BR0317728A - Fungicidas com base em heterociclos contendo nitrogênio - Google Patents
Fungicidas com base em heterociclos contendo nitrogênioInfo
- Publication number
- BR0317728A BR0317728A BR0317728-9A BR0317728A BR0317728A BR 0317728 A BR0317728 A BR 0317728A BR 0317728 A BR0317728 A BR 0317728A BR 0317728 A BR0317728 A BR 0317728A
- Authority
- BR
- Brazil
- Prior art keywords
- alkyl
- alkoxy
- halo
- alkylthio
- heteroaryl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
"FUNGICIDAS COM BASE EM HETEROCICLOS CONTENDO NITROGêNIO". A presente invenção refere-se a compostos fungicidas tendo a fórmula geral (1): fórmula (1) em que W, Z e um dentre X e Y são N e qualquer um dentre X e Y é CR¬8¬; R¬8¬ é H, halo, C~ 1-4~alquila, C~ 1-4~alcóxi, C~ 1-4~alquiltio ou halo(C~ 1-4~)alquila; R e R¬ 2~ são independentemente H, halo, C~1-8~alquila, C~ 1-8~,alcóxi, C~ 1-8~alquiltio, C~ 2-8~,alquenila, C~ 2-8~alquinila, ciano ou NR¬ 3¬R¬ 4¬, contanto que pelo menos um dentre R e R¬ 2¬ seja NR¬ 3¬R¬ 4¬; R¬ 1¬ é halo, C~ 1-8~alquila, C~ 2-8~alquenila, C~ 2-8~alquinila, C~ 3-8~Cicloalquila, C~ 3-8~cicloalquil(C~ 1-6~)alquila, C~ 1-8~alcóxi, C~ 1-8~alquiltio, arila, arilóxi, ariltio, heteroarila, heteroarilóxi, heteroariltio, aril(C~ 1-4~)alquila, aril(C~ 1-4~)aicóxi, heteroaril(C~ 1-4~) alquila, heteroaril(C~ 1-4~)aicóxi, aril(C~ 1-4~)alquiltio, heteroaril(C~ 1-4~)alquiltio, morfolino, piperidino ou pirrolidino; R¬ 3¬ e R¬ 4¬ São independentemente H, C~ 1-8~ alquila, C~ 2-8~alquenila, C~ 2-8~ alquinila, arila, aril(C~ 1-8~)alquila, C~ 3-8~cicloalquila, C~ 3-8~ cicloalquil(C~ 1-6~)alquila, heteroarila, heteroaril(C~ 1-8~)alquila, NR¬ 5¬R¬ 6¬, contanto que igualmente R¬ 3¬ e R¬ 4¬ não sejam H ou NR¬ 6¬ R¬ 6¬ ou R¬ 3¬ e R¬ 4¬ juntos formam uma cadeia de C~ 3-7~alquileno ou C~ 3-7~alquenileno opcionalmente substituída com um ou mais grupos de C~ 1-4~alquila ou C~ 1-4~aLcóxi ou juntamente com o átomo de nitrogênio ao qual eles são ligados, R¬ 3¬e R¬ 4¬formam um anel de morfolina, tiomorfolina, S-óxido de tiomorfolina ou S-dióxido de tiomorfolina ou um anel de N-(C~ 1-4~) alquila de piperazina ou piperazina (especialmente N-metila); e R¬ 5¬ e R¬ 6¬ São independentemente H, C~ 1-8~alquila, C~ 2-8~alquenila, C~ 2-8~alquinila, arila, aril(C~ 1-8~) alquila, C~ 3-8~CiCloalquila, C~ 3~,cicloalquil(C~ 1-5~)alquila, heteroarila ou heteroaril(C~ 1-8~)alquila; qualquer das porções ou grupos de alquila, alquenila, alquinila ou cicloalquila anteriores (não ser para R¬ 8¬) sendo opcionalmente substituídos com halogênio, ciano, C~ 1-6~alcóxi, C~ 1-6~alquilcarbonila, C~ 1-6~alcoxicarbonila, C~ 1-6~ haloalcóxi, C~ 1-6~alquiltio, tri(C~ 1-4~)alquilsilila, C~ 1-6~alquilamino ou C~ 1-6~dialquilamino, quaisquer dos anéis de morfolina, tiomorfolina, piperidina, piperazina e pirrolidina anteriores sendo opcionalmente substituídos com C~ 1-4~alquila (especialmente metila) e quaisquer das porções ou grupos de arila ou heteroarila anteriores sendo opcionalmente substituídos com um ou mais substituintes selecionados de halo, hidróxi, mercapto, C~ 1-6~alquila, C~ 2-6~alquenila, C~ 2-6~alquinila, C~ 1-6~alcóxi, C~ 2-6~alquenilóxi, C~ 2-6~alquinilóxi, halo(C~ 1-6~)alquila, halo(C~ 1-6~)alcóxi, C~ 1-6~alquiltio, halo(C~ 1-6~)alquiltio, hidróxi(C~ 1-6~)alquila, C~ 1-4~alcóxi(C~ 1-6~)alquila, C~ 3-6~ Cicloalquila, C~ 3-6~cicloalquil(C~ 1-4~)alquila, fenóxi, benzilóxi, benzoilóxi, ciano, isociano, tiocianato, isotiocianato, nitro, -NR<39><39><39>R<39><39><39><39>, -NHCOR<39><39><39>, -NHCONR<39><39><39>R<39><39><39><39>, -CONR<39><39><39>R<39><39><39>, -SO~ 2~R<39><39><39>, -OSO~ 2~R<39><39><39>, -COR<39><39><39>, -CR<39><39><39>=NR<39><39><39><39> ou -N=CR<39><39><39>R<39><39><39><39>, em que R<39><39><39> e R<39><39><39><39> são independentemente hidrogênio, C~ 1-4~ alquila, halo(C~ 1-4~)alquila, C~ 1-4~ alcóxi, halo(C~ 1-4~)alcóxi, C~ 1-4~ alquiltio, C~ 3-6~Cicloalquila, C~ 3-6~Cicloalquil(C~ 1-4~)alquila, fenila ou benzila, os grupos de fenila e benzila sendo opcionalmente substituídos com halogênio, C~ 1-4~alquila ou C~ 1-4~alcóxi.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0230021.8A GB0230021D0 (en) | 2002-12-23 | 2002-12-23 | Fungicides |
| PCT/GB2003/005261 WO2004056829A1 (en) | 2002-12-23 | 2003-12-03 | Fungicides based on nitrogen-containing heterocycles |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0317728A true BR0317728A (pt) | 2005-11-22 |
Family
ID=9950324
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0317728-9A BR0317728A (pt) | 2002-12-23 | 2003-12-03 | Fungicidas com base em heterociclos contendo nitrogênio |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US20060100203A1 (pt) |
| EP (1) | EP1575956B1 (pt) |
| JP (1) | JP2006516130A (pt) |
| KR (1) | KR20050088210A (pt) |
| CN (1) | CN100338065C (pt) |
| AR (1) | AR042662A1 (pt) |
| AT (1) | ATE358131T1 (pt) |
| AU (1) | AU2003288412A1 (pt) |
| BR (1) | BR0317728A (pt) |
| CA (1) | CA2510376A1 (pt) |
| CR (1) | CR7861A (pt) |
| DE (1) | DE60312889T2 (pt) |
| DK (1) | DK1575956T3 (pt) |
| EC (1) | ECSP055862A (pt) |
| EG (1) | EG23771A (pt) |
| ES (1) | ES2283845T3 (pt) |
| GB (1) | GB0230021D0 (pt) |
| GT (1) | GT200300301A (pt) |
| IL (1) | IL169187A0 (pt) |
| MX (1) | MXPA05006669A (pt) |
| PT (1) | PT1575956E (pt) |
| RU (1) | RU2005123332A (pt) |
| TW (1) | TW200425834A (pt) |
| WO (1) | WO2004056829A1 (pt) |
| ZA (1) | ZA200504297B (pt) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0230020D0 (en) | 2002-12-23 | 2003-01-29 | Syngenta Ltd | Fungicides |
| GB0230018D0 (en) | 2002-12-23 | 2003-01-29 | Syngenta Ltd | Fungicides |
| US8293751B2 (en) | 2003-01-14 | 2012-10-23 | Arena Pharmaceuticals, Inc. | 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia |
| GB0413955D0 (en) * | 2004-06-22 | 2004-07-28 | Syngenta Participations Ag | Chemical compounds |
| GB0614471D0 (en) | 2006-07-20 | 2006-08-30 | Syngenta Ltd | Herbicidal Compounds |
| JP5142492B2 (ja) * | 2006-08-01 | 2013-02-13 | 東ソー株式会社 | （１−メチル−２，２，２−トリフルオロ）エチルアミン類およびその製造方法 |
| US20100093738A1 (en) * | 2006-10-06 | 2010-04-15 | Basf Se | Fungicidal Compounds and Fungicidal Compositions |
| GB0800855D0 (en) * | 2008-01-17 | 2008-02-27 | Syngenta Ltd | Herbicidal compounds |
| EP2619198A1 (en) | 2010-09-22 | 2013-07-31 | Arena Pharmaceuticals, Inc. | Modulators of the gpr119 receptor and the treatment of disorders related thereto |
| AU2016205361C1 (en) | 2015-01-06 | 2021-04-08 | Arena Pharmaceuticals, Inc. | Methods of treating conditions related to the S1P1 receptor |
| DK3310760T3 (da) | 2015-06-22 | 2022-10-24 | Arena Pharm Inc | Krystallinsk L-argininsalt af (R)-2-(7-(4-cyclopentyl-3-(trifluormethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3- yl)eddikesyre til anvendelse ved S1P1-receptor-associerede lidelser |
| CA3029104A1 (en) * | 2016-06-24 | 2017-12-28 | Bayer Cropscience Aktiengesellschaft | 3-amino-1,2,4-triazine derivatives and their use for controlling undesired plant growth |
| CA3053418A1 (en) | 2017-02-16 | 2018-08-23 | Arena Pharmaceuticals, Inc. | Compounds and methods for treatment of primary biliary cholangitis |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3984412A (en) * | 1974-07-25 | 1976-10-05 | E. R. Squibb & Sons, Inc. | Amino derivatives of pyrido[2,3-b]pyrazine carboxylic acids and esters |
| DE4131029A1 (de) * | 1991-09-18 | 1993-07-29 | Basf Ag | Substituierte pyrido (2,3-d) pyrimidine als antidots |
| DE4308014A1 (de) * | 1993-03-13 | 1994-09-15 | Hoechst Schering Agrevo Gmbh | Kondensierte Stickstoffheterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel und Fungizide |
| DE10121101A1 (de) * | 2001-04-27 | 2002-10-31 | Bayer Ag | Triazolopyrimidine |
| DE10121162A1 (de) * | 2001-04-30 | 2002-10-31 | Bayer Ag | Triazolopyrimidine |
-
2002
- 2002-12-23 GB GBGB0230021.8A patent/GB0230021D0/en not_active Ceased
-
2003
- 2003-12-03 BR BR0317728-9A patent/BR0317728A/pt not_active IP Right Cessation
- 2003-12-03 AU AU2003288412A patent/AU2003288412A1/en not_active Abandoned
- 2003-12-03 AT AT03780333T patent/ATE358131T1/de not_active IP Right Cessation
- 2003-12-03 RU RU2005123332/04A patent/RU2005123332A/ru not_active Application Discontinuation
- 2003-12-03 ES ES03780333T patent/ES2283845T3/es not_active Expired - Lifetime
- 2003-12-03 PT PT03780333T patent/PT1575956E/pt unknown
- 2003-12-03 WO PCT/GB2003/005261 patent/WO2004056829A1/en active IP Right Grant
- 2003-12-03 DE DE60312889T patent/DE60312889T2/de not_active Expired - Fee Related
- 2003-12-03 KR KR1020057011794A patent/KR20050088210A/ko not_active Application Discontinuation
- 2003-12-03 CA CA002510376A patent/CA2510376A1/en not_active Abandoned
- 2003-12-03 EP EP03780333A patent/EP1575956B1/en not_active Expired - Lifetime
- 2003-12-03 MX MXPA05006669A patent/MXPA05006669A/es active IP Right Grant
- 2003-12-03 US US10/540,039 patent/US20060100203A1/en not_active Abandoned
- 2003-12-03 CN CNB200380107318XA patent/CN100338065C/zh not_active Expired - Fee Related
- 2003-12-03 DK DK03780333T patent/DK1575956T3/da active
- 2003-12-03 JP JP2004561604A patent/JP2006516130A/ja active Pending
- 2003-12-22 AR ARP030104803A patent/AR042662A1/es unknown
- 2003-12-23 TW TW092136602A patent/TW200425834A/zh unknown
- 2003-12-23 GT GT200300301A patent/GT200300301A/es unknown
-
2005
- 2005-05-26 ZA ZA200504297A patent/ZA200504297B/en unknown
- 2005-06-07 CR CR7861A patent/CR7861A/es not_active Application Discontinuation
- 2005-06-15 IL IL169187A patent/IL169187A0/en unknown
- 2005-06-17 EC EC2005005862A patent/ECSP055862A/es unknown
- 2005-06-21 EG EGNA2005000341 patent/EG23771A/xx active
Also Published As
| Publication number | Publication date |
|---|---|
| DK1575956T3 (da) | 2007-08-06 |
| ZA200504297B (en) | 2005-11-28 |
| EG23771A (en) | 2007-08-08 |
| WO2004056829A1 (en) | 2004-07-08 |
| ES2283845T3 (es) | 2007-11-01 |
| TW200425834A (en) | 2004-12-01 |
| ATE358131T1 (de) | 2007-04-15 |
| KR20050088210A (ko) | 2005-09-02 |
| EP1575956B1 (en) | 2007-03-28 |
| MXPA05006669A (es) | 2005-08-16 |
| CN1729194A (zh) | 2006-02-01 |
| CR7861A (es) | 2005-12-02 |
| ECSP055862A (es) | 2005-09-20 |
| AU2003288412A1 (en) | 2004-07-14 |
| DE60312889T2 (de) | 2008-01-17 |
| GB0230021D0 (en) | 2003-01-29 |
| RU2005123332A (ru) | 2006-05-10 |
| DE60312889D1 (de) | 2007-05-10 |
| JP2006516130A (ja) | 2006-06-22 |
| CN100338065C (zh) | 2007-09-19 |
| GT200300301A (es) | 2006-10-03 |
| IL169187A0 (en) | 2008-02-09 |
| EP1575956A1 (en) | 2005-09-21 |
| AR042662A1 (es) | 2005-06-29 |
| US20060100203A1 (en) | 2006-05-11 |
| CA2510376A1 (en) | 2004-07-08 |
| PT1575956E (pt) | 2007-07-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A E 8A ANUIDADE(S). |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2144 DE 07/02/2012. |