CR6698A - Antagonistas del factor liberador de corticotropina - Google Patents
Antagonistas del factor liberador de corticotropinaInfo
- Publication number
- CR6698A CR6698A CR6698A CR6698A CR6698A CR 6698 A CR6698 A CR 6698A CR 6698 A CR6698 A CR 6698A CR 6698 A CR6698 A CR 6698A CR 6698 A CR6698 A CR 6698A
- Authority
- CR
- Costa Rica
- Prior art keywords
- release factor
- factor antagonists
- disorders
- corticotropine
- antagonists
- Prior art date
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
- C07D213/643—2-Phenoxypyridines; Derivatives thereof
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- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
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Abstract
Consiste en antagonistas del factor liberador de corticotripina (CRF) que tienen las formulas I; II y III, donde las lineas de puntos, A, B, Y, Z, G, R3, R4, R5, R6, R16 Y R17, son como se han definido en la solicitud, y procedimientos para prepararlos. Estos compuestos y sus sales farmaceuticamente aceptables son utiles en el tratamiento de trastornos que incluyen trastornos del sistema nervioso central (CNS) y trastornos relacionados con el estres.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US17661100P | 2000-01-18 | 2000-01-18 |
Publications (1)
Publication Number | Publication Date |
---|---|
CR6698A true CR6698A (es) | 2004-01-14 |
Family
ID=22645084
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR6698A CR6698A (es) | 2000-01-18 | 2002-07-08 | Antagonistas del factor liberador de corticotropina |
Country Status (36)
Country | Link |
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US (1) | US6833378B2 (es) |
EP (1) | EP1263732A1 (es) |
JP (1) | JP2003520272A (es) |
KR (1) | KR20020063934A (es) |
CN (1) | CN1395566A (es) |
AP (1) | AP2002002583A0 (es) |
AR (1) | AR027221A1 (es) |
AU (1) | AU779995B2 (es) |
BG (1) | BG106853A (es) |
BR (1) | BR0107662A (es) |
CA (1) | CA2397633A1 (es) |
CO (1) | CO5271658A1 (es) |
CR (1) | CR6698A (es) |
CZ (1) | CZ20022390A3 (es) |
EA (2) | EA200300834A1 (es) |
EE (1) | EE200200400A (es) |
GT (1) | GT200100007A (es) |
HN (1) | HN2001000006A (es) |
HR (1) | HRP20020599A2 (es) |
HU (1) | HUP0204272A3 (es) |
IL (1) | IL150632A0 (es) |
IS (1) | IS6445A (es) |
MA (1) | MA26864A1 (es) |
MX (1) | MXPA02007047A (es) |
NO (1) | NO20023424L (es) |
OA (1) | OA12157A (es) |
PA (1) | PA8510001A1 (es) |
PE (1) | PE20011166A1 (es) |
PL (1) | PL357589A1 (es) |
SK (1) | SK10062002A3 (es) |
SV (1) | SV2002000289A (es) |
TN (1) | TNSN01008A1 (es) |
UY (1) | UY26544A1 (es) |
WO (1) | WO2001053263A1 (es) |
YU (1) | YU54402A (es) |
ZA (1) | ZA200205660B (es) |
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2001
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- 2001-01-05 SK SK1006-2002A patent/SK10062002A3/sk unknown
- 2001-01-05 AU AU23905/01A patent/AU779995B2/en not_active Ceased
- 2001-01-05 BR BR0107662-0A patent/BR0107662A/pt not_active IP Right Cessation
- 2001-01-05 MX MXPA02007047A patent/MXPA02007047A/es unknown
- 2001-01-05 EA EA200300834A patent/EA200300834A1/ru unknown
- 2001-01-05 OA OA1200200206A patent/OA12157A/en unknown
- 2001-01-05 PL PL01357589A patent/PL357589A1/xx not_active Application Discontinuation
- 2001-01-05 EE EEP200200400A patent/EE200200400A/xx unknown
- 2001-01-05 KR KR1020027009229A patent/KR20020063934A/ko not_active Application Discontinuation
- 2001-01-05 CN CN01803846A patent/CN1395566A/zh active Pending
- 2001-01-05 AP APAP/P/2002/002583A patent/AP2002002583A0/en unknown
- 2001-01-05 HU HU0204272A patent/HUP0204272A3/hu unknown
- 2001-01-05 JP JP2001553267A patent/JP2003520272A/ja active Pending
- 2001-01-05 IL IL15063201A patent/IL150632A0/xx unknown
- 2001-01-05 EP EP01900209A patent/EP1263732A1/en not_active Withdrawn
- 2001-01-05 CZ CZ20022390A patent/CZ20022390A3/cs unknown
- 2001-01-05 CA CA002397633A patent/CA2397633A1/en not_active Abandoned
- 2001-01-05 YU YU54402A patent/YU54402A/sh unknown
- 2001-01-05 EA EA200200688A patent/EA200200688A1/ru unknown
- 2001-01-12 HN HN2001000006A patent/HN2001000006A/es unknown
- 2001-01-16 AR ARP010100176A patent/AR027221A1/es not_active Application Discontinuation
- 2001-01-16 PE PE2001000038A patent/PE20011166A1/es not_active Application Discontinuation
- 2001-01-17 TN TNTNSN01008A patent/TNSN01008A1/fr unknown
- 2001-01-17 GT GT200100007A patent/GT200100007A/es unknown
- 2001-01-17 CO CO01003117A patent/CO5271658A1/es not_active Application Discontinuation
- 2001-01-17 US US09/761,995 patent/US6833378B2/en not_active Expired - Fee Related
- 2001-01-18 PA PA20018510001A patent/PA8510001A1/es unknown
- 2001-01-18 UY UY26544A patent/UY26544A1/es not_active Application Discontinuation
- 2001-01-22 SV SV2001000289A patent/SV2002000289A/es not_active Application Discontinuation
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2002
- 2002-06-20 BG BG106853A patent/BG106853A/bg unknown
- 2002-06-25 IS IS6445A patent/IS6445A/is unknown
- 2002-07-08 CR CR6698A patent/CR6698A/es not_active Application Discontinuation
- 2002-07-11 MA MA26728A patent/MA26864A1/fr unknown
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