CA2156065A1 - Immunomodulateurs a base d'uree et d'amide macrocyclique - Google Patents

Immunomodulateurs a base d'uree et d'amide macrocyclique

Info

Publication number
CA2156065A1
CA2156065A1 CA002156065A CA2156065A CA2156065A1 CA 2156065 A1 CA2156065 A1 CA 2156065A1 CA 002156065 A CA002156065 A CA 002156065A CA 2156065 A CA2156065 A CA 2156065A CA 2156065 A1 CA2156065 A1 CA 2156065A1
Authority
CA
Canada
Prior art keywords
ethyl
compound
configuration
och3
och2c
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002156065A
Other languages
English (en)
Inventor
Rolf Wagner
Jay R. Luly
Yat Sun Or
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2156065A1 publication Critical patent/CA2156065A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
CA002156065A 1993-03-17 1994-03-11 Immunomodulateurs a base d'uree et d'amide macrocyclique Abandoned CA2156065A1 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US3295893A 1993-03-17 1993-03-17
US08/032,958 1993-03-17
US14941993A 1993-11-09 1993-11-09
US08/149,419 1993-11-09

Publications (1)

Publication Number Publication Date
CA2156065A1 true CA2156065A1 (fr) 1994-09-29

Family

ID=26709099

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002156065A Abandoned CA2156065A1 (fr) 1993-03-17 1994-03-11 Immunomodulateurs a base d'uree et d'amide macrocyclique

Country Status (4)

Country Link
EP (1) EP0689545A4 (fr)
JP (1) JPH08507789A (fr)
CA (1) CA2156065A1 (fr)
WO (1) WO1994021642A1 (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6376517B1 (en) * 1998-08-14 2002-04-23 Gpi Nil Holdings, Inc. Pipecolic acid derivatives for vision and memory disorders
US6121257A (en) * 1999-03-31 2000-09-19 Abbott Laboratories Sulfamate containing macrocyclic immunomodulators
GB0125443D0 (en) 2001-10-23 2001-12-12 Novartis Ag Organic Compounds
CA2498191C (fr) 2002-09-18 2012-04-10 Trustees Of The University Of Pennsylvania Methode d'inhibition de la neovascularisation choroidienne
US7920906B2 (en) 2005-03-10 2011-04-05 Dexcom, Inc. System and methods for processing analyte sensor data for sensor calibration
US9247900B2 (en) 2004-07-13 2016-02-02 Dexcom, Inc. Analyte sensor
US20070045902A1 (en) 2004-07-13 2007-03-01 Brauker James H Analyte sensor
US8170803B2 (en) 2004-07-13 2012-05-01 Dexcom, Inc. Transcutaneous analyte sensor
TW200637552A (en) * 2005-01-20 2006-11-01 Array Biopharma Inc Macrocyclic analogs for the treatment of immunoregulatory disorders and respiratory diseases
EP1853259A1 (fr) 2005-02-09 2007-11-14 Macusight, Inc. Formulations pour un traitement oculaire
WO2007092620A2 (fr) 2006-02-09 2007-08-16 Macusight, Inc. Formulations stables et leurs procedes de preparation et d'utilisation
AU2007230964B2 (en) 2006-03-23 2012-07-19 Santen Pharmaceutical Co., Ltd. Formulations and methods for vascular permeability-related diseases or conditions

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5565560A (en) * 1991-05-13 1996-10-15 Merck & Co., Inc. O-Aryl,O-alkyl,O-alkenyl and O-alkynylmacrolides having immunosuppressive activity
US5250678A (en) * 1991-05-13 1993-10-05 Merck & Co., Inc. O-aryl, O-alkyl, O-alkenyl and O-alkynylmacrolides having immunosuppressive activity
US5561228A (en) * 1991-09-05 1996-10-01 Abbott Laboratories Macrocyclic immunomodulators

Also Published As

Publication number Publication date
EP0689545A1 (fr) 1996-01-03
EP0689545A4 (fr) 1996-04-24
WO1994021642A1 (fr) 1994-09-29
JPH08507789A (ja) 1996-08-20

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Legal Events

Date Code Title Description
FZDE Dead