CA2081011A1 - Carboxamides de spiro[benzofurancycloalcane] agissant comme antagonistes 5ht3 - Google Patents

Carboxamides de spiro[benzofurancycloalcane] agissant comme antagonistes 5ht3

Info

Publication number
CA2081011A1
CA2081011A1 CA002081011A CA2081011A CA2081011A1 CA 2081011 A1 CA2081011 A1 CA 2081011A1 CA 002081011 A CA002081011 A CA 002081011A CA 2081011 A CA2081011 A CA 2081011A CA 2081011 A1 CA2081011 A1 CA 2081011A1
Authority
CA
Canada
Prior art keywords
azabicyclo
benzofuran
cyclohexane
oct
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002081011A
Other languages
English (en)
Inventor
Raymond D. Youssefyeh
Henry F. Campbell
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Rhone Poulenc Rorer International Holdings Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2081011A1 publication Critical patent/CA2081011A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Furan Compounds (AREA)
CA002081011A 1990-04-23 1991-04-09 Carboxamides de spiro[benzofurancycloalcane] agissant comme antagonistes 5ht3 Abandoned CA2081011A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51270990A 1990-04-23 1990-04-23
US512,709 1990-04-23

Publications (1)

Publication Number Publication Date
CA2081011A1 true CA2081011A1 (fr) 1991-10-24

Family

ID=24040214

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002081011A Abandoned CA2081011A1 (fr) 1990-04-23 1991-04-09 Carboxamides de spiro[benzofurancycloalcane] agissant comme antagonistes 5ht3

Country Status (4)

Country Link
JP (1) JPH05506222A (fr)
AU (1) AU7657991A (fr)
CA (1) CA2081011A1 (fr)
WO (1) WO1991016888A1 (fr)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3732146A1 (de) * 1987-09-24 1989-04-06 Merck Patent Gmbh Azachromanderivate

Also Published As

Publication number Publication date
WO1991016888A1 (fr) 1991-11-14
JPH05506222A (ja) 1993-09-16
AU7657991A (en) 1991-11-27

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Legal Events

Date Code Title Description
FZDE Dead