CY1116272T1 - Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη - Google Patents

Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη

Info

Publication number
CY1116272T1
CY1116272T1 CY20151100089T CY151100089T CY1116272T1 CY 1116272 T1 CY1116272 T1 CY 1116272T1 CY 20151100089 T CY20151100089 T CY 20151100089T CY 151100089 T CY151100089 T CY 151100089T CY 1116272 T1 CY1116272 T1 CY 1116272T1
Authority
CY
Cyprus
Prior art keywords
methylnaltrexon
particles containing
pharmaceutical particles
pharmaceutical compositions
pharmaceutical
Prior art date
Application number
CY20151100089T
Other languages
English (en)
Inventor
Suketu P Sanghvi
Thomas A Boyd
Original Assignee
Progenics Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33299842&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1116272(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Progenics Pharmaceuticals, Inc. filed Critical Progenics Pharmaceuticals, Inc.
Publication of CY1116272T1 publication Critical patent/CY1116272T1/el

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    • AHUMAN NECESSITIES
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    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/047Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates having two or more hydroxy groups, e.g. sorbitol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
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    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
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    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
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    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Inorganic Chemistry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Otolaryngology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Gastroenterology & Hepatology (AREA)

Abstract

Περιγράφονται σταθερές φαρμακευτικές συνθέσεις, χρήσιμες για χορήγηση μεθυλναλτρεξόνης, καθώς και οι μέθοδοι για την κατασκευή τους. Κιτ, συμπεριλαμβανομένων αυτών των φαρμακευτικών συνθέσεων, παρέχονται επίσης.
CY20151100089T 2003-04-08 2015-01-28 Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη CY1116272T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US46161103P 2003-04-08 2003-04-08
EP04759349.6A EP1615646B2 (en) 2003-04-08 2004-04-08 Pharmaceutical formulations containing methylnaltrexone

Publications (1)

Publication Number Publication Date
CY1116272T1 true CY1116272T1 (el) 2017-02-08

Family

ID=33299842

Family Applications (3)

Application Number Title Priority Date Filing Date
CY20151100090T CY1116373T1 (el) 2003-04-08 2015-01-28 Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη
CY20151100091T CY1116372T1 (el) 2003-04-08 2015-01-28 Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη
CY20151100089T CY1116272T1 (el) 2003-04-08 2015-01-28 Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη

Family Applications Before (2)

Application Number Title Priority Date Filing Date
CY20151100090T CY1116373T1 (el) 2003-04-08 2015-01-28 Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη
CY20151100091T CY1116372T1 (el) 2003-04-08 2015-01-28 Φαρμακευτικα σκευασματα που περιεχουν μεθυλναλτρεξονη

Country Status (19)

Country Link
US (8) US20040266806A1 (el)
EP (3) EP1615646B2 (el)
JP (3) JP2006522818A (el)
CN (2) CN1767831B (el)
AU (2) AU2004229463B2 (el)
BR (1) BRPI0409133B8 (el)
CA (2) CA2811272C (el)
CY (3) CY1116373T1 (el)
DK (3) DK2368553T3 (el)
ES (3) ES2528631T3 (el)
HK (2) HK1082181A1 (el)
HR (3) HRP20150039T1 (el)
IL (1) IL171228A (el)
MX (1) MXPA05010817A (el)
PL (3) PL2368553T3 (el)
PT (3) PT1615646E (el)
RU (1) RU2362560C2 (el)
SI (3) SI2368553T1 (el)
WO (1) WO2004091623A1 (el)

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IL171228A (en) 2016-05-31
JP6262169B2 (ja) 2018-01-17
PL2368553T3 (pl) 2015-05-29
PT2368553E (pt) 2015-03-03
EP2368553B1 (en) 2014-12-31
EP1615646B1 (en) 2014-12-24
CY1116373T1 (el) 2017-02-08
HRP20150039T1 (hr) 2015-06-05
RU2362560C2 (ru) 2009-07-27
CN104383542B (zh) 2017-09-26
US20100261746A1 (en) 2010-10-14
US20170258911A1 (en) 2017-09-14
CA2811272A1 (en) 2004-10-28
AU2010202824B2 (en) 2013-05-02
ES2528631T3 (es) 2015-02-11
US20100261744A1 (en) 2010-10-14
US8552025B2 (en) 2013-10-08
PT1615646E (pt) 2015-02-12
US20190358328A1 (en) 2019-11-28
ES2527870T3 (es) 2015-02-02
CA2521379A1 (en) 2004-10-28
JP2006522818A (ja) 2006-10-05
CN104383542A (zh) 2015-03-04
US20100267758A1 (en) 2010-10-21
BRPI0409133A (pt) 2006-05-02
ES2528669T3 (es) 2015-02-11
SI1615646T2 (sl) 2022-11-30
PL1615646T5 (pl) 2022-12-19
US9669096B2 (en) 2017-06-06
ES2527870T5 (es) 2022-10-14
AU2004229463A1 (en) 2004-10-28
DK1615646T3 (en) 2015-02-02
SI2368553T1 (sl) 2015-05-29
US20040266806A1 (en) 2004-12-30
CA2521379C (en) 2013-07-02
BRPI0409133B1 (pt) 2019-09-03
HK1082181A1 (en) 2006-06-02

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