CA3128711A1 - Bakuchiol compositions for treatment of post inflammatory hyperpigmentation - Google Patents
Bakuchiol compositions for treatment of post inflammatory hyperpigmentation Download PDFInfo
- Publication number
- CA3128711A1 CA3128711A1 CA3128711A CA3128711A CA3128711A1 CA 3128711 A1 CA3128711 A1 CA 3128711A1 CA 3128711 A CA3128711 A CA 3128711A CA 3128711 A CA3128711 A CA 3128711A CA 3128711 A1 CA3128711 A1 CA 3128711A1
- Authority
- CA
- Canada
- Prior art keywords
- bakuchiol
- inflammatory
- composition
- pih
- skin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- LFYJSSARVMHQJB-QIXNEVBVSA-N bakuchiol Chemical compound CC(C)=CCC[C@@](C)(C=C)\C=C\C1=CC=C(O)C=C1 LFYJSSARVMHQJB-QIXNEVBVSA-N 0.000 title claims abstract description 209
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- 229920002647 polyamide Polymers 0.000 description 1
- 229920000573 polyethylene Polymers 0.000 description 1
- 229940050929 polyethylene glycol 3350 Drugs 0.000 description 1
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- 239000008057 potassium phosphate buffer Substances 0.000 description 1
- 238000001556 precipitation Methods 0.000 description 1
- 238000009597 pregnancy test Methods 0.000 description 1
- BDERNNFJNOPAEC-UHFFFAOYSA-N propan-1-ol Chemical compound CCCO BDERNNFJNOPAEC-UHFFFAOYSA-N 0.000 description 1
- 230000000069 prophylactic effect Effects 0.000 description 1
- 238000011321 prophylaxis Methods 0.000 description 1
- 239000000473 propyl gallate Substances 0.000 description 1
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- 229940075579 propyl gallate Drugs 0.000 description 1
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 description 1
- 102000004169 proteins and genes Human genes 0.000 description 1
- 108090000623 proteins and genes Proteins 0.000 description 1
- 239000012673 purified plant extract Substances 0.000 description 1
- 238000010992 reflux Methods 0.000 description 1
- 230000003252 repetitive effect Effects 0.000 description 1
- 238000011160 research Methods 0.000 description 1
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- 229930182490 saponin Natural products 0.000 description 1
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- 238000006748 scratching Methods 0.000 description 1
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- 229930000044 secondary metabolite Natural products 0.000 description 1
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- 201000000849 skin cancer Diseases 0.000 description 1
- 229910000029 sodium carbonate Inorganic materials 0.000 description 1
- 235000017550 sodium carbonate Nutrition 0.000 description 1
- 235000019812 sodium carboxymethyl cellulose Nutrition 0.000 description 1
- 229920001027 sodium carboxymethylcellulose Polymers 0.000 description 1
- FQENQNTWSFEDLI-UHFFFAOYSA-J sodium diphosphate Chemical compound [Na+].[Na+].[Na+].[Na+].[O-]P([O-])(=O)OP([O-])([O-])=O FQENQNTWSFEDLI-UHFFFAOYSA-J 0.000 description 1
- HRZFUMHJMZEROT-UHFFFAOYSA-L sodium disulfite Chemical compound [Na+].[Na+].[O-]S(=O)S([O-])(=O)=O HRZFUMHJMZEROT-UHFFFAOYSA-L 0.000 description 1
- 239000000176 sodium gluconate Substances 0.000 description 1
- 235000012207 sodium gluconate Nutrition 0.000 description 1
- 229940005574 sodium gluconate Drugs 0.000 description 1
- 229940010747 sodium hyaluronate Drugs 0.000 description 1
- 235000019333 sodium laurylsulphate Nutrition 0.000 description 1
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- 235000010262 sodium metabisulphite Nutrition 0.000 description 1
- 235000019832 sodium triphosphate Nutrition 0.000 description 1
- OGBHACNFHJJTQT-UHFFFAOYSA-M sodium;4-butoxycarbonylphenolate Chemical compound [Na+].CCCCOC(=O)C1=CC=C([O-])C=C1 OGBHACNFHJJTQT-UHFFFAOYSA-M 0.000 description 1
- 229950011392 sorbitan stearate Drugs 0.000 description 1
- 239000000600 sorbitol Substances 0.000 description 1
- 239000008223 sterile water Substances 0.000 description 1
- 235000021286 stilbenes Nutrition 0.000 description 1
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- RTKIYNMVFMVABJ-UHFFFAOYSA-L thimerosal Chemical compound [Na+].CC[Hg]SC1=CC=CC=C1C([O-])=O RTKIYNMVFMVABJ-UHFFFAOYSA-L 0.000 description 1
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- 208000037816 tissue injury Diseases 0.000 description 1
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- 229940100611 topical cream Drugs 0.000 description 1
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- 230000002110 toxicologic effect Effects 0.000 description 1
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- 235000010487 tragacanth Nutrition 0.000 description 1
- 239000000196 tragacanth Substances 0.000 description 1
- 229940116362 tragacanth Drugs 0.000 description 1
- GYDJEQRTZSCIOI-LJGSYFOKSA-N tranexamic acid Chemical compound NC[C@H]1CC[C@H](C(O)=O)CC1 GYDJEQRTZSCIOI-LJGSYFOKSA-N 0.000 description 1
- 229960000401 tranexamic acid Drugs 0.000 description 1
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- HTJNEBVCZXHBNJ-XCTPRCOBSA-H trimagnesium;(2r)-2-[(1s)-1,2-dihydroxyethyl]-3,4-dihydroxy-2h-furan-5-one;diphosphate Chemical compound [Mg+2].[Mg+2].[Mg+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O.OC[C@H](O)[C@H]1OC(=O)C(O)=C1O HTJNEBVCZXHBNJ-XCTPRCOBSA-H 0.000 description 1
- 239000001226 triphosphate Substances 0.000 description 1
- LENZDBCJOHFCAS-UHFFFAOYSA-N tris Chemical compound OCC(N)(CO)CO LENZDBCJOHFCAS-UHFFFAOYSA-N 0.000 description 1
- 230000007306 turnover Effects 0.000 description 1
- 238000009281 ultraviolet germicidal irradiation Methods 0.000 description 1
- 229930195735 unsaturated hydrocarbon Chemical group 0.000 description 1
- 210000002700 urine Anatomy 0.000 description 1
- 235000015112 vegetable and seed oil Nutrition 0.000 description 1
- 235000013311 vegetables Nutrition 0.000 description 1
- 230000000007 visual effect Effects 0.000 description 1
- 235000019154 vitamin C Nutrition 0.000 description 1
- 239000011718 vitamin C Substances 0.000 description 1
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- 229940046009 vitamin E Drugs 0.000 description 1
- 235000019165 vitamin E Nutrition 0.000 description 1
- 239000011709 vitamin E Substances 0.000 description 1
- 150000003712 vitamin E derivatives Chemical class 0.000 description 1
- 238000007704 wet chemistry method Methods 0.000 description 1
- 239000012224 working solution Substances 0.000 description 1
- 229910001845 yogo sapphire Inorganic materials 0.000 description 1
- UHVMMEOXYDMDKI-JKYCWFKZSA-L zinc;1-(5-cyanopyridin-2-yl)-3-[(1s,2s)-2-(6-fluoro-2-hydroxy-3-propanoylphenyl)cyclopropyl]urea;diacetate Chemical compound [Zn+2].CC([O-])=O.CC([O-])=O.CCC(=O)C1=CC=C(F)C([C@H]2[C@H](C2)NC(=O)NC=2N=CC(=CC=2)C#N)=C1O UHVMMEOXYDMDKI-JKYCWFKZSA-L 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
- A61K31/05—Phenols
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/60—Salicylic acid; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/16—Emollients or protectives, e.g. against radiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/18—Antioxidants, e.g. antiradicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Toxicology (AREA)
- Biochemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Emergency Medicine (AREA)
- Birds (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Cosmetics (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161438890P | 2011-02-02 | 2011-02-02 | |
| US61/438,890 | 2011-02-02 | ||
| PCT/US2011/026594 WO2012105990A1 (en) | 2011-02-02 | 2011-03-01 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
| USPCT/US2011/026594 | 2011-03-01 | ||
| CA2826262A CA2826262C (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2826262A Division CA2826262C (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3128711A1 true CA3128711A1 (en) | 2012-08-09 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2826262A Active CA2826262C (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
| CA3128711A Pending CA3128711A1 (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
| CA3128715A Pending CA3128715A1 (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
| CA3128718A Pending CA3128718A1 (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2826262A Active CA2826262C (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3128715A Pending CA3128715A1 (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
| CA3128718A Pending CA3128718A1 (en) | 2011-02-02 | 2012-02-02 | Bakuchiol compositions for treatment of post inflammatory hyperpigmentation |
Country Status (8)
| Country | Link |
|---|---|
| KR (5) | KR101954118B1 (ko) |
| CN (2) | CN105147533B (ko) |
| AU (1) | AU2012212153B9 (ko) |
| BR (1) | BR112013019798A2 (ko) |
| CA (4) | CA2826262C (ko) |
| HK (1) | HK1215792A1 (ko) |
| MX (1) | MX350719B (ko) |
| WO (1) | WO2012105990A1 (ko) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10471035B2 (en) | 2014-10-20 | 2019-11-12 | Sunny BioDiscovery | Compositions and methods for using esters of meroterpenes and of other resveratrol analogues |
| CN105675741A (zh) * | 2015-12-30 | 2016-06-15 | 成都九芝堂金鼎药业有限公司 | 一种测定生发丸中有效成分含量的方法 |
| KR20190116858A (ko) | 2018-04-05 | 2019-10-15 | 주식회사 엑소코바이오 | 줄기세포 유래의 엑소좀 및/또는 세포외 소포체를 유효성분으로 포함하는 조성물의 염증후 과색소침착의 예방, 완화, 감소 내지는 제거 용도 |
| CN111544317B (zh) * | 2020-04-29 | 2022-01-14 | 珀莱雅化妆品股份有限公司 | 一种抗衰老组合物阳离子纳米脂质体及其制备方法与应用 |
| CN114478196B (zh) * | 2021-01-27 | 2023-11-10 | 江苏巴帝恩生物科技有限公司 | 一种从春榆根里提取补骨脂酚并纯化的方法及在化妆品中的应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2617473B2 (ja) | 1987-06-30 | 1997-06-04 | キヤノン株式会社 | 情報入力装置 |
| KR20130125411A (ko) * | 2005-05-09 | 2013-11-18 | 유니젠, 인크. | 바쿠치올의 조성물 및 그것의 제조방법 |
| WO2008143761A1 (en) * | 2007-05-14 | 2008-11-27 | Sytheon Ltd. | Sunscreen compositions and methods |
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2011
- 2011-03-01 WO PCT/US2011/026594 patent/WO2012105990A1/en active Application Filing
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2012
- 2012-02-02 CA CA2826262A patent/CA2826262C/en active Active
- 2012-02-02 KR KR1020137022953A patent/KR101954118B1/ko active IP Right Grant
- 2012-02-02 KR KR1020237013482A patent/KR102642352B1/ko active IP Right Grant
- 2012-02-02 CN CN201510390680.7A patent/CN105147533B/zh active Active
- 2012-02-02 CA CA3128711A patent/CA3128711A1/en active Pending
- 2012-02-02 KR KR1020197005663A patent/KR102156731B1/ko active IP Right Grant
- 2012-02-02 CA CA3128715A patent/CA3128715A1/en active Pending
- 2012-02-02 KR KR1020217038833A patent/KR102525516B1/ko active IP Right Grant
- 2012-02-02 AU AU2012212153A patent/AU2012212153B9/en active Active
- 2012-02-02 CN CN201280015007.XA patent/CN103458882B/zh active Active
- 2012-02-02 MX MX2013008890A patent/MX350719B/es active IP Right Grant
- 2012-02-02 KR KR1020207026173A patent/KR102333655B1/ko active IP Right Grant
- 2012-02-02 CA CA3128718A patent/CA3128718A1/en active Pending
- 2012-02-02 BR BR112013019798A patent/BR112013019798A2/pt not_active Application Discontinuation
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2016
- 2016-04-01 HK HK16103749.0A patent/HK1215792A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN103458882B (zh) | 2015-08-05 |
| AU2012212153A1 (en) | 2013-08-29 |
| KR102525516B1 (ko) | 2023-04-24 |
| CN105147533B (zh) | 2018-07-31 |
| KR20210145864A (ko) | 2021-12-02 |
| CN105147533A (zh) | 2015-12-16 |
| WO2012105990A1 (en) | 2012-08-09 |
| BR112013019798A2 (pt) | 2017-07-04 |
| KR20230058727A (ko) | 2023-05-03 |
| CA2826262C (en) | 2021-10-26 |
| KR101954118B1 (ko) | 2019-03-05 |
| KR20140008364A (ko) | 2014-01-21 |
| HK1215792A1 (zh) | 2016-09-15 |
| KR102333655B1 (ko) | 2021-12-01 |
| KR20190025740A (ko) | 2019-03-11 |
| MX350719B (es) | 2017-09-14 |
| AU2012212153B9 (en) | 2017-05-11 |
| KR102642352B1 (ko) | 2024-02-28 |
| KR102156731B1 (ko) | 2020-09-16 |
| AU2012212153B2 (en) | 2017-04-06 |
| MX2013008890A (es) | 2013-10-17 |
| CA3128718A1 (en) | 2012-08-09 |
| CN103458882A (zh) | 2013-12-18 |
| CA2826262A1 (en) | 2012-08-09 |
| KR20200108120A (ko) | 2020-09-16 |
| CA3128715A1 (en) | 2012-08-09 |
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