CA2156065A1 - Immunomodulateurs a base d'uree et d'amide macrocyclique - Google Patents
Immunomodulateurs a base d'uree et d'amide macrocycliqueInfo
- Publication number
- CA2156065A1 CA2156065A1 CA002156065A CA2156065A CA2156065A1 CA 2156065 A1 CA2156065 A1 CA 2156065A1 CA 002156065 A CA002156065 A CA 002156065A CA 2156065 A CA2156065 A CA 2156065A CA 2156065 A1 CA2156065 A1 CA 2156065A1
- Authority
- CA
- Canada
- Prior art keywords
- ethyl
- compound
- configuration
- och3
- och2c
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US3295893A | 1993-03-17 | 1993-03-17 | |
US08/032,958 | 1993-03-17 | ||
US14941993A | 1993-11-09 | 1993-11-09 | |
US08/149,419 | 1993-11-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2156065A1 true CA2156065A1 (fr) | 1994-09-29 |
Family
ID=26709099
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002156065A Abandoned CA2156065A1 (fr) | 1993-03-17 | 1994-03-11 | Immunomodulateurs a base d'uree et d'amide macrocyclique |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP0689545A4 (fr) |
JP (1) | JPH08507789A (fr) |
CA (1) | CA2156065A1 (fr) |
WO (1) | WO1994021642A1 (fr) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6376517B1 (en) * | 1998-08-14 | 2002-04-23 | Gpi Nil Holdings, Inc. | Pipecolic acid derivatives for vision and memory disorders |
US6121257A (en) * | 1999-03-31 | 2000-09-19 | Abbott Laboratories | Sulfamate containing macrocyclic immunomodulators |
GB0125443D0 (en) | 2001-10-23 | 2001-12-12 | Novartis Ag | Organic Compounds |
CA2498191C (fr) | 2002-09-18 | 2012-04-10 | Trustees Of The University Of Pennsylvania | Methode d'inhibition de la neovascularisation choroidienne |
US7920906B2 (en) | 2005-03-10 | 2011-04-05 | Dexcom, Inc. | System and methods for processing analyte sensor data for sensor calibration |
US9247900B2 (en) | 2004-07-13 | 2016-02-02 | Dexcom, Inc. | Analyte sensor |
US20070045902A1 (en) | 2004-07-13 | 2007-03-01 | Brauker James H | Analyte sensor |
US8170803B2 (en) | 2004-07-13 | 2012-05-01 | Dexcom, Inc. | Transcutaneous analyte sensor |
TW200637552A (en) * | 2005-01-20 | 2006-11-01 | Array Biopharma Inc | Macrocyclic analogs for the treatment of immunoregulatory disorders and respiratory diseases |
EP1853259A1 (fr) | 2005-02-09 | 2007-11-14 | Macusight, Inc. | Formulations pour un traitement oculaire |
WO2007092620A2 (fr) | 2006-02-09 | 2007-08-16 | Macusight, Inc. | Formulations stables et leurs procedes de preparation et d'utilisation |
AU2007230964B2 (en) | 2006-03-23 | 2012-07-19 | Santen Pharmaceutical Co., Ltd. | Formulations and methods for vascular permeability-related diseases or conditions |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5565560A (en) * | 1991-05-13 | 1996-10-15 | Merck & Co., Inc. | O-Aryl,O-alkyl,O-alkenyl and O-alkynylmacrolides having immunosuppressive activity |
US5250678A (en) * | 1991-05-13 | 1993-10-05 | Merck & Co., Inc. | O-aryl, O-alkyl, O-alkenyl and O-alkynylmacrolides having immunosuppressive activity |
US5561228A (en) * | 1991-09-05 | 1996-10-01 | Abbott Laboratories | Macrocyclic immunomodulators |
-
1994
- 1994-03-11 WO PCT/US1994/002692 patent/WO1994021642A1/fr not_active Application Discontinuation
- 1994-03-11 JP JP6521135A patent/JPH08507789A/ja active Pending
- 1994-03-11 EP EP94910923A patent/EP0689545A4/fr not_active Withdrawn
- 1994-03-11 CA CA002156065A patent/CA2156065A1/fr not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP0689545A1 (fr) | 1996-01-03 |
EP0689545A4 (fr) | 1996-04-24 |
WO1994021642A1 (fr) | 1994-09-29 |
JPH08507789A (ja) | 1996-08-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FZDE | Dead |