BR112018005811A2 - composição farmacêutica para administração na mucosa nasal - Google Patents
composição farmacêutica para administração na mucosa nasalInfo
- Publication number
- BR112018005811A2 BR112018005811A2 BR112018005811-4A BR112018005811A BR112018005811A2 BR 112018005811 A2 BR112018005811 A2 BR 112018005811A2 BR 112018005811 A BR112018005811 A BR 112018005811A BR 112018005811 A2 BR112018005811 A2 BR 112018005811A2
- Authority
- BR
- Brazil
- Prior art keywords
- oxytocin
- nasal mucosa
- pharmaceutical composition
- acid addition
- addition salt
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/74—Synthetic polymeric materials
- A61K31/765—Polymers containing oxygen
- A61K31/78—Polymers containing oxygen of acrylic acid or derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/095—Oxytocins; Vasopressins; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0043—Nose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/10—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Immunology (AREA)
- Gastroenterology & Hepatology (AREA)
- Inorganic Chemistry (AREA)
- Otolaryngology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Peptides Or Proteins (AREA)
Abstract
a presente invenção aborda o problema de prover gotas nasais que podem alcançar alta absorção de oxitocina, que é um hormônio peptídeo, um sal de adição de ácido de oxitocina ou um derivado de oxitocina ou o sal de adição de ácido através de uma mucosa nasal e que tem menos problemas de segurança. a presente invenção é uma composição farmacêutica destinada para ser administrada a uma mucosa nasal, distinguida por compreender oxitocina ou o sal de adição de ácido e um polímero de carboxivinila e ter uma razão de pressão osmótica menor que 1.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2015214481 | 2015-10-30 | ||
JP2015-214481 | 2015-10-30 | ||
PCT/JP2016/082897 WO2017073798A1 (ja) | 2015-10-30 | 2016-10-28 | 鼻粘膜投与用医薬組成物 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112018005811A2 true BR112018005811A2 (pt) | 2018-10-16 |
Family
ID=58630599
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112018005811-4A BR112018005811A2 (pt) | 2015-10-30 | 2016-10-28 | composição farmacêutica para administração na mucosa nasal |
Country Status (17)
Country | Link |
---|---|
US (1) | US10849978B2 (pt) |
EP (1) | EP3369429B1 (pt) |
JP (1) | JP6629877B2 (pt) |
KR (1) | KR20180066071A (pt) |
CN (1) | CN108135959B (pt) |
AU (1) | AU2016346823A1 (pt) |
BR (1) | BR112018005811A2 (pt) |
CA (1) | CA2995839A1 (pt) |
DK (1) | DK3369429T3 (pt) |
ES (1) | ES2774128T3 (pt) |
HK (1) | HK1249856A1 (pt) |
MX (1) | MX2018005363A (pt) |
PL (1) | PL3369429T3 (pt) |
PT (1) | PT3369429T (pt) |
RU (1) | RU2725664C2 (pt) |
TW (1) | TWI745313B (pt) |
WO (1) | WO2017073798A1 (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2019131723A1 (ja) | 2017-12-27 | 2019-07-04 | 武田薬品工業株式会社 | 薬物の投与方法 |
WO2020061414A1 (en) * | 2018-09-20 | 2020-03-26 | Levo Therapeutics, Inc. | Stable intranasal formulations of carbetocin |
FR3088193B1 (fr) | 2018-11-13 | 2021-01-22 | Andrea Fox | Composition aqueuse, son procede de fabrication, et dispositif d’administration nasal |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5142420A (en) | 1974-10-08 | 1976-04-10 | Matsushita Electric Ind Co Ltd | Tajushingobunrihoshiki |
JPS60123426A (ja) | 1983-12-07 | 1985-07-02 | Eisai Co Ltd | 経鼻投与用セクレチン製剤 |
JP2734554B2 (ja) | 1988-09-12 | 1998-03-30 | 藤沢薬品工業株式会社 | インスリン様成長因子iの点鼻用液剤 |
US5158761A (en) * | 1989-04-05 | 1992-10-27 | Toko Yakuhin Kogyo Kabushiki Kaisha | Spray gel base and spray gel preparation using thereof |
JP3705620B2 (ja) | 1994-12-28 | 2005-10-12 | 帝国臓器製薬株式会社 | 経粘膜投与用製剤 |
US5521283A (en) * | 1995-01-31 | 1996-05-28 | Eli Lilly And Company | Anti-obesity proteins |
TWI243687B (en) | 1998-04-21 | 2005-11-21 | Teijin Ltd | Pharmaceutical composition for application to mucosa |
US8268791B2 (en) | 2004-08-25 | 2012-09-18 | Aegis Therapeutics, Llc. | Alkylglycoside compositions for drug administration |
US9023793B2 (en) * | 2006-09-29 | 2015-05-05 | Retrophin, Inc. | Intranasal carbetocin formulations and methods for the treatment of autism |
CA2689476C (en) | 2007-06-07 | 2014-08-05 | Nastech Pharmaceutical Company Inc. | Intranasal carbetocin formulations and methods for the treatment of autism |
EP2543387B1 (en) * | 2010-03-02 | 2016-10-26 | The University of Tokushima | Mucosal vaccine |
SE536091C2 (sv) | 2011-04-14 | 2013-04-30 | Pep Tonic Medical Ab | Farmaceutisk komposition innehållande oxytocin eller fragment eller varianter därav och åtminstone en icke-jonisk cellulosaeter |
JP6304744B2 (ja) * | 2013-12-20 | 2018-04-04 | 国立大学法人福井大学 | 愛着障害治療剤 |
-
2016
- 2016-10-28 CN CN201680063129.4A patent/CN108135959B/zh active Active
- 2016-10-28 EP EP16860025.2A patent/EP3369429B1/en active Active
- 2016-10-28 JP JP2017547363A patent/JP6629877B2/ja active Active
- 2016-10-28 WO PCT/JP2016/082897 patent/WO2017073798A1/ja active Application Filing
- 2016-10-28 MX MX2018005363A patent/MX2018005363A/es unknown
- 2016-10-28 PL PL16860025T patent/PL3369429T3/pl unknown
- 2016-10-28 CA CA2995839A patent/CA2995839A1/en not_active Abandoned
- 2016-10-28 ES ES16860025T patent/ES2774128T3/es active Active
- 2016-10-28 AU AU2016346823A patent/AU2016346823A1/en not_active Abandoned
- 2016-10-28 DK DK16860025.2T patent/DK3369429T3/da active
- 2016-10-28 BR BR112018005811-4A patent/BR112018005811A2/pt active Search and Examination
- 2016-10-28 RU RU2018118986A patent/RU2725664C2/ru active
- 2016-10-28 TW TW105135103A patent/TWI745313B/zh active
- 2016-10-28 KR KR1020187009565A patent/KR20180066071A/ko not_active Application Discontinuation
- 2016-10-28 US US15/750,378 patent/US10849978B2/en active Active
- 2016-10-28 PT PT168600252T patent/PT3369429T/pt unknown
-
2018
- 2018-07-19 HK HK18109333.7A patent/HK1249856A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
JPWO2017073798A1 (ja) | 2018-05-31 |
KR20180066071A (ko) | 2018-06-18 |
CN108135959B (zh) | 2021-12-31 |
CA2995839A1 (en) | 2017-05-04 |
RU2018118986A3 (pt) | 2020-01-15 |
PT3369429T (pt) | 2020-02-20 |
US10849978B2 (en) | 2020-12-01 |
TWI745313B (zh) | 2021-11-11 |
HK1249856A1 (zh) | 2018-11-16 |
CN108135959A (zh) | 2018-06-08 |
TW201729830A (zh) | 2017-09-01 |
PL3369429T3 (pl) | 2020-06-15 |
DK3369429T3 (da) | 2020-02-10 |
MX2018005363A (es) | 2018-09-05 |
EP3369429A1 (en) | 2018-09-05 |
AU2016346823A1 (en) | 2018-03-08 |
RU2018118986A (ru) | 2019-12-02 |
WO2017073798A1 (ja) | 2017-05-04 |
JP6629877B2 (ja) | 2020-01-15 |
RU2725664C2 (ru) | 2020-07-03 |
EP3369429B1 (en) | 2019-12-11 |
ES2774128T3 (es) | 2020-07-16 |
EP3369429A4 (en) | 2018-10-31 |
US20180228902A1 (en) | 2018-08-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
|
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
B06U | Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette] |