CN106879256B - 2-氨基-苯并咪唑衍生物及其作为5-脂氧合酶和/或前列腺素e合成酶抑制剂的应用 - Google Patents
2-氨基-苯并咪唑衍生物及其作为5-脂氧合酶和/或前列腺素e合成酶抑制剂的应用 Download PDFInfo
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- CN106879256B CN106879256B CN201580053161.XA CN201580053161A CN106879256B CN 106879256 B CN106879256 B CN 106879256B CN 201580053161 A CN201580053161 A CN 201580053161A CN 106879256 B CN106879256 B CN 106879256B
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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| PCT/EP2015/067644 WO2016016421A1 (en) | 2014-07-31 | 2015-07-31 | 2-amino-benzimidazole derivatives and their use as 5-lipoxygenase and/or prostaglandin e synthase inhibitors |
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| JP6849197B2 (ja) * | 2016-02-12 | 2021-03-24 | ファーマクシス リミテッド | リジルオキシダーゼのインドールおよびアザインドールハロアリルアミン誘導体阻害剤およびその使用 |
| GB201617630D0 (en) | 2016-10-18 | 2016-11-30 | Cellcentric Ltd | Pharmaceutical compounds |
| CN107141282B (zh) * | 2017-03-29 | 2019-11-05 | 重庆文理学院 | 一种苯并咪唑杂氮环丁酮衍生物及其在抗肿瘤药物中的应用 |
| HRP20250272T1 (hr) | 2017-10-19 | 2025-04-25 | Teijin Pharma Limited | Derivati benzimidazola i njihova uporaba |
| GB201806320D0 (en) | 2018-04-18 | 2018-05-30 | Cellcentric Ltd | Process |
| JP2021534215A (ja) * | 2018-08-24 | 2021-12-09 | ゼニオプロ ゲーエムベーハー | 病的症状の治療における使用のための芳香族分子 |
| EP3939975A4 (en) * | 2019-03-15 | 2022-11-30 | Nippon Soda Co., Ltd. | HETEROCYCLIC COMPOUND AND AGRICULTURAL OR HORTICULTURAL BACTERICIDE |
| EP4081199A4 (en) * | 2019-12-23 | 2024-01-17 | SRI International | LIPOXYGENASE INHIBITORS |
| CN115667224A (zh) * | 2020-02-26 | 2023-01-31 | 斯克里普斯研究学院 | 具有抗炎活性的scl15a4小分子的抑制剂 |
| KR20240035820A (ko) | 2021-07-09 | 2024-03-18 | 플렉시움 인코포레이티드 | Ikzf2를 조절하는 아릴 화합물 및 약학 조성물 |
| WO2023107705A1 (en) | 2021-12-10 | 2023-06-15 | Incyte Corporation | Bicyclic amines as cdk12 inhibitors |
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- 2015-07-31 JP JP2017504727A patent/JP6785217B2/ja active Active
- 2015-07-31 SG SG11201700439VA patent/SG11201700439VA/en unknown
- 2015-07-31 CA CA2955565A patent/CA2955565A1/en not_active Abandoned
- 2015-07-31 BR BR112017001918A patent/BR112017001918A2/pt not_active Application Discontinuation
- 2015-07-31 ES ES15748009T patent/ES2795748T3/es active Active
- 2015-07-31 CN CN201580053161.XA patent/CN106879256B/zh active Active
- 2015-07-31 WO PCT/EP2015/067644 patent/WO2016016421A1/en not_active Ceased
- 2015-07-31 US US15/327,560 patent/US11447486B2/en active Active
- 2015-07-31 RU RU2017103148A patent/RU2732416C2/ru active
- 2015-07-31 AU AU2015295248A patent/AU2015295248B2/en active Active
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Also Published As
| Publication number | Publication date |
|---|---|
| RU2017103148A3 (https=) | 2018-10-04 |
| EP3177597B1 (en) | 2020-03-11 |
| JP6785217B2 (ja) | 2020-11-18 |
| US20170166563A1 (en) | 2017-06-15 |
| EP3177597A1 (en) | 2017-06-14 |
| ES2795748T3 (es) | 2020-11-24 |
| KR102494596B1 (ko) | 2023-01-31 |
| SG11201700439VA (en) | 2017-02-27 |
| US11447486B2 (en) | 2022-09-20 |
| AU2015295248B2 (en) | 2019-05-16 |
| WO2016016421A1 (en) | 2016-02-04 |
| AU2015295248A1 (en) | 2017-02-02 |
| CN106879256A (zh) | 2017-06-20 |
| RU2732416C2 (ru) | 2020-09-16 |
| RU2017103148A (ru) | 2018-08-30 |
| BR112017001918A2 (pt) | 2017-11-28 |
| KR20170045234A (ko) | 2017-04-26 |
| CA2955565A1 (en) | 2016-02-04 |
| JP2017522339A (ja) | 2017-08-10 |
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