DD151310A5 - Verfahren zur herstellung von 6-alpha-und 6-beta-substituierten penicillansaeurederivaten - Google Patents

Verfahren zur herstellung von 6-alpha-und 6-beta-substituierten penicillansaeurederivaten Download PDF

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Publication number
DD151310A5
DD151310A5 DD80221165A DD22116580A DD151310A5 DD 151310 A5 DD151310 A5 DD 151310A5 DD 80221165 A DD80221165 A DD 80221165A DD 22116580 A DD22116580 A DD 22116580A DD 151310 A5 DD151310 A5 DD 151310A5
Authority
DD
German Democratic Republic
Prior art keywords
acid
ester
formula
group
beta
Prior art date
Application number
DD80221165A
Other languages
German (de)
English (en)
Inventor
John E G Kemp
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DD151310A5 publication Critical patent/DD151310A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04—Preparation
    • C07D499/10—Modification of an amino radical directly attached in position 6
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DD80221165A 1979-05-19 1980-05-16 Verfahren zur herstellung von 6-alpha-und 6-beta-substituierten penicillansaeurederivaten DD151310A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7917505 1979-05-19

Publications (1)

Publication Number Publication Date
DD151310A5 true DD151310A5 (de) 1981-10-14

Family

ID=10505288

Family Applications (1)

Application Number Title Priority Date Filing Date
DD80221165A DD151310A5 (de) 1979-05-19 1980-05-16 Verfahren zur herstellung von 6-alpha-und 6-beta-substituierten penicillansaeurederivaten

Country Status (28)

Country Link
US (1) US4356122A (ja)
JP (1) JPS5941994B2 (ja)
KR (1) KR840000079B1 (ja)
AR (1) AR225038A1 (ja)
AT (1) AT366694B (ja)
AU (1) AU517488B2 (ja)
BE (1) BE883319A (ja)
CA (1) CA1140916A (ja)
CH (1) CH650262A5 (ja)
CS (1) CS214756B2 (ja)
DD (1) DD151310A5 (ja)
DE (1) DE3018847C2 (ja)
DK (1) DK155180A (ja)
ES (1) ES8105737A1 (ja)
FI (1) FI71562C (ja)
FR (1) FR2457293A1 (ja)
GR (1) GR68461B (ja)
IE (1) IE49804B1 (ja)
IL (1) IL60097A (ja)
IT (1) IT1140946B (ja)
LU (1) LU82458A1 (ja)
NL (1) NL180937C (ja)
NO (1) NO801473L (ja)
PH (1) PH15033A (ja)
PL (1) PL224188A1 (ja)
PT (1) PT71253A (ja)
SE (1) SE449995B (ja)
ZA (1) ZA802908B (ja)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA803742B (en) * 1979-07-02 1981-06-24 Beecham Group Ltd Penicillanic acid derivatives, their preparation and use
JPS6034969A (ja) * 1983-08-08 1985-02-22 Toyama Chem Co Ltd 新規なペニシラン酸誘導体およびその塩類

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5749555B2 (ja) * 1973-04-04 1982-10-22
US4282149A (en) * 1977-03-21 1981-08-04 Massachusetts Institute Of Technology Carbon and oxygen analogs of penicillin
US4265882A (en) * 1977-10-03 1981-05-05 Massachusetts Institute Of Technology Sulphur analogs of penicillins having a nucleophile substituted in the 6 and 7 position, respectively

Also Published As

Publication number Publication date
US4356122A (en) 1982-10-26
LU82458A1 (fr) 1980-10-08
FR2457293B1 (ja) 1983-05-20
KR840000079B1 (ko) 1984-02-08
AU517488B2 (en) 1981-08-06
DK155180A (da) 1980-11-20
IL60097A (en) 1983-02-23
IE49804B1 (en) 1985-12-25
PH15033A (en) 1982-05-20
FI71562B (fi) 1986-10-10
ES491612A0 (es) 1981-05-16
CA1140916A (en) 1983-02-08
SE449995B (sv) 1987-06-01
BE883319A (fr) 1980-11-14
FI801581A (fi) 1980-11-20
KR830002769A (ko) 1983-05-30
AT366694B (de) 1982-04-26
NL8002843A (nl) 1980-11-21
JPS55157588A (en) 1980-12-08
CS214756B2 (en) 1982-05-28
DE3018847C2 (de) 1982-09-30
NL180937C (nl) 1987-05-18
IT1140946B (it) 1986-10-10
AU5846880A (en) 1980-11-27
NL180937B (nl) 1986-12-16
IT8022104A0 (it) 1980-05-16
DE3018847A1 (de) 1980-12-11
CH650262A5 (de) 1985-07-15
ES8105737A1 (es) 1981-05-16
FI71562C (fi) 1987-01-19
ZA802908B (en) 1981-05-27
ATA259780A (de) 1981-09-15
JPS5941994B2 (ja) 1984-10-11
PT71253A (en) 1980-06-01
AR225038A1 (es) 1982-02-15
NO801473L (no) 1980-11-20
IL60097A0 (en) 1980-07-31
IE801024L (en) 1980-11-19
PL224188A1 (ja) 1981-02-13
SE8003676L (sv) 1980-11-20
FR2457293A1 (fr) 1980-12-19
GR68461B (ja) 1981-12-30

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