BR9809968A - Aplicação de derivados tiazolidinadiona no tratamento da pcos e diabetes gestacional - Google Patents

Aplicação de derivados tiazolidinadiona no tratamento da pcos e diabetes gestacional

Info

Publication number
BR9809968A
BR9809968A BR9809968-0A BR9809968A BR9809968A BR 9809968 A BR9809968 A BR 9809968A BR 9809968 A BR9809968 A BR 9809968A BR 9809968 A BR9809968 A BR 9809968A
Authority
BR
Brazil
Prior art keywords
pcos
treatment
application
gestational diabetes
insulin
Prior art date
Application number
BR9809968-0A
Other languages
English (en)
Inventor
Tammy Antonucci
Dean Lockwood
Rebecca Norris
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of BR9809968A publication Critical patent/BR9809968A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Patente de Invenção: <B>"APLICAçãO DE DERIVADOS TIAZOLIDINADIONA NO TRATAMENTO DA PCOS E DIABETES GESTACIONAL"<D>. São usados novos métodos de utilização de derivados tiazolidinona e agentes anti-hiperglicêmicos relacionados pata tratar populações com risco de desenvolver diabetes mellitus não-dependente de insulina (NIDDM) e complicações originadas destas. Em uma modalidade, os compostos da invenção são usados para tratar a PCOS de modo a impedir ou retardar o início do diabetes mellitus não-dependente de insulina. Em outra modalidade, os compostos da invenção são usados para tratar diabetes gestacional de modo a impedir ou retardar o início do diabetes mellitus não-dependente de insulina.
BR9809968-0A 1997-06-04 1998-05-21 Aplicação de derivados tiazolidinadiona no tratamento da pcos e diabetes gestacional BR9809968A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/868,608 US6046222A (en) 1993-09-15 1997-06-04 Use of thiazolidinedione derivatives in the treatment of polycystic ovary syndrome, gestational diabetes and disease states at risk for progressing to noninsulin-dependent diabetes mellitus
PCT/US1998/010472 WO1998055121A1 (en) 1997-06-04 1998-05-21 Use of thiazolidinedione derivatives in the treatment of polycystic ovary syndrome and gestational diabetes

Publications (1)

Publication Number Publication Date
BR9809968A true BR9809968A (pt) 2000-08-01

Family

ID=25352002

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9809968-0A BR9809968A (pt) 1997-06-04 1998-05-21 Aplicação de derivados tiazolidinadiona no tratamento da pcos e diabetes gestacional

Country Status (15)

Country Link
US (3) US6046222A (pt)
EP (1) EP0984780B1 (pt)
JP (1) JP2002511859A (pt)
KR (1) KR20010013337A (pt)
AT (1) ATE303147T1 (pt)
BR (1) BR9809968A (pt)
CA (1) CA2283319A1 (pt)
DE (1) DE69831406D1 (pt)
HU (1) HUP0003876A3 (pt)
IL (1) IL131801A0 (pt)
IS (1) IS5194A (pt)
NO (1) NO995932L (pt)
PL (1) PL348773A1 (pt)
WO (1) WO1998055121A1 (pt)
ZA (1) ZA984798B (pt)

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Also Published As

Publication number Publication date
US6130216A (en) 2000-10-10
NO995932D0 (no) 1999-12-03
IL131801A0 (en) 2001-03-19
NO995932L (no) 1999-12-03
PL348773A1 (en) 2002-06-17
WO1998055121A1 (en) 1998-12-10
US5972944A (en) 1999-10-26
CA2283319A1 (en) 1998-12-10
ATE303147T1 (de) 2005-09-15
HUP0003876A2 (hu) 2002-01-28
KR20010013337A (ko) 2001-02-26
EP0984780B1 (en) 2005-08-31
JP2002511859A (ja) 2002-04-16
HUP0003876A3 (en) 2002-04-29
DE69831406D1 (de) 2005-10-06
US6046222A (en) 2000-04-04
IS5194A (is) 1999-09-24
EP0984780A1 (en) 2000-03-15
ZA984798B (en) 1998-12-29

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 9A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1912 DE 28/08/2007.