BR0211169A - Process for preparing amidine derivatives - Google Patents

Process for preparing amidine derivatives

Info

Publication number
BR0211169A
BR0211169A BR0211169A BR0211169A BR0211169A BR 0211169 A BR0211169 A BR 0211169A BR 0211169 A BR0211169 A BR 0211169A BR 0211169 A BR0211169 A BR 0211169A BR 0211169 A BR0211169 A BR 0211169A
Authority
BR
Brazil
Prior art keywords
process
amidine derivatives
carried out
preparing amidine
preparing
Prior art date
Application number
BR0211169A
Other languages
Portuguese (pt)
Inventor
Toshiaki Masui
Kyozo Kawata
Takayuki Kasai
Makoto Kakinuma
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to JP2001215361 priority Critical
Application filed by Shionogi & Co filed Critical Shionogi & Co
Priority to PCT/JP2002/007142 priority patent/WO2003008421A1/en
Publication of BR0211169A publication Critical patent/BR0211169A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14Ortho-condensed systems

Abstract

"PROCESSO PARA PREPARAçãO DE DERIVADOS DE AMIDINA". "PROCESS FOR amidine DERIVATIVES PREPARATION". A presente invenção refere-se a um processo para produção de derivados de amidina representado pelo seguinte esquema de reação, caracterizado pelo fato de que as reações das etapas 1 e 3 são realizadas em acetonitrila e a reação da etapa 2 é realizada em acetona The present invention relates to a process for producing amidine derivative represented by the following reaction scheme, characterized by the fact that the reactions of steps 1 and 3 are carried out in acetonitrile and the reaction of the step 2 is carried out in acetone
BR0211169A 2001-07-16 2002-07-15 Process for preparing amidine derivatives BR0211169A (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2001215361 2001-07-16
PCT/JP2002/007142 WO2003008421A1 (en) 2001-07-16 2002-07-15 Process for preparation of amidine derivatives

Publications (1)

Publication Number Publication Date
BR0211169A true BR0211169A (en) 2004-08-10

Family

ID=19050015

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0211169A BR0211169A (en) 2001-07-16 2002-07-15 Process for preparing amidine derivatives

Country Status (9)

Country Link
US (1) US6987187B2 (en)
EP (1) EP1408041A4 (en)
JP (1) JPWO2003008421A1 (en)
KR (1) KR20040027878A (en)
CN (1) CN1250550C (en)
BR (1) BR0211169A (en)
CA (1) CA2453664A1 (en)
MX (1) MXPA04000449A (en)
WO (1) WO2003008421A1 (en)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10162114A1 (en) * 2001-12-12 2003-06-26 Schering Ag New N-phenyl (hetero)aryl-carboximidamides are potent nitrogen monoxide synthase inhibitors, useful e.g. for treating neurodegenerative, cardiovascular, autoimmune and/or inflammatory diseases
AU2004266658A1 (en) 2003-08-12 2005-03-03 3M Innovative Properties Company Hydroxylamine substituted imidazo-containing compounds
KR101106812B1 (en) 2003-08-27 2012-01-19 쓰리엠 이노베이티브 프로퍼티즈 컴파니 Aryloxy and Arylalkyleneoxy Substituted Imidazoquinolines
WO2005023190A2 (en) 2003-09-05 2005-03-17 3M Innovative Properties Company Treatment for cd5+ b cell lymphoma
BRPI0414856A (en) 2003-10-03 2006-11-21 3M Innovative Properties Co alkoxy-substituted imidazoquinoline
US7544697B2 (en) 2003-10-03 2009-06-09 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and analogs thereof
WO2005048933A2 (en) 2003-11-14 2005-06-02 3M Innovative Properties Company Oxime substituted imidazo ring compounds
US8598192B2 (en) 2003-11-14 2013-12-03 3M Innovative Properties Company Hydroxylamine substituted imidazoquinolines
CA2547020C (en) 2003-11-25 2014-03-25 3M Innovative Properties Company 1h-imidazo[4,5-c]pyridine-4-amine derivatives as immune response modifier
JP2007517035A (en) 2003-12-29 2007-06-28 スリーエム イノベイティブ プロパティズ カンパニー Arylalkenyl and arylalkynyl substituted imidazoquinoline
US8735421B2 (en) 2003-12-30 2014-05-27 3M Innovative Properties Company Imidazoquinolinyl sulfonamides
WO2005094531A2 (en) 2004-03-24 2005-10-13 3M Innovative Properties Company Amide substituted imidazopyridines, imidazoquinolines, and imidazonaphthyridines
US8017779B2 (en) 2004-06-15 2011-09-13 3M Innovative Properties Company Nitrogen containing heterocyclyl substituted imidazoquinolines and imidazonaphthyridines
US8026366B2 (en) 2004-06-18 2011-09-27 3M Innovative Properties Company Aryloxy and arylalkyleneoxy substituted thiazoloquinolines and thiazolonaphthyridines
WO2006038923A2 (en) 2004-06-18 2006-04-13 3M Innovative Properties Company Aryl substituted imidazonaphthyridines
WO2006065280A2 (en) 2004-06-18 2006-06-22 3M Innovative Properties Company Isoxazole, dihydroisoxazole, and oxadiazole substituted imidazo ring compounds and methods
AU2005326708C1 (en) 2004-12-30 2012-08-30 3M Innovative Properties Company Substituted chiral fused [1,2]imidazo[4,5-c] ring compounds
US7943609B2 (en) 2004-12-30 2011-05-17 3M Innovative Proprerties Company Chiral fused [1,2]imidazo[4,5-C] ring compounds
AU2006210392A1 (en) 2005-02-04 2006-08-10 Coley Pharmaceutical Group, Inc. Aqueous gel formulations containing immune response modifiers
JP2008530113A (en) 2005-02-11 2008-08-07 コーリー ファーマシューティカル グループ,インコーポレイテッド Oxime and hydroxylamine-substituted imidazo [4,5-c] ring compounds and methods
WO2006107851A1 (en) 2005-04-01 2006-10-12 Coley Pharmaceutical Group, Inc. 1-substituted pyrazolo (3,4-c) ring compounds as modulators of cytokine biosynthesis for the treatment of viral infections and neoplastic diseases
US7943610B2 (en) 2005-04-01 2011-05-17 3M Innovative Properties Company Pyrazolopyridine-1,4-diamines and analogs thereof
JP4551962B2 (en) * 2005-09-23 2010-09-29 コーリー ファーマシューティカル グループ,インコーポレイテッド Method for 1H- imidazo [4,5-c] pyridine and its analogues
WO2008008432A2 (en) 2006-07-12 2008-01-17 Coley Pharmaceutical Group, Inc. Substituted chiral fused( 1,2) imidazo (4,5-c) ring compounds and methods
US8461328B2 (en) * 2010-01-12 2013-06-11 Genentech, Inc. Tricyclic heterocyclic compounds, compositions and methods of use thereof
CN105940002B (en) 2014-02-03 2018-09-25 生命医药公司 ROR-γ-dihydro-pyrrole and pyridine inhibitor
MX2017004906A (en) 2014-10-14 2017-12-07 Vitae Pharmaceuticals Inc Dihydropyrrolopyridine inhibitors of ror-gamma.
US9845308B2 (en) 2014-11-05 2017-12-19 Vitae Pharmaceuticals, Inc. Isoindoline inhibitors of ROR-gamma
US9663515B2 (en) 2014-11-05 2017-05-30 Vitae Pharmaceuticals, Inc. Dihydropyrrolopyridine inhibitors of ROR-gamma
WO2017024018A1 (en) 2015-08-05 2017-02-09 Vitae Pharmaceuticals, Inc. Modulators of ror-gamma
US9481674B1 (en) 2016-06-10 2016-11-01 Vitae Pharmaceuticals, Inc. Dihydropyrrolopyridine inhibitors of ROR-gamma

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL157443B1 (en) * 1988-12-22 1992-05-29 Method for preparation of the new, n-phenylcarbamyle derivatives of difurylethane and difurylvinylchloride
US5378848A (en) 1992-02-12 1995-01-03 Shionogi & Co., Ltd. Condensed imidazopyridine derivatives
IL151877D0 (en) * 2000-03-30 2003-04-10 Shionogi & Co A process for producing imidazopyridine derivatives and a crystal form of an imidazopyridine derivative

Also Published As

Publication number Publication date
EP1408041A1 (en) 2004-04-14
US20040167157A1 (en) 2004-08-26
WO2003008421A1 (en) 2003-01-30
CN1250550C (en) 2006-04-12
JPWO2003008421A1 (en) 2004-11-11
CN1555378A (en) 2004-12-15
MXPA04000449A (en) 2004-03-18
KR20040027878A (en) 2004-04-01
EP1408041A4 (en) 2005-08-17
US6987187B2 (en) 2006-01-17
CA2453664A1 (en) 2003-01-30

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired