BR112012026016A2 - combinação de um inibidor macrocíclico de hcv, um não-nucleosídeo e um nucleosídeo - Google Patents
combinação de um inibidor macrocíclico de hcv, um não-nucleosídeo e um nucleosídeoInfo
- Publication number
- BR112012026016A2 BR112012026016A2 BR112012026016A BR112012026016A BR112012026016A2 BR 112012026016 A2 BR112012026016 A2 BR 112012026016A2 BR 112012026016 A BR112012026016 A BR 112012026016A BR 112012026016 A BR112012026016 A BR 112012026016A BR 112012026016 A2 BR112012026016 A2 BR 112012026016A2
- Authority
- BR
- Brazil
- Prior art keywords
- nucleoside
- combination
- macrocyclic
- hcv inhibitor
- inhibitor
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
combinação de um inibidor macrocíclico de hcv, um não-nucleosídeo e um nucleosídeo. a presente invenção refere-se a uma combinação de um inibidor de hcv protease macrocíciclo, um inibidor de hcv polimerase de não-nucleosídeo macrocíclico e um inibidor de hcv polimerase de nucleosídeo.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10159825 | 2010-04-13 | ||
PCT/EP2011/055836 WO2011128378A1 (en) | 2010-04-13 | 2011-04-13 | Combination of a macrocyclic inhibitor of hcv, a non-nucleoside and a nucleoside |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112012026016A2 true BR112012026016A2 (pt) | 2016-06-07 |
Family
ID=42237337
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112012026016A BR112012026016A2 (pt) | 2010-04-13 | 2011-04-13 | combinação de um inibidor macrocíclico de hcv, um não-nucleosídeo e um nucleosídeo |
Country Status (14)
Country | Link |
---|---|
US (1) | US20130028865A1 (pt) |
EP (1) | EP2558091A1 (pt) |
JP (1) | JP5989635B2 (pt) |
KR (1) | KR20130057990A (pt) |
CN (1) | CN102844028B (pt) |
AU (1) | AU2011239974B2 (pt) |
BR (1) | BR112012026016A2 (pt) |
CA (1) | CA2796243A1 (pt) |
EA (1) | EA201291042A1 (pt) |
HK (1) | HK1180222A1 (pt) |
MX (1) | MX2012011963A (pt) |
NZ (1) | NZ602552A (pt) |
SG (2) | SG10201506652QA (pt) |
WO (1) | WO2011128378A1 (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20070211A1 (es) | 2005-07-29 | 2007-05-12 | Medivir Ab | Compuestos macrociclicos como inhibidores del virus de hepatitis c |
TWI454476B (zh) | 2008-07-08 | 2014-10-01 | Tibotec Pharm Ltd | 用作c型肝炎病毒抑制劑之巨環吲哚衍生物 |
CN104780921A (zh) * | 2012-08-31 | 2015-07-15 | 杨森制药公司 | Hcv的大环蛋白酶抑制剂、非核苷hcv抑制剂和利托那韦的组合 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2552319C (en) | 2004-01-30 | 2012-08-21 | Medivir Ab | Hcv ns-3 serine protease inhibitors |
PE20070211A1 (es) * | 2005-07-29 | 2007-05-12 | Medivir Ab | Compuestos macrociclicos como inhibidores del virus de hepatitis c |
KR20090078347A (ko) | 2006-10-10 | 2009-07-17 | 메디비르 아베 | Hcv 뉴클레오시드 억제제 |
TWI454476B (zh) * | 2008-07-08 | 2014-10-01 | Tibotec Pharm Ltd | 用作c型肝炎病毒抑制劑之巨環吲哚衍生物 |
TW201023858A (en) * | 2008-09-18 | 2010-07-01 | Ortho Mcneil Janssen Pharm | Synergistic combinations of a macrocyclic inhibitor of HCV and a nucleoside |
AR077125A1 (es) * | 2009-06-23 | 2011-08-03 | Gilead Sciences Inc | Combinaciones farmaceuticas utiles para tratar el vhc |
-
2011
- 2011-04-13 KR KR1020127028453A patent/KR20130057990A/ko not_active Application Discontinuation
- 2011-04-13 EA EA201291042A patent/EA201291042A1/ru unknown
- 2011-04-13 CA CA2796243A patent/CA2796243A1/en not_active Abandoned
- 2011-04-13 WO PCT/EP2011/055836 patent/WO2011128378A1/en active Application Filing
- 2011-04-13 NZ NZ602552A patent/NZ602552A/en not_active IP Right Cessation
- 2011-04-13 EP EP11715219A patent/EP2558091A1/en not_active Ceased
- 2011-04-13 CN CN201180018701.2A patent/CN102844028B/zh not_active Expired - Fee Related
- 2011-04-13 SG SG10201506652QA patent/SG10201506652QA/en unknown
- 2011-04-13 JP JP2013504263A patent/JP5989635B2/ja not_active Expired - Fee Related
- 2011-04-13 BR BR112012026016A patent/BR112012026016A2/pt not_active Application Discontinuation
- 2011-04-13 MX MX2012011963A patent/MX2012011963A/es unknown
- 2011-04-13 US US13/640,657 patent/US20130028865A1/en not_active Abandoned
- 2011-04-13 SG SG2012075057A patent/SG184524A1/en unknown
- 2011-04-13 AU AU2011239974A patent/AU2011239974B2/en not_active Ceased
-
2013
- 2013-06-26 HK HK13107522.7A patent/HK1180222A1/zh not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
MX2012011963A (es) | 2012-12-17 |
JP2013523866A (ja) | 2013-06-17 |
NZ602552A (en) | 2014-09-26 |
CA2796243A1 (en) | 2011-10-20 |
US20130028865A1 (en) | 2013-01-31 |
EP2558091A1 (en) | 2013-02-20 |
KR20130057990A (ko) | 2013-06-03 |
SG10201506652QA (en) | 2015-10-29 |
AU2011239974A1 (en) | 2012-10-25 |
AU2011239974B2 (en) | 2015-12-03 |
JP5989635B2 (ja) | 2016-09-07 |
EA201291042A1 (ru) | 2013-03-29 |
SG184524A1 (en) | 2012-11-29 |
WO2011128378A1 (en) | 2011-10-20 |
CN102844028B (zh) | 2016-04-06 |
HK1180222A1 (zh) | 2013-10-18 |
CN102844028A (zh) | 2012-12-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B65X | Notification of requirement for priority examination of patent application | ||
B65Y | Grant of priority examination of the patent application (request complies with dec. 132/06 of 20061117) | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B11E | Dismissal acc. art. 34 of ipl - requirements for examination incomplete | ||
B11T | Dismissal of application maintained [chapter 11.20 patent gazette] |