CH628623A5 - Process for the preparation of N-aryl-N-(4-piperidinyl)arylacetamides - Google Patents
Process for the preparation of N-aryl-N-(4-piperidinyl)arylacetamides Download PDFInfo
- Publication number
- CH628623A5 CH628623A5 CH1194876A CH1194876A CH628623A5 CH 628623 A5 CH628623 A5 CH 628623A5 CH 1194876 A CH1194876 A CH 1194876A CH 1194876 A CH1194876 A CH 1194876A CH 628623 A5 CH628623 A5 CH 628623A5
- Authority
- CH
- Switzerland
- Prior art keywords
- group
- parts
- formula
- piperidinyl
- acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
- C07D211/66—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4 having a hetero atom as the second substituent in position 4
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US61513175A | 1975-09-23 | 1975-09-23 | |
US71375676A | 1976-08-12 | 1976-08-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
CH628623A5 true CH628623A5 (en) | 1982-03-15 |
Family
ID=27087421
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CH1194876A CH628623A5 (en) | 1975-09-23 | 1976-09-21 | Process for the preparation of N-aryl-N-(4-piperidinyl)arylacetamides |
Country Status (29)
Country | Link |
---|---|
JP (1) | JPS6016417B2 (fi) |
AT (1) | AT363935B (fi) |
AU (1) | AU510029B2 (fi) |
BG (1) | BG27543A3 (fi) |
CA (1) | CA1068271A (fi) |
CH (1) | CH628623A5 (fi) |
CS (1) | CS222663B2 (fi) |
DE (1) | DE2642856A1 (fi) |
DK (1) | DK150478C (fi) |
ES (1) | ES451768A1 (fi) |
FI (1) | FI61482C (fi) |
FR (1) | FR2325377A1 (fi) |
GB (1) | GB1539473A (fi) |
GR (1) | GR58469B (fi) |
HU (1) | HU172964B (fi) |
IE (1) | IE43802B1 (fi) |
IL (1) | IL50522A (fi) |
IT (1) | IT1073893B (fi) |
LU (1) | LU75837A1 (fi) |
NL (1) | NL187267C (fi) |
NO (1) | NO147672C (fi) |
NZ (1) | NZ181972A (fi) |
PH (1) | PH12497A (fi) |
PL (2) | PL192578A1 (fi) |
PT (1) | PT65631B (fi) |
RO (1) | RO70079A (fi) |
SE (1) | SE427839B (fi) |
SU (1) | SU747424A3 (fi) |
YU (1) | YU39973B (fi) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA765684B (en) * | 1975-09-23 | 1978-04-26 | Janssen Pharmaceutica Nv | Novel n-aryl-n-(1-l-4-piperidinyl)-arylacetamides |
JPS62260786A (ja) * | 1986-05-08 | 1987-11-13 | 株式会社ヘキトク | 燻瓦の製造ラインにおける焼成工程後の表面仕上げ装置 |
JO2769B1 (en) | 2005-10-26 | 2014-03-15 | جانسين فارماسوتيكا ان. في | Rapid decomposition of physiologically antagonistic agents of the 2-dopamine receptor |
JO2642B1 (en) | 2006-12-08 | 2012-06-17 | جانسين فارماسوتيكا ان. في | Dopamine 2 receptor antagonists are rapidly hydrolyzed |
JO2849B1 (en) | 2007-02-13 | 2015-03-15 | جانسين فارماسوتيكا ان. في | Dopamine 2 receptor antagonists are rapidly hydrolyzed |
US8933101B2 (en) | 2007-04-23 | 2015-01-13 | Janssen Pharmaceutica Nv | Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists |
JP2010525013A (ja) * | 2007-04-23 | 2010-07-22 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 高速解離性ドパミン2受容体アンタゴニストとしてのピリジン誘導体 |
DK2148873T3 (da) | 2007-04-23 | 2012-11-26 | Janssen Pharmaceutica Nv | 4-alkoxypyridazinderivater som hurtigt dissocierende dopamin 2- receptorantagonister |
US8530474B2 (en) | 2008-07-03 | 2013-09-10 | Janssen Pharmaceutica Nv | Substituted 6-(1-piperazinyl)-pyridazines as 5-HT6 receptor antagonists |
WO2010012758A1 (en) | 2008-07-31 | 2010-02-04 | Janssen Pharmaceutica Nv | Piperazin-1-yl-trifluoromethyl-substituted-pyridines as fast dissociating dopamine 2 receptor antagonists |
-
1976
- 1976-09-06 NO NO763054A patent/NO147672C/no unknown
- 1976-09-08 NZ NZ181972A patent/NZ181972A/xx unknown
- 1976-09-16 FR FR7627870A patent/FR2325377A1/fr active Granted
- 1976-09-17 AU AU17878/76A patent/AU510029B2/en not_active Expired
- 1976-09-20 LU LU75837A patent/LU75837A1/xx unknown
- 1976-09-20 CA CA261,551A patent/CA1068271A/en not_active Expired
- 1976-09-20 RO RO7687590A patent/RO70079A/ro unknown
- 1976-09-21 IT IT51370/76A patent/IT1073893B/it active
- 1976-09-21 GB GB39099/76A patent/GB1539473A/en not_active Expired
- 1976-09-21 JP JP51112527A patent/JPS6016417B2/ja not_active Expired
- 1976-09-21 IL IL50522A patent/IL50522A/xx unknown
- 1976-09-21 GR GR51742A patent/GR58469B/el unknown
- 1976-09-21 CH CH1194876A patent/CH628623A5/de not_active IP Right Cessation
- 1976-09-22 PL PL19257876A patent/PL192578A1/xx not_active IP Right Cessation
- 1976-09-22 YU YU2336/76A patent/YU39973B/xx unknown
- 1976-09-22 IE IE2095/76A patent/IE43802B1/en unknown
- 1976-09-22 FI FI762698A patent/FI61482C/fi not_active IP Right Cessation
- 1976-09-22 HU HU76JA00000767A patent/HU172964B/hu not_active IP Right Cessation
- 1976-09-22 SE SE7610501A patent/SE427839B/xx not_active IP Right Cessation
- 1976-09-22 NL NLAANVRAGE7610513,A patent/NL187267C/xx not_active IP Right Cessation
- 1976-09-22 AT AT0702976A patent/AT363935B/de not_active IP Right Cessation
- 1976-09-22 PT PT65631A patent/PT65631B/pt unknown
- 1976-09-22 CS CS766139A patent/CS222663B2/cs unknown
- 1976-09-22 ES ES451768A patent/ES451768A1/es not_active Expired
- 1976-09-22 DK DK427876A patent/DK150478C/da active
- 1976-09-22 PL PL1976216213A patent/PL117323B1/pl unknown
- 1976-09-22 PH PH18928A patent/PH12497A/en unknown
- 1976-09-23 DE DE19762642856 patent/DE2642856A1/de active Granted
- 1976-09-23 BG BG7634265A patent/BG27543A3/xx unknown
- 1976-09-23 SU SU762405548A patent/SU747424A3/ru active
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DE2503815C2 (de) | Indazol-Derivate, Verfahren zu ihrer Herstellung und Arzneimittel | |
DD267728A5 (de) | Verfahren zur herstellung von arylcyclobutylalkylamin-derivaten | |
CH628623A5 (en) | Process for the preparation of N-aryl-N-(4-piperidinyl)arylacetamides | |
DE2047658A1 (fi) | ||
DD149511A5 (de) | Verfahren zur herstellung von 9-aminoalkylfluorenen | |
EP0110869B1 (de) | Thienylessigsäureamidderivate und pharmazeutisch verträgliche Säureadditionssalze hiervon sowie Verfahren zu deren Herstellung | |
DE3642497A1 (de) | Substituierte aminopropionsaeureamide, verfahren zu ihrer herstellung, diese enthaltende mittel und ihre verwendung sowie die bei der herstellung anfallenden neuen zwischenprodukte | |
DE69803979T2 (de) | Verfahren zur herstellung von carboxamido-4-azasteroiden | |
DE2515146A1 (de) | Carbonsaeureamide, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel | |
DE3889208T2 (de) | Thioformamid-Derivate. | |
DE812669C (de) | Verfahren zur Herstellung von 1-Aryl-cyclopenten-(3)-1-nitrilen, deren Carbonsaeuren, deren basischen Estern und Amiden und deren Salzen | |
DE1793612C (fi) | ||
DE2943809A1 (de) | 1-mercaptoacylpiperazin-2-carbonsaeure-verbindungen und ihre salze, verfahren zu ihrer herstellung und ihre verwendung bei der bekaempfung von hypertonie | |
DE2430510C3 (de) | 16,17-Dihydroapovincaminsäureamide, Verfahren zu deren Herstellung und Arzneimittel, welche diese Verbingungen enthalten | |
DE2435816A1 (de) | Substituierte nitrobenzophenonderivate und ihre salze sowie ihre verwendung und verfahren zur herstellung derselben | |
DE2720915C2 (de) | N↓1↓-Acyl-2-hydroxy-1,3-diaminopropane und Arzneimittel mit diesen Verbindungen als Wirkstoff | |
DD151447A1 (de) | Verfahren zur herstellung von amidinen und deren salzen | |
CH513158A (de) | Verfahren zur Herstellung von Pyrrolinverbindungen | |
AT234691B (de) | Verfahren zur Herstellung von neuen Piperidinderivaten | |
DE2338409A1 (de) | Neues verfahren zur herstellung von 2-acylamino-benzylaminen | |
DD149664A5 (de) | Verfahren zur herstellung von 1,1'-biphenyl-2-yl-alkylamin-derivaten | |
DE2166258C3 (de) | Aminoalkohole, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneipräparate | |
DE2429373A1 (de) | Verfahren zur herstellung neuer heterocyclischer verbindungen | |
DE844897C (de) | Verfahren zur Herstellung von Diamidinderivaten | |
DE2104312C3 (de) | (α,α,β,β-Tetrafluorphenäthyl)-α,α-dimethylbenzylaminderivate, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PL | Patent ceased |