BG61975B1 - Индолови производни, методи и междинни съединения за тяхнотополучаване, фармацевтични състави, които ги съдържат, иприложението им - Google Patents

Индолови производни, методи и междинни съединения за тяхнотополучаване, фармацевтични състави, които ги съдържат, иприложението им Download PDF

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Publication number
BG61975B1
BG61975B1 BG97632A BG9763293A BG61975B1 BG 61975 B1 BG61975 B1 BG 61975B1 BG 97632 A BG97632 A BG 97632A BG 9763293 A BG9763293 A BG 9763293A BG 61975 B1 BG61975 B1 BG 61975B1
Authority
BG
Bulgaria
Prior art keywords
indole
ylmethyl
alkyl
aryl
hydrogen
Prior art date
Application number
BG97632A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG97632A (bg
Inventor
John E. Macor
Martin J. Wythes
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24393510&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG61975(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of BG97632A publication Critical patent/BG97632A/bg
Publication of BG61975B1 publication Critical patent/BG61975B1/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Addiction (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Lasers (AREA)
  • Electroluminescent Light Sources (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG97632A 1990-10-15 1993-04-14 Индолови производни, методи и междинни съединения за тяхнотополучаване, фармацевтични състави, които ги съдържат, иприложението им BG61975B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59792890A 1990-10-15 1990-10-15
PCT/US1991/007194 WO1992006973A1 (fr) 1990-10-15 1991-10-08 Derives d'indole

Publications (2)

Publication Number Publication Date
BG97632A BG97632A (bg) 1994-03-31
BG61975B1 true BG61975B1 (bg) 1998-11-30

Family

ID=24393510

Family Applications (1)

Application Number Title Priority Date Filing Date
BG97632A BG61975B1 (bg) 1990-10-15 1993-04-14 Индолови производни, методи и междинни съединения за тяхнотополучаване, фармацевтични състави, които ги съдържат, иприложението им

Country Status (33)

Country Link
EP (1) EP0592438B1 (fr)
JP (2) JP2575272B2 (fr)
KR (1) KR0179053B1 (fr)
CN (1) CN1039322C (fr)
AT (1) ATE157361T1 (fr)
AU (1) AU651637B2 (fr)
BG (1) BG61975B1 (fr)
BR (2) BR9106978A (fr)
CA (1) CA2091562C (fr)
DE (3) DE10299004I2 (fr)
DK (1) DK0592438T5 (fr)
EG (1) EG20224A (fr)
ES (1) ES2104733T3 (fr)
FI (1) FI105812B (fr)
GR (1) GR3025087T3 (fr)
HU (2) HUT64326A (fr)
IE (1) IE913555A1 (fr)
IL (3) IL115117A (fr)
LU (1) LU90902I2 (fr)
MX (1) MX9101606A (fr)
MY (1) MY111683A (fr)
NL (1) NL300070I2 (fr)
NO (3) NO305121B1 (fr)
NZ (2) NZ240217A (fr)
OA (1) OA09874A (fr)
PL (3) PL169987B1 (fr)
PT (1) PT99218B (fr)
RO (1) RO111767B1 (fr)
RU (1) RU2095360C1 (fr)
SG (1) SG54270A1 (fr)
WO (1) WO1992006973A1 (fr)
YU (1) YU48088B (fr)
ZA (1) ZA918156B (fr)

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ATE170836T1 (de) * 1993-08-31 1998-09-15 Pfizer 5-arylindolderivate
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Also Published As

Publication number Publication date
CA2091562A1 (fr) 1992-04-16
DK0592438T5 (da) 1999-12-06
HUT64326A (en) 1993-12-28
YU165391A (sh) 1994-01-20
PL168919B1 (pl) 1996-05-31
PT99218A (pt) 1992-09-30
DE10299004I1 (de) 2002-05-08
BG97632A (bg) 1994-03-31
NO2001019I1 (no) 2001-12-03
IL99701A0 (en) 1992-08-18
EP0592438B1 (fr) 1997-08-27
PT99218B (pt) 1999-04-30
RO111767B1 (ro) 1997-01-30
HU225055B1 (en) 2006-05-29
IL115117A (en) 1996-11-14
EP0592438A1 (fr) 1994-04-20
CN1062529A (zh) 1992-07-08
JPH093063A (ja) 1997-01-07
FI931667A0 (fi) 1993-04-14
GR3025087T3 (en) 1998-01-30
DE69127468D1 (de) 1997-10-02
AU8950491A (en) 1992-05-20
JPH05507288A (ja) 1993-10-21
ES2104733T3 (es) 1997-10-16
NZ240217A (en) 1995-05-26
DK0592438T3 (da) 1997-09-29
CA2091562C (fr) 2001-03-27
MY111683A (en) 2000-11-30
MX9101606A (es) 1992-06-05
WO1992006973A1 (fr) 1992-04-30
ATE157361T1 (de) 1997-09-15
JP2575272B2 (ja) 1997-01-22
EG20224A (en) 1997-12-31
PL169987B1 (en) 1996-09-30
FI931667A (fi) 1993-04-14
NL300070I2 (nl) 2002-03-01
HU9301098D0 (en) 1993-07-28
NO985607D0 (no) 1998-12-01
SG54270A1 (en) 1998-11-16
BR9106978A (pt) 1993-09-28
IL99701A (en) 1996-10-31
YU48088B (sh) 1997-01-08
IE913555A1 (en) 1992-04-22
RU2095360C1 (ru) 1997-11-10
CN1039322C (zh) 1998-07-29
PL170330B1 (pl) 1996-11-29
JP2677777B2 (ja) 1997-11-17
KR0179053B1 (ko) 1999-03-20
DE69127468T2 (de) 1998-01-02
NO931378L (no) 1993-04-14
ZA918156B (en) 1993-04-14
IL115117A0 (en) 1995-12-08
NL300070I1 (nl) 2002-02-01
DE10299004I2 (de) 2006-03-16
NO931378D0 (no) 1993-04-14
FI105812B (fi) 2000-10-13
LU90902I2 (fr) 2002-06-26
AU651637B2 (en) 1994-07-28
BR1100080A (pt) 2000-06-06
NO985607L (no) 1998-12-01
DE9190141U1 (de) 1993-07-15
OA09874A (en) 1994-09-15
NZ270675A (en) 1997-07-27
NO305121B1 (no) 1999-04-06

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