CA2412864A1 - Methodes de preparation et utilisation, et formulations pharmaceutiques renfermant 7.alpha.,11.beta.-dimethyl-17.beta.-hydroxyestra-4,14-dien-3-one et leurs 17-esters - Google Patents
Methodes de preparation et utilisation, et formulations pharmaceutiques renfermant 7.alpha.,11.beta.-dimethyl-17.beta.-hydroxyestra-4,14-dien-3-one et leurs 17-esters Download PDFInfo
- Publication number
- CA2412864A1 CA2412864A1 CA002412864A CA2412864A CA2412864A1 CA 2412864 A1 CA2412864 A1 CA 2412864A1 CA 002412864 A CA002412864 A CA 002412864A CA 2412864 A CA2412864 A CA 2412864A CA 2412864 A1 CA2412864 A1 CA 2412864A1
- Authority
- CA
- Canada
- Prior art keywords
- beta
- androgen
- hydroxyestra
- dien
- alpha
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Abstract
L'invention concerne des procédés d'utilisation de 7 alpha ,11ss-diméthyl-17ss-hydroxyestra-4,14-dièn-3-one (III), de 7 alpha -méthyl-17ss hydroxyestra-4,14-dièn-3-one, et des esters en position 17 de ces composés destinés à diverses thérapies hormonales, des formes de dosage orale et parentérale contenant ces composés actifs, ainsi que leurs procédés de préparation.
Applications Claiming Priority (7)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US19353000P | 2000-03-31 | 2000-03-31 | |
US60/193,530 | 2000-03-31 | ||
US19444000P | 2000-04-04 | 2000-04-04 | |
US60/194,440 | 2000-04-04 | ||
PCT/US2001/010293 WO2001074839A2 (fr) | 2000-03-31 | 2001-03-30 | Procedes de preparation et d'utilisation de7$g(a),11?-dimethyl-17?-hydroxy-4-estren-3-one 17?-$i(trans)-4-$i(n)-butylcyclohexane carboxylate et 7$g(a),11?-dimethyl-17?-hydroxyestr-4-en-3-one 17-undecanoate |
WOPCT/US01/10293 | 2001-03-30 | ||
PCT/US2002/009886 WO2003045398A1 (fr) | 2001-03-30 | 2002-03-29 | Procedes de fabrication de formulations pharmaceutiques comprenant du 7alpha, 11beta-dimethy-17beta-hydroxyestra-4, 14-dien-3-one et des esters en position 17 de ce compose |
Publications (2)
Publication Number | Publication Date |
---|---|
CA2412864A1 true CA2412864A1 (fr) | 2002-03-29 |
CA2412864C CA2412864C (fr) | 2010-06-22 |
Family
ID=27359057
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA2412864A Expired - Fee Related CA2412864C (fr) | 2000-03-31 | 2002-03-29 | Methodes de preparation et utilisation, et formulations pharmaceutiques renfermant 7.alpha.,11.beta.-dimethyl-17.beta.-hydroxyestra-4,14-dien-3-one et leurs 17-esters |
Country Status (1)
Country | Link |
---|---|
CA (1) | CA2412864C (fr) |
-
2002
- 2002-03-29 CA CA2412864A patent/CA2412864C/fr not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
CA2412864C (fr) | 2010-06-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
MKLA | Lapsed |
Effective date: 20220301 |
|
MKLA | Lapsed |
Effective date: 20200831 |