CY1116594T1 - Μεθοδος και ενδιαμεσα για την παρασκευη αναλογων καρβα-νουκλεοσιδικων υποκαταστατων - Google Patents

Μεθοδος και ενδιαμεσα για την παρασκευη αναλογων καρβα-νουκλεοσιδικων υποκαταστατων

Info

Publication number
CY1116594T1
CY1116594T1 CY20131100791T CY131100791T CY1116594T1 CY 1116594 T1 CY1116594 T1 CY 1116594T1 CY 20131100791 T CY20131100791 T CY 20131100791T CY 131100791 T CY131100791 T CY 131100791T CY 1116594 T1 CY1116594 T1 CY 1116594T1
Authority
CY
Cyprus
Prior art keywords
intermediates
carbon
preparation
nucleoside substitutes
nucleoside
Prior art date
Application number
CY20131100791T
Other languages
English (en)
Inventor
Thomas Butler
Aesop Cho
Benjamin R Graetz
Choung U Kim
Samuel E Metobo
Oliver L Saunders
Andrew W Waltman
Jie Xu
Lijun Zhang
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP10757699.3A external-priority patent/EP2480559B1/en
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of CY1116594T1 publication Critical patent/CY1116594T1/el

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Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Παρέχονται διαδικασίες και ενδιάμεσα για την σύνθεση νουκλεοσιδίων των ετερόκυκλων pyrrolo[Ι,2-f][1,2,4]triazinyl και imidazo[1,2-f][1,2,4]triazinyl του τύπου Ι.
CY20131100791T 2009-09-21 2013-09-12 Μεθοδος και ενδιαμεσα για την παρασκευη αναλογων καρβα-νουκλεοσιδικων υποκαταστατων CY1116594T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24429909A 2009-09-21 2009-09-21
EP10757699.3A EP2480559B1 (en) 2009-09-21 2010-09-20 Processes and intermediates for the preparation of 1'-cyano-carbanucleoside analogs

Publications (1)

Publication Number Publication Date
CY1116594T1 true CY1116594T1 (el) 2017-03-15

Family

ID=58459745

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20131100791T CY1116594T1 (el) 2009-09-21 2013-09-12 Μεθοδος και ενδιαμεσα για την παρασκευη αναλογων καρβα-νουκλεοσιδικων υποκαταστατων

Country Status (1)

Country Link
CY (1) CY1116594T1 (el)

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