BR9814672A - Preparação farmacêutica sob a forma de comprimidos de esferóides e processo de fabricação da mesma - Google Patents
Preparação farmacêutica sob a forma de comprimidos de esferóides e processo de fabricação da mesmaInfo
- Publication number
- BR9814672A BR9814672A BR9814672-6A BR9814672A BR9814672A BR 9814672 A BR9814672 A BR 9814672A BR 9814672 A BR9814672 A BR 9814672A BR 9814672 A BR9814672 A BR 9814672A
- Authority
- BR
- Brazil
- Prior art keywords
- tablets
- spheroids
- manufacturing process
- pharmaceutical preparation
- spheroid
- Prior art date
Links
- 239000000825 pharmaceutical preparation Substances 0.000 title abstract 4
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000004480 active ingredient Substances 0.000 abstract 1
- 230000006835 compression Effects 0.000 abstract 1
- 238000007906 compression Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- PBJUNZJWGZTSKL-MRXNPFEDSA-N tiagabine Chemical compound C1=CSC(C(=CCCN2C[C@@H](CCC2)C(O)=O)C2=C(C=CS2)C)=C1C PBJUNZJWGZTSKL-MRXNPFEDSA-N 0.000 abstract 1
- 229960001918 tiagabine Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Emergency Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
Abstract
"PREPARAçãO FARMACêUTICA SOB A FORMA DE COMPRIMIDOS DE ESFERóIDES E PROCESSO DE FABRICAçãO DA MESMA". A presente invenção refere-se a uma nova forma galênica apresentada na forma de esferóides, contendo um ou mais princípios ativos, com exceção da tiagabina. A presente invenção estende-se também ao processo de preparação destes esferóides e às preparações farmacêuticas multiparticuladas, como comprimidos, contendo estes esferóides. Estas preparações farmacêuticas destinam-se à liberação dos esferóides que elas contêm, e caracterizam-se pela ausência de uma alteração do perfil de liberação do princípio ativo ou dos princípios ativos subseq³entemente a uma eventualmente etapa de compressão.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9714631A FR2771291B1 (fr) | 1997-11-21 | 1997-11-21 | Spheroides, procede de preparation et compositions pharmaceutiques |
PCT/IB1998/001911 WO1999026608A1 (fr) | 1997-11-21 | 1998-11-19 | Spheroides, procede de preparation et compositions pharmaceutiques |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9814672A true BR9814672A (pt) | 2000-10-03 |
Family
ID=9513635
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9814672-6A BR9814672A (pt) | 1997-11-21 | 1998-11-19 | Preparação farmacêutica sob a forma de comprimidos de esferóides e processo de fabricação da mesma |
Country Status (29)
Country | Link |
---|---|
US (1) | US6077544A (pt) |
EP (1) | EP1032374B1 (pt) |
JP (1) | JP2001523706A (pt) |
KR (1) | KR100502938B1 (pt) |
CN (1) | CN1223341C (pt) |
AT (1) | ATE246496T1 (pt) |
AU (1) | AU744580B2 (pt) |
BG (1) | BG65117B1 (pt) |
BR (1) | BR9814672A (pt) |
CA (1) | CA2310147C (pt) |
CZ (1) | CZ299110B6 (pt) |
DE (1) | DE69817010T2 (pt) |
DK (1) | DK1032374T3 (pt) |
EA (1) | EA003324B1 (pt) |
ES (1) | ES2203989T3 (pt) |
FR (1) | FR2771291B1 (pt) |
HR (1) | HRP20000323B1 (pt) |
HU (1) | HU230053B1 (pt) |
IL (2) | IL136215A0 (pt) |
MX (1) | MXPA00004959A (pt) |
NO (1) | NO329728B1 (pt) |
NZ (1) | NZ504662A (pt) |
PL (1) | PL193878B1 (pt) |
PT (1) | PT1032374E (pt) |
SK (1) | SK284493B6 (pt) |
TR (1) | TR200002130T2 (pt) |
WO (1) | WO1999026608A1 (pt) |
YU (1) | YU31000A (pt) |
ZA (1) | ZA9810631B (pt) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2790668B1 (fr) * | 1999-03-12 | 2002-07-26 | D B F | Granules contenant une substance vegetale et leur procede de preparation |
WO2000059467A1 (fr) | 1999-04-06 | 2000-10-12 | Laboratoires Des Produits Ethiques Ethypharm | Suspension pharmaceutique buvable d'ibuprofene |
FR2794646B1 (fr) | 1999-06-09 | 2001-09-21 | Ethypharm Lab Prod Ethiques | Microgranules de sulfate de morphine, procede de preparation et composition les contenant |
AU2002344842A1 (en) | 2001-06-22 | 2003-01-08 | Genencor International, Inc. | Highly impact-resistant granules |
AR034813A1 (es) † | 2001-07-20 | 2004-03-17 | Novartis Ag | Composiciones farmaceuticas y uso de las mismas |
US8101209B2 (en) | 2001-10-09 | 2012-01-24 | Flamel Technologies | Microparticulate oral galenical form for the delayed and controlled release of pharmaceutical active principles |
FR2830447B1 (fr) * | 2001-10-09 | 2004-04-16 | Flamel Tech Sa | Forme galenique orale microparticulaire pour la liberation retardee et controlee de principes actifs pharmaceutiques |
FR2837100B1 (fr) | 2002-03-18 | 2004-07-23 | Flamel Tech Sa | Comprimes a bases de microcapsules a liberation modifiee |
EP1492511B3 (fr) | 2002-04-09 | 2012-05-02 | Flamel Technologies | Formulation pharmaceutique orale sous forme de suspension aqueuse de microcapsules permettant la liberation modifiee de principe(s) actif(s) |
MXPA04009979A (es) * | 2002-04-09 | 2004-12-13 | Flamel Tech Sa | Formulacion farmaceutica oral bajo forma de suspension acuosa de microcapsulas que permiten la liberacion modificada de amoxicilina. |
FR2838647B1 (fr) * | 2002-04-23 | 2006-02-17 | Particules enrobees a liberation prolongee, leur procede de preparation et comprimes les contenant | |
US20040013737A1 (en) * | 2002-07-19 | 2004-01-22 | Philippe Becourt | Taste masked oral composition of telithromycin |
FR2845289B1 (fr) * | 2002-10-04 | 2004-12-03 | Ethypharm Sa | Spheroides, procede de preparation et compositions pharmaceutiques. |
US9107804B2 (en) | 2002-12-10 | 2015-08-18 | Nortec Development Associates, Inc. | Method of preparing biologically active formulations |
NZ523946A (en) * | 2003-01-31 | 2004-06-25 | Carl Ernest Alexander | Portable hygiene compositions comprising a semi-solid gel and active ingredients in bead form for use in personal oral, dental or skin care |
ES2221804B1 (es) * | 2003-06-18 | 2006-04-01 | Lipofoods, S.L. | Microcapsulas para la administracion de ingredientes activos. |
JP5171038B2 (ja) * | 2003-10-10 | 2013-03-27 | エティファルム | イチョウ・エキスを含む放出持続性の微小顆粒およびそのような顆粒の製造方法 |
FR2861990B1 (fr) | 2003-11-10 | 2006-02-10 | Nouveaux Produits Pharma | Comprimes faiblement doses a reseau de polymeres |
EP1737433B1 (en) * | 2004-04-12 | 2007-11-14 | Pfizer Products Incorporated | Taste-masked drugs in rupturing multiparticulates |
US20070224269A1 (en) * | 2004-06-10 | 2007-09-27 | Rubino Orapin P | Controlled Release Pharmaceutical Formulation |
FR2883179B1 (fr) * | 2005-03-18 | 2009-04-17 | Ethypharm Sa | Comprime enrobe |
US20070286900A1 (en) * | 2006-06-09 | 2007-12-13 | Catherine Herry | Low dose tablets of opioid analgesics and preparation process |
US20100233257A1 (en) * | 2006-06-09 | 2010-09-16 | Ethypharm | Low dose sublingual tablets of opioid analgesics and preparation process |
US11116728B2 (en) | 2006-11-30 | 2021-09-14 | Bend Research, Inc. | Multiparticulates of spray-coated drug and polymer on a meltable core |
EP2091519B1 (en) * | 2006-11-30 | 2015-06-24 | Bend Research, Inc | Multiparticulates of spray-coated drug and polymer on a meltable core |
EP2468263A1 (en) | 2010-12-23 | 2012-06-27 | Laboratorios Del. Dr. Esteve, S.A. | Compressed solid dosage forms |
WO2019217686A1 (en) | 2018-05-11 | 2019-11-14 | Stolle Machinery Company, Llc | Infeed assembly full inspection assembly |
EP3790820A4 (en) | 2018-05-11 | 2022-01-26 | Stolle Machinery Company, LLC | QUICK CHANGE TRANSFER ARRANGEMENT |
WO2019217645A1 (en) | 2018-05-11 | 2019-11-14 | Stolle Machinery Company, Llc | Process shaft tooling assembly |
WO2019217667A1 (en) | 2018-05-11 | 2019-11-14 | Stolle Machinery Company, Llc | Quick change tooling assembly |
BR112020022970A2 (pt) | 2018-05-11 | 2021-02-02 | Stolle Machinery Company, Llc | recursos de mudança rápida de conjunto de alimentação |
JP7312196B2 (ja) | 2018-05-11 | 2023-07-20 | ストール マシーナリ カンパニー,エルエルシー | 回転マニホールド |
JP7331017B2 (ja) | 2018-05-11 | 2023-08-22 | ストール マシーナリ カンパニー,エルエルシー | 駆動アセンブリ |
US11420242B2 (en) | 2019-08-16 | 2022-08-23 | Stolle Machinery Company, Llc | Reformer assembly |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4684516A (en) * | 1983-08-01 | 1987-08-04 | Alra Laboratories, Inc. | Sustained release tablets and method of making same |
NZ230763A (en) * | 1988-09-27 | 1991-10-25 | Takeda Chemical Industries Ltd | Production of granules having a core by spraying the cores with a dispersion of hydroxypropylcellulose, optionally incorporating an active ingredient |
EP0418596A3 (en) * | 1989-09-21 | 1991-10-23 | American Cyanamid Company | Controlled release pharmaceutical compositions from spherical granules in tabletted oral dosage unit form |
JP2572673B2 (ja) * | 1990-07-25 | 1997-01-16 | エスエス製薬株式会社 | 徐放性錠剤 |
FR2679451B1 (fr) * | 1991-07-22 | 1994-09-09 | Prographarm Laboratoires | Comprime multiparticulaire a delitement rapide. |
GB9117361D0 (en) * | 1991-08-12 | 1991-09-25 | Euro Celtique Sa | Oral dosage form |
FR2692146B1 (fr) * | 1992-06-16 | 1995-06-02 | Ethypharm Sa | Compositions stables de microgranules d'omeprazole gastro-protégés et leur procédé d'obtention. |
SI9420040A (en) * | 1993-06-14 | 1996-08-31 | Janssen Pharmaceutica Nv | Extended release, film coated tablet of astemizole and pseudoephedrine |
SE9402422D0 (sv) * | 1994-07-08 | 1994-07-08 | Astra Ab | New beads for controlled release and a pharmaceutical preparation containing the same |
SE9600070D0 (sv) * | 1996-01-08 | 1996-01-08 | Astra Ab | New oral pharmaceutical dosage forms |
FR2771292B1 (fr) * | 1997-11-21 | 2000-02-18 | Ethypharm Lab Prod Ethiques | Spheroides contenant de la tiagabine, procede de preparation et compositions pharmaceutiques |
-
1997
- 1997-11-21 FR FR9714631A patent/FR2771291B1/fr not_active Expired - Lifetime
-
1998
- 1998-10-19 TR TR2000/02130T patent/TR200002130T2/xx unknown
- 1998-11-19 BR BR9814672-6A patent/BR9814672A/pt not_active Application Discontinuation
- 1998-11-19 KR KR10-2000-7005544A patent/KR100502938B1/ko not_active IP Right Cessation
- 1998-11-19 EP EP98954683A patent/EP1032374B1/fr not_active Expired - Lifetime
- 1998-11-19 JP JP2000521810A patent/JP2001523706A/ja active Pending
- 1998-11-19 PT PT98954683T patent/PT1032374E/pt unknown
- 1998-11-19 DK DK98954683T patent/DK1032374T3/da active
- 1998-11-19 CZ CZ20001849A patent/CZ299110B6/cs not_active IP Right Cessation
- 1998-11-19 NZ NZ504662A patent/NZ504662A/xx not_active IP Right Cessation
- 1998-11-19 CN CNB988124270A patent/CN1223341C/zh not_active Expired - Lifetime
- 1998-11-19 MX MXPA00004959A patent/MXPA00004959A/es unknown
- 1998-11-19 AT AT98954683T patent/ATE246496T1/de active
- 1998-11-19 ES ES98954683T patent/ES2203989T3/es not_active Expired - Lifetime
- 1998-11-19 AU AU11704/99A patent/AU744580B2/en not_active Expired
- 1998-11-19 PL PL98340659A patent/PL193878B1/pl unknown
- 1998-11-19 YU YU31000A patent/YU31000A/sh unknown
- 1998-11-19 DE DE69817010T patent/DE69817010T2/de not_active Expired - Lifetime
- 1998-11-19 EA EA200000548A patent/EA003324B1/ru not_active IP Right Cessation
- 1998-11-19 CA CA2310147A patent/CA2310147C/fr not_active Expired - Lifetime
- 1998-11-19 SK SK756-2000A patent/SK284493B6/sk unknown
- 1998-11-19 HU HU0100562A patent/HU230053B1/hu unknown
- 1998-11-19 IL IL13621598A patent/IL136215A0/xx active IP Right Grant
- 1998-11-19 WO PCT/IB1998/001911 patent/WO1999026608A1/fr active IP Right Grant
- 1998-11-20 ZA ZA9810631A patent/ZA9810631B/xx unknown
- 1998-11-23 US US09/197,466 patent/US6077544A/en not_active Expired - Lifetime
-
2000
- 2000-05-18 IL IL136215A patent/IL136215A/en not_active IP Right Cessation
- 2000-05-19 HR HR20000323A patent/HRP20000323B1/xx not_active IP Right Cessation
- 2000-05-19 NO NO20002605A patent/NO329728B1/no not_active IP Right Cessation
- 2000-06-06 BG BG104511A patent/BG65117B1/bg unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PRESENTE PEDIDO, UMA VEZ QUE O MESMO NAO ATENDE AO DISPOSTO NOS ARTIGOS 8O E 13 DA LPI. |
|
B12B | Appeal against refusal [chapter 12.2 patent gazette] |