B2 (en) 2011-08-24 2015-10-06 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US10745411B2 (en) 2011-08-24 2020-08-18 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma

Also Published As

Publication number Publication date
RO60647A (ru) 1976-08-15
SU419032A3 (ru) 1974-03-05
SU428607A3 (ru) 1974-05-15
PL84258B1 (ru) 1976-03-31
RO60600A (ru) 1976-09-15
PL83617B1 (ru) 1975-12-31
ZA705482B (en) 1971-05-27
BG17969A3 (ru) 1974-03-05
PL84246B1 (ru) 1976-03-31

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